IL121625A - תכשיר המכיל 2 - אמינו - 2 - (-2 (-4 אוקטילפניל) אתיל) פרופן - 1, 3, - דיול לשימוש מקומי חיצוני - Google Patents
תכשיר המכיל 2 - אמינו - 2 - (-2 (-4 אוקטילפניל) אתיל) פרופן - 1, 3, - דיול לשימוש מקומי חיצוניInfo
- Publication number
- IL121625A IL121625A IL12162596A IL12162596A IL121625A IL 121625 A IL121625 A IL 121625A IL 12162596 A IL12162596 A IL 12162596A IL 12162596 A IL12162596 A IL 12162596A IL 121625 A IL121625 A IL 121625A
- Authority
- IL
- Israel
- Prior art keywords
- compound
- present
- external preparation
- ointment
- acid
- Prior art date
Links
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
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- Health & Medical Sciences (AREA)
- Public Health (AREA)
- Immunology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Emergency Medicine (AREA)
- Epidemiology (AREA)
- Pulmonology (AREA)
- Transplantation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicinal Preparation (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP34250395 | 1995-12-28 | ||
| PCT/JP1996/003757 WO1997024112A1 (fr) | 1995-12-28 | 1996-12-24 | Preparation a usage externe |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| IL121625A0 IL121625A0 (en) | 1998-02-08 |
| IL121625A true IL121625A (he) | 2001-09-13 |
Family
ID=18354257
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IL12162596A IL121625A (he) | 1995-12-28 | 1996-12-24 | תכשיר המכיל 2 - אמינו - 2 - (-2 (-4 אוקטילפניל) אתיל) פרופן - 1, 3, - דיול לשימוש מקומי חיצוני |
Country Status (16)
| Country | Link |
|---|---|
| US (2) | US6121329A (he) |
| EP (1) | EP0812588B1 (he) |
| AT (1) | ATE279185T1 (he) |
| AU (1) | AU705320B2 (he) |
| CA (1) | CA2213989C (he) |
| CZ (1) | CZ285953B6 (he) |
| DE (1) | DE69633613T2 (he) |
| ES (1) | ES2230571T3 (he) |
| HU (1) | HU224814B1 (he) |
| IL (1) | IL121625A (he) |
| NZ (1) | NZ324453A (he) |
| PT (1) | PT812588E (he) |
| RU (1) | RU2156127C2 (he) |
| SI (1) | SI0812588T1 (he) |
| SK (1) | SK282225B6 (he) |
| WO (1) | WO1997024112A1 (he) |
Families Citing this family (60)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6476004B1 (en) | 1996-07-18 | 2002-11-05 | Mitsubishi Pharma Corporation | Pharmaceutical composition |
| JP2002241272A (ja) * | 1996-07-18 | 2002-08-28 | Mitsubishi Pharma Corp | 医薬処方組成物 |
| GB9624038D0 (en) | 1996-11-19 | 1997-01-08 | Sandoz Ltd | Organic compounds |
| SI0990440T1 (sl) * | 1997-02-27 | 2009-04-30 | Novartis Ag | Farmacevtski sestavek, ki obsega 2-amino-2-(2-(4-oktilfenil)etil)propan-1,3-diol, lecitin in saharid |
| KR100406823B1 (ko) | 1998-04-27 | 2003-11-21 | 후지사와 야꾸힝 고교 가부시키가이샤 | 의약 조성물 |
| US20020006901A1 (en) * | 1999-02-05 | 2002-01-17 | Aldo T. Iacono | Use of aerosolized cyclosporine for prevention and treatment of pulmonary disease |
| US7683044B2 (en) * | 1999-03-25 | 2010-03-23 | Center For Molecular Medicine And Immunology | Sphingomyelin therapy of autoimmune disease |
| EP1165137B1 (en) * | 1999-03-25 | 2006-08-02 | Center For Molecular Medicine And Immunology | Sphingomyelin containing preparation for the enhancement of tumor therapy |
| JP2004507552A (ja) | 2000-08-31 | 2004-03-11 | メルク エンド カムパニー インコーポレーテッド | 免疫調節剤としてのリン酸誘導体 |
| JP4318921B2 (ja) * | 2001-02-22 | 2009-08-26 | ノバルティス アクチエンゲゼルシャフト | 移植片の機能発現遅延の処置のための医薬の製造のためのリンパ球ホーミング促進剤の使用 |
| US20030124174A1 (en) * | 2001-10-25 | 2003-07-03 | Endo Pharmaceuticals, Inc | Method for treating non-neuropathic pain |
| KR100836547B1 (ko) * | 2002-01-11 | 2008-06-10 | 상꾜 가부시키가이샤 | 아미노 알코올 유도체 또는 포스폰산 유도체 및 이들을함유하는 의약 조성물 |
| AU2003233119A1 (en) | 2002-05-08 | 2003-11-11 | Neuronova Ab | Modulation of neural stem cells with s1p or lpa receptor agonists |
| KR20120035220A (ko) * | 2003-01-22 | 2012-04-13 | 센주 세이야꾸 가부시키가이샤 | 안질환 치료용 경피 흡수형 제제, 그 사용, 및 안질환 치료약의 눈의 국소 조직으로의 이행 방법 |
| GB0307866D0 (en) * | 2003-04-04 | 2003-05-14 | Novartis Ag | Pharmaceutical composition |
| HUE028247T2 (en) | 2003-04-08 | 2016-12-28 | Novartis Ag | A solid oral composition comprising S1P receptor agonist and sugar alcohol |
| US7524887B2 (en) | 2003-06-06 | 2009-04-28 | Sanofi-Aventis Deutschland Gmbh | 2-amino-1,3-propanediol compounds for the treatment of acute pain |
| EP1484057A1 (en) * | 2003-06-06 | 2004-12-08 | Aventis Pharma Deutschland GmbH | Use of 2-amino-1-3-propanediol derivatives for the manufacture of a medicament for the treatment of various types of pain |
| BRPI0414193A (pt) * | 2003-09-09 | 2006-10-31 | 3M Innovative Properties Co | composição antimicrobiana, kit antimicrobiano e métodos de usar a composição e de aplicar uma composição antimicrobiana a um substrato |
| US20050058673A1 (en) | 2003-09-09 | 2005-03-17 | 3M Innovative Properties Company | Antimicrobial compositions and methods |
| GB0324210D0 (en) * | 2003-10-15 | 2003-11-19 | Novartis Ag | Organic compounds |
| GB0329498D0 (en) * | 2003-12-19 | 2004-01-28 | Novartis Ag | Organic compounds |
| GB0500020D0 (en) * | 2005-01-04 | 2005-02-09 | Novartis Ag | Organic compounds |
| RU2332212C2 (ru) | 2004-02-24 | 2008-08-27 | Санкио Компани, Лимитед | Аминоспирт |
| US20050232894A1 (en) * | 2004-04-20 | 2005-10-20 | Weiner Gregory M | Antimicrobial skin treatment composition and methods for producing and using an antimicrobial skin treatment composition |
| PT1773307E (pt) * | 2004-07-30 | 2015-01-14 | Novartis Ag | Formulações de compostos à base de 2-amino-1,3- propanodiol |
| US8313763B2 (en) * | 2004-10-04 | 2012-11-20 | Tolmar Therapeutics, Inc. | Sustained delivery formulations of rapamycin compounds |
| CA2582374A1 (en) * | 2004-10-04 | 2006-04-20 | Qlt Usa, Inc. | Ocular delivery of polymeric delivery formulations |
| MX2007006373A (es) * | 2004-11-29 | 2007-06-20 | Novartis Ag | Regimen de dosificacion de un agonista del receptor s1p. |
| US20080233053A1 (en) * | 2005-02-07 | 2008-09-25 | Pharmalight Inc. | Method and Device for Ophthalmic Administration of Active Pharmaceutical Ingredients |
| GB0504544D0 (en) * | 2005-03-04 | 2005-04-13 | Novartis Ag | Organic compounds |
| JP2008533048A (ja) | 2005-03-10 | 2008-08-21 | スリーエム イノベイティブ プロパティズ カンパニー | 耳の感染症の治療方法 |
| MX2007010908A (es) | 2005-03-10 | 2007-12-05 | 3M Innovative Properties Co | Composiciones antimicrobianas que comprenden esteres de acidos hidroxicarboxilicos. |
| US20060229364A1 (en) * | 2005-03-10 | 2006-10-12 | 3M Innovative Properties Company | Antiviral compositions and methods of use |
| KR20070113284A (ko) | 2005-03-10 | 2007-11-28 | 쓰리엠 이노베이티브 프로퍼티즈 캄파니 | 미생물 오염의 감소방법 |
| US8633161B2 (en) * | 2005-03-24 | 2014-01-21 | The Ohio State University Research Foundation | Therapeutic agents for the treatment of leukemia |
| US20080009545A1 (en) * | 2006-02-21 | 2008-01-10 | The Ohio State University Research Foundation | Anticancer agents |
| WO2007143081A2 (en) * | 2006-06-02 | 2007-12-13 | The Ohio State University Research Foundation | Therapeutic agents for the treatment of lymphoid malignancies |
| US20080075793A1 (en) * | 2006-09-21 | 2008-03-27 | Dunshee Wayne K | Antiviral compositions and methods of use |
| MY159358A (en) | 2007-10-12 | 2016-12-30 | Novartis Ag | Compositions comprising sphingosine 1 phosphate (s1p) receptor modulators |
| EP2278960B2 (en) | 2008-03-17 | 2019-11-13 | Actelion Pharmaceuticals Ltd. | Dosing regimen for a selective sip1 receptor agonist |
| AU2010236655A1 (en) * | 2009-04-13 | 2011-11-17 | The Ohio State University Research Foundation | Protein phosphatase 2A-activating agents |
| WO2010121111A1 (en) * | 2009-04-17 | 2010-10-21 | The Ohio State University Research Foundation | Antiadhesion agents |
| US8766005B2 (en) | 2009-07-24 | 2014-07-01 | Ratiopharm Gmbh | Process for producing fingolimod salts |
| CN101966145A (zh) * | 2010-09-21 | 2011-02-09 | 浙江大学 | 2-氨基-2-(2-[4-辛基苯基]乙基)-1,3-丙二醇盐酸盐制剂及其制备方法 |
| WO2012071524A1 (en) | 2010-11-24 | 2012-05-31 | Ratiopharm Gmbh | Arylsulfonate salts of fingolimod and processes for preparation thereof |
| US8309768B2 (en) | 2010-11-29 | 2012-11-13 | The Ohio State University Research Foundation | FTY720-derived anticancer agents |
| SG191286A1 (en) | 2011-01-07 | 2013-07-31 | Novartis Ag | Immunosuppressant formulations |
| AR085749A1 (es) | 2011-04-01 | 2013-10-23 | Novartis Ag | Formulaciones |
| RU2496486C1 (ru) | 2012-07-11 | 2013-10-27 | Александр Васильевич Иващенко | Фармацевтическая композиция с улучшенной сыпучестью, лекарственное средство, способ получения и применение |
| US10172789B2 (en) | 2013-01-24 | 2019-01-08 | Palvella Therapeutics Llc | Compositions for transdermal delivery of mTOR inhibitors |
| WO2015053879A1 (en) | 2013-10-11 | 2015-04-16 | Teikoku Pharma Usa, Inc. | Sphingosine-1-phosphate receptor agonist iontophoretic devices and methods of using the same |
| US10022340B2 (en) | 2013-10-11 | 2018-07-17 | Teikoku Pharma Usa, Inc. | Topical sphingosine-1-phosphate receptor agonist formulations and methods of using the same |
| US9925138B2 (en) | 2015-01-20 | 2018-03-27 | Handa Pharmaceuticals, Llc | Stable solid fingolimod dosage forms |
| CA2973540A1 (en) | 2015-02-26 | 2016-09-01 | Novartis Ag | Treatment of autoimmune disease in a patient receiving additionally a beta-blocker |
| WO2018129364A1 (en) | 2017-01-06 | 2018-07-12 | Palvella Therapeutics Llc | Anhydrous compositions of mtor inhibitors and methods of use |
| US10798783B2 (en) * | 2017-02-15 | 2020-10-06 | Continuous Composites Inc. | Additively manufactured composite heater |
| US11434200B2 (en) | 2017-03-09 | 2022-09-06 | Novartis Ag | Solid forms comprising an oxime ether compound and a coformer, compositions and methods of use thereof |
| SG11201911841PA (en) * | 2017-07-05 | 2020-01-30 | Jiangyin Mucocare Pharmaceutical Co Ltd | Topical formulations comprising montelukast and combinations with mussel adhesive proteins |
| JP2021530463A (ja) | 2018-07-02 | 2021-11-11 | パルヴェラ セラピューティクス、インク． | ｍＴＯＲ阻害剤の無水組成物および使用方法 |
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| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0356399A3 (en) * | 1988-08-26 | 1991-03-20 | Sandoz Ag | Substituted 4-azatricyclo (22.3.1.04.9) octacos-18-ene derivatives, their preparation and pharmaceutical compositions containing them |
| EP0501579A1 (en) * | 1991-02-28 | 1992-09-02 | Merck Frosst Canada Inc. | Naphthalene lactones as inhibitors of leukotriene biosynthesis |
| IL102236A0 (en) * | 1991-06-27 | 1993-01-14 | Ltt Inst Co Ltd | Topical preparations containing cyclosporin |
| IT1252865B (it) * | 1991-12-31 | 1995-06-28 | Lifegroup Spa | N-acilderivati di aminoalcooli attivi come autocoidi locali ed utilizzabili nella terapia dei processi autoimmuni |
| IT1252866B (it) * | 1991-12-31 | 1995-06-28 | Lifegroup Spa | N-acilderivati di aminoalcooli con acidi policarbossilici atti alla modulazione dei mastociti nei processi infiammatori su base neuroimmunogenica |
| DK0627406T3 (da) * | 1992-10-21 | 1999-07-12 | Taito Co | 2-Amino-1,3-propandiolforbindelser og immunundertrykkende midler |
| JPH06256182A (ja) * | 1993-03-05 | 1994-09-13 | L T T Kenkyusho:Kk | 外用製剤 |
| JPH07188046A (ja) * | 1993-12-27 | 1995-07-25 | L T T Kenkyusho:Kk | シクロスポリン含有外用治療薬及びその製造方法 |
| EP0694308A4 (en) * | 1994-02-17 | 1997-09-10 | Shiseido Co Ltd | CYCLOSPORIN EMULSION COMPOSITION |
| JPH1180026A (ja) * | 1997-09-02 | 1999-03-23 | Yoshitomi Pharmaceut Ind Ltd | 新規免疫抑制剤、その使用方法およびその同定方法 |
-
1996
- 1996-12-24 WO PCT/JP1996/003757 patent/WO1997024112A1/ja active IP Right Grant
- 1996-12-24 PT PT96942623T patent/PT812588E/pt unknown
- 1996-12-24 SK SK1157-97A patent/SK282225B6/sk not_active IP Right Cessation
- 1996-12-24 HU HU9800034A patent/HU224814B1/hu unknown
- 1996-12-24 EP EP96942623A patent/EP0812588B1/en not_active Expired - Lifetime
- 1996-12-24 AU AU11729/97A patent/AU705320B2/en not_active Expired
- 1996-12-24 US US08/894,728 patent/US6121329A/en not_active Expired - Lifetime
- 1996-12-24 NZ NZ324453A patent/NZ324453A/xx not_active IP Right Cessation
- 1996-12-24 IL IL12162596A patent/IL121625A/he not_active IP Right Cessation
- 1996-12-24 CZ CZ972704A patent/CZ285953B6/cs not_active IP Right Cessation
- 1996-12-24 SI SI9630694T patent/SI0812588T1/xx unknown
- 1996-12-24 DE DE69633613T patent/DE69633613T2/de not_active Expired - Lifetime
- 1996-12-24 CA CA002213989A patent/CA2213989C/en not_active Expired - Lifetime
- 1996-12-24 AT AT96942623T patent/ATE279185T1/de active
- 1996-12-24 RU RU97115893/14A patent/RU2156127C2/ru active
- 1996-12-24 ES ES96942623T patent/ES2230571T3/es not_active Expired - Lifetime
-
2000
- 2000-06-12 US US09/592,550 patent/US6197829B1/en not_active Expired - Lifetime
Also Published As
| Publication number | Publication date |
|---|---|
| NZ324453A (en) | 2000-03-27 |
| ES2230571T3 (es) | 2005-05-01 |
| AU1172997A (en) | 1997-07-28 |
| HUP9800034A2 (hu) | 1999-05-28 |
| SK115797A3 (en) | 1998-02-04 |
| EP0812588A1 (en) | 1997-12-17 |
| RU2156127C2 (ru) | 2000-09-20 |
| US6197829B1 (en) | 2001-03-06 |
| WO1997024112A1 (fr) | 1997-07-10 |
| AU705320B2 (en) | 1999-05-20 |
| SK282225B6 (sk) | 2001-12-03 |
| CA2213989A1 (en) | 1997-07-10 |
| CZ270497A3 (cs) | 1998-01-14 |
| IL121625A0 (en) | 1998-02-08 |
| HUP9800034A3 (en) | 1999-12-28 |
| HU224814B1 (en) | 2006-02-28 |
| US6121329A (en) | 2000-09-19 |
| CA2213989C (en) | 2007-05-29 |
| PT812588E (pt) | 2005-01-31 |
| DE69633613D1 (de) | 2004-11-18 |
| CZ285953B6 (cs) | 1999-12-15 |
| ATE279185T1 (de) | 2004-10-15 |
| SI0812588T1 (en) | 2005-02-28 |
| EP0812588A4 (en) | 2002-11-06 |
| EP0812588B1 (en) | 2004-10-13 |
| DE69633613T2 (de) | 2006-02-09 |
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| EXP | Patent expired |