IL130716A - (-) E - 2 (-4,3 dichlorocinamyl) - 1 cyclopropylmethyl-piperidine and its use in the preparation of anti-diarrheal preparations - Google Patents

(-) E - 2 (-4,3 dichlorocinamyl) - 1 cyclopropylmethyl-piperidine and its use in the preparation of anti-diarrheal preparations

Info

Publication number
IL130716A
IL130716A IL13071698A IL13071698A IL130716A IL 130716 A IL130716 A IL 130716A IL 13071698 A IL13071698 A IL 13071698A IL 13071698 A IL13071698 A IL 13071698A IL 130716 A IL130716 A IL 130716A
Authority
IL
Israel
Prior art keywords
dichlorocinnamyl
piperidine
preparation
cyclopropylmethylpiperidine
compound
Prior art date
Application number
IL13071698A
Other languages
English (en)
Hebrew (he)
Other versions
IL130716A0 (en
Original Assignee
Parke Davis
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Parke Davis filed Critical Parke Davis
Publication of IL130716A0 publication Critical patent/IL130716A0/xx
Publication of IL130716A publication Critical patent/IL130716A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D211/00Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/08Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
    • C07D211/18Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/12Antidiarrhoeals

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
IL13071698A 1997-03-05 1998-03-04 (-) E - 2 (-4,3 dichlorocinamyl) - 1 cyclopropylmethyl-piperidine and its use in the preparation of anti-diarrheal preparations IL130716A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR9702713A FR2760455B1 (fr) 1997-03-05 1997-03-05 (-)e-2-(3,4-dichloro-cinnamyl)-1-cyclopropylmethyl- piperidine, son utilite antidiarrheique
PCT/EP1998/001564 WO1998039296A1 (fr) 1997-03-05 1998-03-04 (-)e-2-(3,4-dichlorocinnamyl)-1-cyclopropylmethyl-piperidine et son utilisation comme antidiarrheique

Publications (2)

Publication Number Publication Date
IL130716A0 IL130716A0 (en) 2000-06-01
IL130716A true IL130716A (en) 2004-02-19

Family

ID=9504511

Family Applications (1)

Application Number Title Priority Date Filing Date
IL13071698A IL130716A (en) 1997-03-05 1998-03-04 (-) E - 2 (-4,3 dichlorocinamyl) - 1 cyclopropylmethyl-piperidine and its use in the preparation of anti-diarrheal preparations

Country Status (12)

Country Link
US (1) US6440997B2 (fr)
EP (1) EP0968187A1 (fr)
JP (1) JP2001513802A (fr)
KR (1) KR20000075973A (fr)
AU (1) AU749902B2 (fr)
BR (1) BR9808823A (fr)
CA (1) CA2277839A1 (fr)
FR (1) FR2760455B1 (fr)
IL (1) IL130716A (fr)
NZ (1) NZ336575A (fr)
WO (1) WO1998039296A1 (fr)
ZA (1) ZA981849B (fr)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1138327A1 (fr) * 2000-03-29 2001-10-04 Warner-Lambert Company Utilisation de dérivés 2-(arylalkenyl)azacycloalkanes pour traiter les désordres gastrointestinaux liés au stress
FR2833945B1 (fr) * 2001-12-21 2004-03-12 Warner Lambert Co N-cyclopropylmethyl-azacycloalcanes, compositions les contenant et procedes de preparation

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5849760A (en) * 1993-12-09 1998-12-15 Institut De Recherche Jouveinal 2-(arylalkenyl)azacycloalkane derivatives as ligands for sigma receptors

Also Published As

Publication number Publication date
CA2277839A1 (fr) 1998-09-11
FR2760455B1 (fr) 1999-04-16
AU7036798A (en) 1998-09-22
EP0968187A1 (fr) 2000-01-05
BR9808823A (pt) 2000-07-04
US6440997B2 (en) 2002-08-27
AU749902B2 (en) 2002-07-04
NZ336575A (en) 2001-10-26
WO1998039296A1 (fr) 1998-09-11
IL130716A0 (en) 2000-06-01
JP2001513802A (ja) 2001-09-04
US20010008897A1 (en) 2001-07-19
KR20000075973A (ko) 2000-12-26
FR2760455A1 (fr) 1998-09-11
ZA981849B (en) 1998-09-01

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Legal Events

Date Code Title Description
FF Patent granted
MM9K Patent not in force due to non-payment of renewal fees
MM9K Patent not in force due to non-payment of renewal fees