IE37782B1 - Penicillin compounds - Google Patents
Penicillin compoundsInfo
- Publication number
- IE37782B1 IE37782B1 IE645/72A IE64572A IE37782B1 IE 37782 B1 IE37782 B1 IE 37782B1 IE 645/72 A IE645/72 A IE 645/72A IE 64572 A IE64572 A IE 64572A IE 37782 B1 IE37782 B1 IE 37782B1
- Authority
- IE
- Ireland
- Prior art keywords
- acylamido
- syn
- isomers
- org
- beta
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/02—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
- C07D307/34—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D307/38—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D307/40—Radicals substituted by oxygen atoms
- C07D307/42—Singly bound oxygen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C271/00—Derivatives of carbamic acids, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups
- C07C271/06—Esters of carbamic acids
- C07C271/08—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms
- C07C271/10—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms
- C07C271/14—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms to carbon atoms of hydrocarbon radicals substituted by halogen atoms or by nitro or nitroso groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D213/54—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
- C07D213/55—Acids; Esters
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/02—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
- C07D307/34—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D307/38—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D307/54—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D307/78—Benzo [b] furans; Hydrogenated benzo [b] furans
- C07D307/79—Benzo [b] furans; Hydrogenated benzo [b] furans with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D307/78—Benzo [b] furans; Hydrogenated benzo [b] furans
- C07D307/79—Benzo [b] furans; Hydrogenated benzo [b] furans with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
- C07D307/81—Radicals substituted by nitrogen atoms not forming part of a nitro radical
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/06—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring carbon atoms
- C07D333/14—Radicals substituted by singly bound hetero atoms other than halogen
- C07D333/16—Radicals substituted by singly bound hetero atoms other than halogen by oxygen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/06—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring carbon atoms
- C07D333/24—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
- C07D333/52—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
- C07D333/54—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
- C07D333/60—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Cephalosporin Compounds (AREA)
Abstract
6 beta-Acylamido-penam-3 alpha-carboxylic acids and their non-toxic derivs. in which the acylamido gp. has the structure R-C(=N ORa)-CO-NH- (where R is H or an org. gp. and Ra is an etherified monovalent org. gp. linked to the O-atom via a C-atom), the cpd. being present as the syn or anti isomer or as a mixt. of these isomers, partic. cpds. of formula (I): (where B is S or SO), have antibacterial activity against gram-positive organisms as well as Haemophilus influenzae. The syn isomers are active against penicillinase-producing Staphylococci and are resistant to various beta-lactamases.
[FR2137898A1]
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB1508271A GB1399086A (en) | 1971-05-14 | 1971-05-14 | Cephalosporin compounds |
Publications (2)
Publication Number | Publication Date |
---|---|
IE37782L IE37782L (en) | 1972-11-14 |
IE37782B1 true IE37782B1 (en) | 1977-10-12 |
Family
ID=10052709
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
IE645/72A IE37782B1 (en) | 1971-05-14 | 1972-05-12 | Penicillin compounds |
Country Status (14)
Country | Link |
---|---|
JP (1) | JPS5248997B1 (en) |
AT (1) | AT329176B (en) |
AU (2) | AU474163B2 (en) |
BE (1) | BE783448A (en) |
CH (1) | CH579571A5 (en) |
DE (1) | DE2223287A1 (en) |
ES (1) | ES402650A1 (en) |
FR (2) | FR2137898A1 (en) |
HU (1) | HU172017B (en) |
IE (1) | IE37782B1 (en) |
IL (1) | IL39428A (en) |
NL (1) | NL7206466A (en) |
PL (1) | PL101031B1 (en) |
ZA (2) | ZA723224B (en) |
Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US7514439B2 (en) | 2005-07-11 | 2009-04-07 | Mitsubishi Tanabe Pharma Corporation | Oxime derivative and preparations thereof |
Families Citing this family (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB1443950A (en) * | 1972-10-25 | 1976-07-28 | Glaxo Lab Ltd | Acylamido-penam-carboxylic acids and their derivatives |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US2542812A (en) * | 1946-04-03 | 1951-02-20 | Walter H Hartung | Preparation of aminoacidamides |
DE1159449B (en) * | 1961-03-22 | 1963-12-19 | Gruenenthal Chemie | Process for the preparation of 6-acylaminopenicillanic acids and their salts |
SE311519B (en) * | 1962-12-14 | 1969-06-16 | Astra Ab |
-
1972
- 1972-05-12 IL IL39428A patent/IL39428A/en unknown
- 1972-05-12 IE IE645/72A patent/IE37782B1/en unknown
- 1972-05-12 HU HU72GA00001095A patent/HU172017B/en unknown
- 1972-05-12 NL NL7206466A patent/NL7206466A/xx not_active Application Discontinuation
- 1972-05-12 BE BE783448A patent/BE783448A/en unknown
- 1972-05-12 PL PL1972155354A patent/PL101031B1/en unknown
- 1972-05-12 DE DE19722223287 patent/DE2223287A1/en active Pending
- 1972-05-12 ZA ZA723224A patent/ZA723224B/en unknown
- 1972-05-12 JP JP47047149A patent/JPS5248997B1/ja active Pending
- 1972-05-12 ES ES402650A patent/ES402650A1/en not_active Expired
- 1972-05-12 CH CH705872A patent/CH579571A5/xx not_active IP Right Cessation
- 1972-05-12 ZA ZA723223A patent/ZA723223B/en unknown
- 1972-05-15 AU AU42298/72A patent/AU474163B2/en not_active Expired
- 1972-05-15 FR FR7217282A patent/FR2137898A1/en active Granted
- 1972-05-15 AT AT420772A patent/AT329176B/en not_active IP Right Cessation
- 1972-05-15 AU AU42299/72A patent/AU475444B2/en not_active Expired
-
1975
- 1975-12-09 FR FR7537636A patent/FR2287231A1/en active Granted
Cited By (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US7514439B2 (en) | 2005-07-11 | 2009-04-07 | Mitsubishi Tanabe Pharma Corporation | Oxime derivative and preparations thereof |
US8119626B2 (en) | 2005-07-11 | 2012-02-21 | Mitsubishi Tanabe Pharma Corporation | Oxime derivative and preparations thereof |
Also Published As
Publication number | Publication date |
---|---|
ES402650A1 (en) | 1976-01-01 |
FR2287231B1 (en) | 1978-09-01 |
BE783448A (en) | 1972-11-13 |
FR2137898B1 (en) | 1976-04-16 |
NL7206466A (en) | 1972-11-16 |
JPS5248997B1 (en) | 1977-12-14 |
DE2223287A1 (en) | 1972-12-07 |
ZA723223B (en) | 1973-02-28 |
AU4229872A (en) | 1974-01-03 |
AU475444B2 (en) | 1976-08-26 |
FR2137898A1 (en) | 1972-12-29 |
AT329176B (en) | 1976-04-26 |
CH579571A5 (en) | 1976-09-15 |
AU4229972A (en) | 1973-12-20 |
IL39428A0 (en) | 1972-07-26 |
AU474163B2 (en) | 1976-07-15 |
ZA723224B (en) | 1973-03-28 |
PL101031B1 (en) | 1978-11-30 |
FR2287231A1 (en) | 1976-05-07 |
IL39428A (en) | 1977-01-31 |
IE37782L (en) | 1972-11-14 |
HU172017B (en) | 1978-05-28 |
ATA420772A (en) | 1975-07-15 |
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