IL141239A0 - Alkynyl-substituted quinolin-2-one derivatives useful as anticancer agents - Google Patents

Alkynyl-substituted quinolin-2-one derivatives useful as anticancer agents

Info

Publication number
IL141239A0
IL141239A0 IL14123999A IL14123999A IL141239A0 IL 141239 A0 IL141239 A0 IL 141239A0 IL 14123999 A IL14123999 A IL 14123999A IL 14123999 A IL14123999 A IL 14123999A IL 141239 A0 IL141239 A0 IL 141239A0
Authority
IL
Israel
Prior art keywords
alkynyl
anticancer agents
derivatives useful
substituted quinolin
quinolin
Prior art date
Application number
IL14123999A
Other languages
English (en)
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of IL141239A0 publication Critical patent/IL141239A0/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/10—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing aromatic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/06—Antipsoriatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
    • C07F7/02—Silicon compounds
    • C07F7/08—Compounds having one or more C—Si linkages
    • C07F7/18—Compounds having one or more C—Si linkages as well as one or more C—O—Si linkages
    • C07F7/1804—Compounds having Si-O-C linkages

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Dermatology (AREA)
  • Urology & Nephrology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
IL14123999A 1998-08-27 1999-08-06 Alkynyl-substituted quinolin-2-one derivatives useful as anticancer agents IL141239A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US9814598P 1998-08-27 1998-08-27
PCT/IB1999/001398 WO2000012499A1 (en) 1998-08-27 1999-08-06 Alkynyl-substituted quinolin-2-one derivatives useful as anticancer agents

Publications (1)

Publication Number Publication Date
IL141239A0 true IL141239A0 (en) 2002-03-10

Family

ID=22267481

Family Applications (1)

Application Number Title Priority Date Filing Date
IL14123999A IL141239A0 (en) 1998-08-27 1999-08-06 Alkynyl-substituted quinolin-2-one derivatives useful as anticancer agents

Country Status (40)

Country Link
US (3) US6150377A (sk)
EP (1) EP1107963B1 (sk)
JP (1) JP3495706B2 (sk)
KR (1) KR20010072991A (sk)
CN (1) CN1314904A (sk)
AP (1) AP2001002079A0 (sk)
AT (1) ATE321037T1 (sk)
AU (1) AU4925499A (sk)
BG (1) BG105365A (sk)
BR (1) BRPI9913138B8 (sk)
CA (2) CA2341690C (sk)
CO (1) CO5130017A1 (sk)
CZ (1) CZ2001660A3 (sk)
DE (1) DE69930518T2 (sk)
DZ (1) DZ2880A1 (sk)
EA (1) EA200100135A1 (sk)
EE (1) EE200100118A (sk)
ES (1) ES2259237T3 (sk)
GE (1) GEP20033001B (sk)
GT (1) GT199900140A (sk)
HK (1) HK1039123A1 (sk)
HR (1) HRP20010142A2 (sk)
HU (1) HUP0103228A3 (sk)
ID (1) ID27562A (sk)
IL (1) IL141239A0 (sk)
IS (1) IS5818A (sk)
MA (1) MA26680A1 (sk)
NO (1) NO20010964L (sk)
NZ (1) NZ509372A (sk)
OA (1) OA11645A (sk)
PA (1) PA8480101A1 (sk)
PE (1) PE20000986A1 (sk)
PL (1) PL346426A1 (sk)
SK (1) SK2442001A3 (sk)
SV (1) SV1999000141A (sk)
TN (1) TNSN99162A1 (sk)
TR (1) TR200101343T2 (sk)
UY (1) UY25682A1 (sk)
WO (1) WO2000012499A1 (sk)
ZA (1) ZA200101173B (sk)

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DE69923849T2 (de) * 1998-08-27 2006-01-12 Pfizer Products Inc., Groton Quinolin-2-on-derivate verwendbar als antikrebsmittel
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CN1340051A (zh) 1999-02-11 2002-03-13 辉瑞产品公司 可用作抗癌剂的杂芳基取代的喹啉－2－酮衍生物
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Also Published As

Publication number Publication date
US6294552B1 (en) 2001-09-25
TR200101343T2 (tr) 2001-09-21
HK1039123A1 (zh) 2002-04-12
CO5130017A1 (es) 2002-02-27
EA200100135A1 (ru) 2001-08-27
EP1107963B1 (en) 2006-03-22
EE200100118A (et) 2002-06-17
GEP20033001B (en) 2003-06-25
HRP20010142A2 (en) 2002-02-28
TNSN99162A1 (fr) 2005-11-10
HUP0103228A2 (hu) 2002-02-28
NO20010964D0 (no) 2001-02-26
NO20010964L (no) 2001-04-26
PA8480101A1 (es) 2003-06-30
UY25682A1 (es) 2000-03-31
DZ2880A1 (fr) 2003-12-15
BG105365A (en) 2001-11-30
CA2341690C (en) 2007-04-17
US6579887B2 (en) 2003-06-17
BR9913138B1 (pt) 2013-11-05
CN1314904A (zh) 2001-09-26
OA11645A (en) 2004-11-16
AU4925499A (en) 2000-03-21
JP3495706B2 (ja) 2004-02-09
GT199900140A (es) 2001-02-14
PE20000986A1 (es) 2000-09-30
US20020128287A1 (en) 2002-09-12
ES2259237T3 (es) 2006-09-16
JP2002523504A (ja) 2002-07-30
KR20010072991A (ko) 2001-07-31
ID27562A (id) 2001-04-12
CZ2001660A3 (cs) 2002-05-15
DE69930518T2 (de) 2006-09-21
CA2341690A1 (en) 2000-03-09
BR9913138A (pt) 2001-05-08
SV1999000141A (es) 2000-07-06
CA2578326C (en) 2009-11-24
SK2442001A3 (en) 2002-10-08
US6150377A (en) 2000-11-21
HUP0103228A3 (en) 2003-01-28
EP1107963A1 (en) 2001-06-20
NZ509372A (en) 2003-08-29
WO2000012499A1 (en) 2000-03-09
DE69930518D1 (de) 2006-05-11
AP2001002079A0 (en) 2001-03-31
ZA200101173B (en) 2002-04-12
ATE321037T1 (de) 2006-04-15
CA2578326A1 (en) 2000-03-09
IS5818A (is) 2001-01-19
MA26680A1 (fr) 2004-12-20
BRPI9913138B8 (pt) 2016-05-17
PL346426A1 (en) 2002-02-11

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