IE61989B1 - Pilocarpine derivatives - Google Patents

Pilocarpine derivatives

Info

Publication number
IE61989B1
IE61989B1 IE24488A IE24488A IE61989B1 IE 61989 B1 IE61989 B1 IE 61989B1 IE 24488 A IE24488 A IE 24488A IE 24488 A IE24488 A IE 24488A IE 61989 B1 IE61989 B1 IE 61989B1
Authority
IE
Ireland
Prior art keywords
compound
methyl
addition salt
formula
free base
Prior art date
Application number
IE24488A
Other languages
English (en)
Other versions
IE880244L (en
Inventor
Georg Bolliger
Rene Amstutz
Gideon Shapiro
Original Assignee
Sandoz Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sandoz Ltd filed Critical Sandoz Ltd
Publication of IE880244L publication Critical patent/IE880244L/en
Publication of IE61989B1 publication Critical patent/IE61989B1/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A61P27/06—Antiglaucoma agents or miotics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Ophthalmology & Optometry (AREA)
  • Psychiatry (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Hydrogenated Pyridines (AREA)
IE24488A 1987-01-31 1988-01-29 Pilocarpine derivatives IE61989B1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE3702940 1987-01-31

Publications (2)

Publication Number Publication Date
IE880244L IE880244L (en) 1988-07-31
IE61989B1 true IE61989B1 (en) 1994-12-14

Family

ID=6319976

Family Applications (1)

Application Number Title Priority Date Filing Date
IE24488A IE61989B1 (en) 1987-01-31 1988-01-29 Pilocarpine derivatives

Country Status (27)

Country Link
US (1) US4835174A (enExample)
JP (1) JPS63201185A (enExample)
KR (1) KR880009013A (enExample)
AT (1) AT395852B (enExample)
AU (1) AU607966B2 (enExample)
BE (1) BE1001005A3 (enExample)
CA (1) CA1327805C (enExample)
CH (1) CH675721A5 (enExample)
CS (1) CS411291A3 (enExample)
DK (1) DK46288A (enExample)
ES (1) ES2008421A6 (enExample)
FI (1) FI90080C (enExample)
FR (1) FR2610322B1 (enExample)
GB (1) GB2200910B (enExample)
GR (1) GR880100042A (enExample)
HU (1) HU204047B (enExample)
IE (1) IE61989B1 (enExample)
IL (1) IL85252A (enExample)
IT (1) IT1219827B (enExample)
LU (1) LU87122A1 (enExample)
MY (1) MY102415A (enExample)
NL (1) NL8800099A (enExample)
NZ (1) NZ223359A (enExample)
PH (1) PH24837A (enExample)
PT (1) PT86666B (enExample)
SE (1) SE466150B (enExample)
ZA (1) ZA88665B (enExample)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4882343A (en) * 1987-08-28 1989-11-21 G. D. Searle & Co. Biarylalkylimidazole derivatives as anti-depressants
US5861431A (en) * 1995-06-07 1999-01-19 Iotek, Inc. Incontinence treatment
BR112020009361A2 (pt) 2017-11-17 2020-10-13 Cellix Bio Private Limited composto de fórmula i, composição farmacêutica para tratar um distúrbio ocular ou complicações do mesmo, método de síntese de composto, método de tratamento de um distúrbio ocular ou complicações do mesmo em um indivíduo que precisa do mesmo e uso de um composto

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2457047A (en) * 1946-02-13 1948-12-21 Monsanto Chemicals 2-(2'-thenyl)-4, 5-dihydroimidazoles and process for making the same
GB1601310A (en) * 1978-05-23 1981-10-28 Lilly Industries Ltd Aryl hydantoins
JPS56131579A (en) * 1980-03-17 1981-10-15 Kissei Pharmaceut Co Ltd Novel 1-substituted imidazole derivative
JPS58150566A (ja) * 1982-03-03 1983-09-07 Yoshitomi Pharmaceut Ind Ltd 新規イミダゾ−ル誘導体
DE3228266A1 (de) * 1982-07-29 1984-02-02 A. Nattermann & Cie GmbH, 5000 Köln Imidazolylalkylthiophene, verfahren zu ihrer herstellung und diese enthaltende pharmazeutische praeparate
DE3329028A1 (de) * 1983-08-11 1985-02-28 Cassella Ag, 6000 Frankfurt Substituierte (2-amino-2-imidazolin-1-yl)-essigsaeurederivate, verfahren zu ihrer herstellung, ihre verwendung und sie enthaltende pharmazeutische zubereitungen

Also Published As

Publication number Publication date
HUT50168A (en) 1989-12-28
FI880430A0 (fi) 1988-01-29
IT1219827B (it) 1990-05-24
CS411291A3 (en) 1992-06-17
ATA18288A (de) 1992-08-15
NZ223359A (en) 1991-03-26
FI880430L (fi) 1988-08-01
NL8800099A (nl) 1988-08-16
CH675721A5 (enExample) 1990-10-31
FR2610322A1 (fr) 1988-08-05
GB2200910B (en) 1991-01-16
ZA88665B (en) 1989-09-27
US4835174A (en) 1989-05-30
ES2008421A6 (es) 1989-07-16
MY102415A (en) 1992-06-17
AT395852B (de) 1993-03-25
IL85252A0 (en) 1988-07-31
FI90080B (fi) 1993-09-15
SE8800293L (sv) 1988-08-01
LU87122A1 (fr) 1988-08-23
IT8847578A0 (it) 1988-01-29
FR2610322B1 (fr) 1990-02-16
PT86666B (pt) 1992-04-30
CA1327805C (en) 1994-03-15
PT86666A (pt) 1988-02-01
GB2200910A (en) 1988-08-17
SE466150B (sv) 1992-01-07
HU204047B (en) 1991-11-28
PH24837A (en) 1990-10-30
GR880100042A (el) 1988-12-16
SE8800293D0 (sv) 1988-01-29
IL85252A (en) 1992-03-29
GB8801804D0 (en) 1988-02-24
BE1001005A3 (fr) 1989-06-06
KR880009013A (ko) 1988-09-13
AU607966B2 (en) 1991-03-21
FI90080C (fi) 1993-12-27
DK46288A (da) 1988-08-01
AU1096088A (en) 1988-08-04
JPS63201185A (ja) 1988-08-19
DK46288D0 (da) 1988-01-29
IE880244L (en) 1988-07-31

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Legal Events

Date Code Title Description
MM4A Patent lapsed