MA26680A1 - Derives de quinoleine-2-one a substituant alcynyle nouveaux, procede pour leur preparation et compositions pharmaceutiques les contenant - Google Patents

Derives de quinoleine-2-one a substituant alcynyle nouveaux, procede pour leur preparation et compositions pharmaceutiques les contenant

Info

Publication number
MA26680A1
MA26680A1 MA25743A MA25743A MA26680A1 MA 26680 A1 MA26680 A1 MA 26680A1 MA 25743 A MA25743 A MA 25743A MA 25743 A MA25743 A MA 25743A MA 26680 A1 MA26680 A1 MA 26680A1
Authority
MA
Morocco
Prior art keywords
alcynyl
quinolein
substitute
derivatives
preparation
Prior art date
Application number
MA25743A
Other languages
English (en)
Inventor
Deborah La Greca Susan
Peter Lyssikatos Joseph
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of MA26680A1 publication Critical patent/MA26680A1/fr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/10Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing aromatic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/06Antipsoriatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F7/00Compounds containing elements of Groups 4 or 14 of the Periodic System
    • C07F7/02Silicon compounds
    • C07F7/08Compounds having one or more C—Si linkages
    • C07F7/18Compounds having one or more C—Si linkages as well as one or more C—O—Si linkages
    • C07F7/1804Compounds having Si-O-C linkages
MA25743A 1998-08-27 1999-08-25 Derives de quinoleine-2-one a substituant alcynyle nouveaux, procede pour leur preparation et compositions pharmaceutiques les contenant MA26680A1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US9814598P 1998-08-27 1998-08-27

Publications (1)

Publication Number Publication Date
MA26680A1 true MA26680A1 (fr) 2004-12-20

Family

ID=22267481

Family Applications (1)

Application Number Title Priority Date Filing Date
MA25743A MA26680A1 (fr) 1998-08-27 1999-08-25 Derives de quinoleine-2-one a substituant alcynyle nouveaux, procede pour leur preparation et compositions pharmaceutiques les contenant

Country Status (40)

Country Link
US (3) US6150377A (fr)
EP (1) EP1107963B1 (fr)
JP (1) JP3495706B2 (fr)
KR (1) KR20010072991A (fr)
CN (1) CN1314904A (fr)
AP (1) AP2001002079A0 (fr)
AT (1) ATE321037T1 (fr)
AU (1) AU4925499A (fr)
BG (1) BG105365A (fr)
BR (1) BRPI9913138B8 (fr)
CA (2) CA2578326C (fr)
CO (1) CO5130017A1 (fr)
CZ (1) CZ2001660A3 (fr)
DE (1) DE69930518T2 (fr)
DZ (1) DZ2880A1 (fr)
EA (1) EA200100135A1 (fr)
EE (1) EE200100118A (fr)
ES (1) ES2259237T3 (fr)
GE (1) GEP20033001B (fr)
GT (1) GT199900140A (fr)
HK (1) HK1039123A1 (fr)
HR (1) HRP20010142A2 (fr)
HU (1) HUP0103228A3 (fr)
ID (1) ID27562A (fr)
IL (1) IL141239A0 (fr)
IS (1) IS5818A (fr)
MA (1) MA26680A1 (fr)
NO (1) NO20010964L (fr)
NZ (1) NZ509372A (fr)
OA (1) OA11645A (fr)
PA (1) PA8480101A1 (fr)
PE (1) PE20000986A1 (fr)
PL (1) PL346426A1 (fr)
SK (1) SK2442001A3 (fr)
SV (1) SV1999000141A (fr)
TN (1) TNSN99162A1 (fr)
TR (1) TR200101343T2 (fr)
UY (1) UY25682A1 (fr)
WO (1) WO2000012499A1 (fr)
ZA (1) ZA200101173B (fr)

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EA200100766A1 (ru) 1999-02-11 2002-02-28 Пфайзер Продактс Инк. Хинолин-2-он замещенные гетероарильные производные, используемые в качестве противоопухолевых агентов
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DE60130976T2 (de) 2000-02-24 2008-07-17 Janssen Pharmaceutica N.V. Dosierschema enthaldend farnesyl protein transferase inhibitoren für die behandlung von krebs
JO2361B1 (en) 2000-06-22 2006-12-12 جانسين فارماسيوتيكا ان. في Enaniumer 1,2-anylated quinoline inhibitor for the transporter - farnesyl
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WO2002024683A1 (fr) 2000-09-25 2002-03-28 Janssen Pharmaceutica N.V. Derives de la quinoleine et de la quinazoline 6-[(phenyle substitue)methyle] inhibiteurs de la farnesyle transferase
AU2001293835A1 (en) * 2000-09-25 2002-04-02 Janssen Pharmaceutica N.V. Farnesyl transferase inhibiting 6-heterocyclylmethyl quinolinone derivatives
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MXPA03005525A (es) 2000-12-19 2003-10-06 Pfizer Prod Inc Formas cristalinas de sales de 2,3-dihidroxibutanodioato de 6-[(4-cloro -fenil)- hidroxi-(3 -metil-3h-imidazol -4-il)-metil] -4-(3-etinil-fenil) -1-metil-1h -quinolein-2 -ona, y metodo de produccion.
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Also Published As

Publication number Publication date
UY25682A1 (es) 2000-03-31
NO20010964L (no) 2001-04-26
CO5130017A1 (es) 2002-02-27
EA200100135A1 (ru) 2001-08-27
NO20010964D0 (no) 2001-02-26
DZ2880A1 (fr) 2003-12-15
HRP20010142A2 (en) 2002-02-28
CA2341690A1 (fr) 2000-03-09
ZA200101173B (en) 2002-04-12
US20020128287A1 (en) 2002-09-12
BG105365A (en) 2001-11-30
SK2442001A3 (en) 2002-10-08
SV1999000141A (es) 2000-07-06
ATE321037T1 (de) 2006-04-15
CN1314904A (zh) 2001-09-26
HUP0103228A3 (en) 2003-01-28
BR9913138B1 (pt) 2013-11-05
AP2001002079A0 (en) 2001-03-31
AU4925499A (en) 2000-03-21
BRPI9913138B8 (pt) 2016-05-17
EP1107963A1 (fr) 2001-06-20
NZ509372A (en) 2003-08-29
US6579887B2 (en) 2003-06-17
GT199900140A (es) 2001-02-14
EE200100118A (et) 2002-06-17
IL141239A0 (en) 2002-03-10
PE20000986A1 (es) 2000-09-30
KR20010072991A (ko) 2001-07-31
TR200101343T2 (tr) 2001-09-21
DE69930518D1 (de) 2006-05-11
US6150377A (en) 2000-11-21
TNSN99162A1 (fr) 2005-11-10
BR9913138A (pt) 2001-05-08
HUP0103228A2 (hu) 2002-02-28
ES2259237T3 (es) 2006-09-16
OA11645A (en) 2004-11-16
CA2578326C (fr) 2009-11-24
ID27562A (id) 2001-04-12
DE69930518T2 (de) 2006-09-21
EP1107963B1 (fr) 2006-03-22
CZ2001660A3 (cs) 2002-05-15
PL346426A1 (en) 2002-02-11
WO2000012499A1 (fr) 2000-03-09
PA8480101A1 (es) 2003-06-30
JP2002523504A (ja) 2002-07-30
IS5818A (is) 2001-01-19
HK1039123A1 (zh) 2002-04-12
JP3495706B2 (ja) 2004-02-09
CA2578326A1 (fr) 2000-03-09
GEP20033001B (en) 2003-06-25
US6294552B1 (en) 2001-09-25
CA2341690C (fr) 2007-04-17

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