IE42881B1 - Rifamycin derivatives - Google Patents
Rifamycin derivativesInfo
- Publication number
- IE42881B1 IE42881B1 IE448/76A IE44876A IE42881B1 IE 42881 B1 IE42881 B1 IE 42881B1 IE 448/76 A IE448/76 A IE 448/76A IE 44876 A IE44876 A IE 44876A IE 42881 B1 IE42881 B1 IE 42881B1
- Authority
- IE
- Ireland
- Prior art keywords
- rifamycin
- cyclobutyl
- compound
- rifamycin compound
- optionally substituted
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D498/08—Bridged systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Communicable Diseases (AREA)
- Pharmacology & Pharmacy (AREA)
- Oncology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB10020/75A GB1478563A (en) | 1975-03-05 | 1975-03-05 | Rifamycin derivatives |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| IE42881L IE42881L (en) | 1976-09-05 |
| IE42881B1 true IE42881B1 (en) | 1980-11-05 |
Family
ID=9959968
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IE448/76A IE42881B1 (en) | 1975-03-05 | 1976-03-04 | Rifamycin derivatives |
Country Status (27)
| Country | Link |
|---|---|
| US (1) | US4002752A (online.php) |
| JP (1) | JPS51113900A (online.php) |
| AR (1) | AR210113A1 (online.php) |
| AT (1) | AT344896B (online.php) |
| BE (1) | BE839255A (online.php) |
| CA (1) | CA1057748A (online.php) |
| CH (1) | CH610325A5 (online.php) |
| DD (1) | DD123888A5 (online.php) |
| DE (1) | DE2608218C3 (online.php) |
| DK (1) | DK136655B (online.php) |
| ES (1) | ES445790A1 (online.php) |
| FI (1) | FI59102C (online.php) |
| FR (1) | FR2302742A1 (online.php) |
| GB (1) | GB1478563A (online.php) |
| HK (1) | HK35282A (online.php) |
| HU (1) | HU170451B (online.php) |
| IE (1) | IE42881B1 (online.php) |
| KE (1) | KE3099A (online.php) |
| LU (1) | LU74478A1 (online.php) |
| MX (1) | MX3737E (online.php) |
| NL (1) | NL165745C (online.php) |
| NO (1) | NO143796C (online.php) |
| PT (1) | PT64866B (online.php) |
| SE (1) | SE420728B (online.php) |
| SU (1) | SU575030A3 (online.php) |
| YU (1) | YU39477B (online.php) |
| ZA (1) | ZA761043B (online.php) |
Families Citing this family (19)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE2728869A1 (de) * | 1976-06-25 | 1977-12-29 | Antibiotice Iasi Intreprindere | Rifamycinen und verfahren zu deren herstellung |
| GR64108B (en) * | 1977-04-15 | 1980-01-24 | Dso Pharmachim | Method for the preparation of azomethine-derivatives of rifamycin s.v |
| GB1576886A (en) * | 1977-04-20 | 1980-10-15 | Lepetit Spa | Rifamycin derivatives |
| GB1594134A (en) * | 1977-11-25 | 1981-07-30 | Holco Investment Inc | Rifamycins |
| AU536524B2 (en) * | 1979-06-28 | 1984-05-10 | Gruppo Lepetit S.P.A. | Water soluble hydrozones of 3-formylifamyan |
| US4447432A (en) * | 1981-11-17 | 1984-05-08 | Farmitalia Carlo Erba S.P.A. | Azino rifamycins |
| US4681938A (en) * | 1984-08-27 | 1987-07-21 | Ciba-Geigy Corporation | Novel polycyclic hydrazones of rifamycins, their manufacture, and their pharmaceutical compositions for treating tuberculosis |
| JPS63501712A (ja) * | 1985-10-18 | 1988-07-14 | チバ−ガイギ− アクチエンゲゼルシヤフト | 置換４−ベンジルピペラジニル化合物 |
| JPH02501301A (ja) * | 1987-09-25 | 1990-05-10 | チバ‐ガイギー アクチェンゲゼルシャフト | ４‐（トリアルキルベンジル）‐ピペラジニル化合物のジアシル誘導体 |
| GB8816620D0 (en) * | 1988-07-13 | 1988-08-17 | Lepetit Spa | Rifapentine hydrohalides |
| KR0170000B1 (ko) * | 1990-06-29 | 1999-02-01 | 레나토 스가르비 | 순수한 결정 형태의 리파펜틴 |
| EP1928890B1 (en) | 2005-08-11 | 2013-04-03 | Targanta Therapeutics Inc. | Phosphonated rifamycins and uses thereof for the prevention and treatment of bone and joint infections |
| US8524691B2 (en) | 2008-08-13 | 2013-09-03 | The Medicines Company | Phosphonated rifamycins and uses thereof for the prevention and treatment of bone and joint infections |
| RU2496475C2 (ru) | 2011-10-26 | 2013-10-27 | Александр Васильевич Иващенко | Фармацевтическая композиция и набор для лечения бактериальных инфекций |
| ES2876004T3 (es) | 2012-08-13 | 2021-11-11 | Adipharm Ead | Formulaciones farmacéuticas que contienen derivados de 3-(4-cinamil-L-piperazinil) amino de 3-formilrifamicina S |
| CN103951677B (zh) * | 2014-03-17 | 2016-04-06 | 四川省长征药业股份有限公司 | 利福喷丁的制备方法 |
| US20240199642A1 (en) * | 2021-04-21 | 2024-06-20 | Interquim S.A. De C.V. | Method for obtaining rifapentine with a new crystalline form |
| CN115047122B (zh) * | 2022-06-29 | 2023-05-02 | 重庆华邦胜凯制药有限公司 | 利福喷丁及其合成过程中所产生的杂质的分析方法 |
| CN117186032A (zh) * | 2023-09-08 | 2023-12-08 | 徐州博康信息化学品有限公司 | 1-氨基-4-环戊基哌嗪及其中间体的制备方法 |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR208F (online.php) * | 1964-07-31 | |||
| AR205434A1 (es) * | 1972-03-27 | 1976-05-07 | Lepetit Spa | Proceso para la preparacion de 3-acilhidrazonometil rifamicinas sv |
| GB1392272A (en) * | 1972-05-31 | 1975-04-30 | Lepetit Spa | 3-formylrifamycin azines |
-
1975
- 1975-03-05 GB GB10020/75A patent/GB1478563A/en not_active Expired
-
1976
- 1976-02-19 NO NO760549A patent/NO143796C/no unknown
- 1976-02-23 ZA ZA1043A patent/ZA761043B/xx unknown
- 1976-02-23 SE SE7602122A patent/SE420728B/xx not_active IP Right Cessation
- 1976-02-25 DK DK78476AA patent/DK136655B/da not_active IP Right Cessation
- 1976-02-26 US US05/661,587 patent/US4002752A/en not_active Expired - Lifetime
- 1976-02-28 DE DE2608218A patent/DE2608218C3/de not_active Expired
- 1976-03-03 AR AR262431A patent/AR210113A1/es active
- 1976-03-03 NL NL7602191.A patent/NL165745C/xx not_active IP Right Cessation
- 1976-03-03 SU SU7602329559A patent/SU575030A3/ru active
- 1976-03-04 HU HULE790A patent/HU170451B/hu unknown
- 1976-03-04 JP JP51023701A patent/JPS51113900A/ja active Granted
- 1976-03-04 IE IE448/76A patent/IE42881B1/en not_active IP Right Cessation
- 1976-03-04 MX MX7636U patent/MX3737E/es unknown
- 1976-03-04 PT PT64866A patent/PT64866B/pt unknown
- 1976-03-04 CH CH271376A patent/CH610325A5/xx not_active IP Right Cessation
- 1976-03-04 CA CA247,156A patent/CA1057748A/en not_active Expired
- 1976-03-04 LU LU74478A patent/LU74478A1/xx unknown
- 1976-03-05 ES ES445790A patent/ES445790A1/es not_active Expired
- 1976-03-05 AT AT162876A patent/AT344896B/de not_active IP Right Cessation
- 1976-03-05 BE BE164907A patent/BE839255A/xx not_active IP Right Cessation
- 1976-03-05 YU YU572/76A patent/YU39477B/xx unknown
- 1976-03-05 DD DD191727A patent/DD123888A5/xx unknown
- 1976-03-05 FR FR7606379A patent/FR2302742A1/fr active Granted
- 1976-03-05 FI FI760561A patent/FI59102C/fi not_active IP Right Cessation
-
1980
- 1980-11-01 KE KE3099A patent/KE3099A/xx unknown
-
1982
- 1982-08-03 HK HK352/82A patent/HK35282A/xx unknown
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| MK9A | Patent expired |