IE42881B1 - Rifamycin derivatives - Google Patents

Rifamycin derivatives

Info

Publication number
IE42881B1
IE42881B1 IE448/76A IE44876A IE42881B1 IE 42881 B1 IE42881 B1 IE 42881B1 IE 448/76 A IE448/76 A IE 448/76A IE 44876 A IE44876 A IE 44876A IE 42881 B1 IE42881 B1 IE 42881B1
Authority
IE
Ireland
Prior art keywords
rifamycin
cyclobutyl
compound
rifamycin compound
optionally substituted
Prior art date
Application number
IE448/76A
Other languages
English (en)
Other versions
IE42881L (en
Original Assignee
Lepetit Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lepetit Spa filed Critical Lepetit Spa
Publication of IE42881L publication Critical patent/IE42881L/xx
Publication of IE42881B1 publication Critical patent/IE42881B1/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/08—Bridged systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
IE448/76A 1975-03-05 1976-03-04 Rifamycin derivatives IE42881B1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB10020/75A GB1478563A (en) 1975-03-05 1975-03-05 Rifamycin derivatives

Publications (2)

Publication Number Publication Date
IE42881L IE42881L (en) 1976-09-05
IE42881B1 true IE42881B1 (en) 1980-11-05

Family

ID=9959968

Family Applications (1)

Application Number Title Priority Date Filing Date
IE448/76A IE42881B1 (en) 1975-03-05 1976-03-04 Rifamycin derivatives

Country Status (27)

Country Link
US (1) US4002752A (en:Method)
JP (1) JPS51113900A (en:Method)
AR (1) AR210113A1 (en:Method)
AT (1) AT344896B (en:Method)
BE (1) BE839255A (en:Method)
CA (1) CA1057748A (en:Method)
CH (1) CH610325A5 (en:Method)
DD (1) DD123888A5 (en:Method)
DE (1) DE2608218C3 (en:Method)
DK (1) DK136655B (en:Method)
ES (1) ES445790A1 (en:Method)
FI (1) FI59102C (en:Method)
FR (1) FR2302742A1 (en:Method)
GB (1) GB1478563A (en:Method)
HK (1) HK35282A (en:Method)
HU (1) HU170451B (en:Method)
IE (1) IE42881B1 (en:Method)
KE (1) KE3099A (en:Method)
LU (1) LU74478A1 (en:Method)
MX (1) MX3737E (en:Method)
NL (1) NL165745C (en:Method)
NO (1) NO143796C (en:Method)
PT (1) PT64866B (en:Method)
SE (1) SE420728B (en:Method)
SU (1) SU575030A3 (en:Method)
YU (1) YU39477B (en:Method)
ZA (1) ZA761043B (en:Method)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2728869A1 (de) * 1976-06-25 1977-12-29 Antibiotice Iasi Intreprindere Rifamycinen und verfahren zu deren herstellung
GR64108B (en) * 1977-04-15 1980-01-24 Dso Pharmachim Method for the preparation of azomethine-derivatives of rifamycin s.v
GB1576886A (en) * 1977-04-20 1980-10-15 Lepetit Spa Rifamycin derivatives
GB1594134A (en) * 1977-11-25 1981-07-30 Holco Investment Inc Rifamycins
AU536524B2 (en) * 1979-06-28 1984-05-10 Gruppo Lepetit S.P.A. Water soluble hydrozones of 3-formylifamyan
US4447432A (en) * 1981-11-17 1984-05-08 Farmitalia Carlo Erba S.P.A. Azino rifamycins
US4681938A (en) * 1984-08-27 1987-07-21 Ciba-Geigy Corporation Novel polycyclic hydrazones of rifamycins, their manufacture, and their pharmaceutical compositions for treating tuberculosis
ATE47857T1 (de) * 1985-10-18 1989-11-15 Ciba Geigy Ag Substituierte 4-benzyl-piperazinyl-verbindungen.
JPH02501301A (ja) * 1987-09-25 1990-05-10 チバ‐ガイギー　アクチェンゲゼルシャフト ４‐（トリアルキルベンジル）‐ピペラジニル化合物のジアシル誘導体
GB8816620D0 (en) * 1988-07-13 1988-08-17 Lepetit Spa Rifapentine hydrohalides
CA2082809C (en) * 1990-06-29 1995-10-17 Marino Nebuloni Pure crystalline form of rifapentine
KR101327635B1 (ko) 2005-08-11 2013-11-12 타간타 테라퓨틱스 인크. 포스폰산화 리파마이신, 및 그의 뼈 및 관절 감염의 저지및 치료 용도
EP2324041A4 (en) 2008-08-13 2012-06-13 Targanta Therapeutics Corp PHOSPHONIZED RIFAMYCINS AND ITS APPLICATION FOR THE PREVENTION AND TREATMENT OF BONE AND JOINT INFECTIONS
RU2496475C2 (ru) 2011-10-26 2013-10-27 Александр Васильевич Иващенко Фармацевтическая композиция и набор для лечения бактериальных инфекций
BR112015002945B1 (pt) 2012-08-13 2021-08-31 Adipharm Ead Formulações farmacêuticas contendo derivados de 3-(4-cinamil-1-piperazinil)-amino de 3- formil-rifamicina sv e 3-formil-rifamicina s e um processo para sua preparação
CN103951677B (zh) * 2014-03-17 2016-04-06 四川省长征药业股份有限公司 利福喷丁的制备方法
MX2023012416A (es) * 2021-04-21 2024-03-05 Interquim S A De C V Proceso de obtencion de rifapentina con una nueva forma cristalina.
CN115047122B (zh) * 2022-06-29 2023-05-02 重庆华邦胜凯制药有限公司 利福喷丁及其合成过程中所产生的杂质的分析方法
CN117186032A (zh) * 2023-09-08 2023-12-08 徐州博康信息化学品有限公司 1-氨基-4-环戊基哌嗪及其中间体的制备方法

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR208F (en:Method) * 1964-07-31
AR205434A1 (es) * 1972-03-27 1976-05-07 Lepetit Spa Proceso para la preparacion de 3-acilhidrazonometil rifamicinas sv
GB1392272A (en) * 1972-05-31 1975-04-30 Lepetit Spa 3-formylrifamycin azines

Also Published As

Publication number Publication date
NO143796B (no) 1981-01-05
FI760561A7 (en:Method) 1976-09-06
YU39477B (en) 1984-12-31
FI59102C (fi) 1981-06-10
PT64866A (en) 1976-04-01
DK78476A (en:Method) 1976-09-06
HK35282A (en) 1982-08-13
GB1478563A (en) 1977-07-06
NO760549L (en:Method) 1976-09-07
AR210113A1 (es) 1977-06-30
SE7602122L (sv) 1976-09-06
HU170451B (en:Method) 1977-06-28
DK136655C (en:Method) 1978-04-17
NL7602191A (nl) 1976-09-07
US4002752A (en) 1977-01-11
LU74478A1 (en:Method) 1976-09-01
JPS51113900A (en) 1976-10-07
BE839255A (fr) 1976-09-06
AU1170476A (en) 1977-09-08
DD123888A5 (en:Method) 1977-01-19
DK136655B (da) 1977-11-07
DE2608218A1 (de) 1976-09-16
DE2608218C3 (de) 1981-12-10
NO143796C (no) 1981-04-15
KE3099A (en) 1981-02-13
DE2608218B2 (de) 1981-02-26
FR2302742A1 (fr) 1976-10-01
SE420728B (sv) 1981-10-26
NL165745B (nl) 1980-12-15
IE42881L (en) 1976-09-05
JPS5530797B2 (en:Method) 1980-08-13
CH610325A5 (en:Method) 1979-04-12
AT344896B (de) 1978-08-10
YU57276A (en) 1982-06-30
FR2302742B1 (en:Method) 1979-10-12
NL165745C (nl) 1981-05-15
MX3737E (es) 1981-06-05
CA1057748A (en) 1979-07-03
SU575030A3 (ru) 1977-09-30
FI59102B (fi) 1981-02-27
ZA761043B (en) 1977-01-26
ATA162876A (de) 1977-12-15
ES445790A1 (es) 1977-06-01
PT64866B (en) 1977-07-20

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