ID30057A - Turunan fenilalaninol - Google Patents

Turunan fenilalaninol

Info

Publication number
ID30057A
ID30057A IDW00200101769A ID20011769A ID30057A ID 30057 A ID30057 A ID 30057A ID W00200101769 A IDW00200101769 A ID W00200101769A ID 20011769 A ID20011769 A ID 20011769A ID 30057 A ID30057 A ID 30057A
Authority
ID
Indonesia
Prior art keywords
alkyl
lower alkyl
alkanoyl
aryl
halo
Prior art date
Application number
IDW00200101769A
Other languages
English (en)
Indonesian (id)
Inventor
Achytharao Sidduri
Jefferson Wright Tilley
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of ID30057A publication Critical patent/ID30057A/id

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C323/00Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
    • C07C323/50Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton
    • C07C323/51Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton
    • C07C323/60Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton with the carbon atom of at least one of the carboxyl groups bound to nitrogen atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/16Amides, e.g. hydroxamic acids
    • A61K31/165Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
    • A61K31/166Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide having the carbon of a carboxamide group directly attached to the aromatic ring, e.g. procainamide, procarbazine, metoclopramide, labetalol
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/06Antiasthmatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/02Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C233/00Carboxylic acid amides
    • C07C233/64Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings
    • C07C233/77Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by amino groups
    • C07C233/80Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by amino groups with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by a carbon atom of a six-membered aromatic ring
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07BGENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00Indexing scheme relating to specific properties of organic compounds
    • C07B2200/07Optical isomers
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2601/00Systems containing only non-condensed rings
    • C07C2601/06Systems containing only non-condensed rings with a five-membered ring
    • C07C2601/08Systems containing only non-condensed rings with a five-membered ring the ring being saturated

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pulmonology (AREA)
  • Rheumatology (AREA)
  • Immunology (AREA)
  • Epidemiology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Pain & Pain Management (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Neurology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pyridine Compounds (AREA)
IDW00200101769A 1999-02-18 2000-02-12 Turunan fenilalaninol ID30057A (id)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US12049899P 1999-02-18 1999-02-18

Publications (1)

Publication Number Publication Date
ID30057A true ID30057A (id) 2001-11-01

Family

ID=22390691

Family Applications (1)

Application Number Title Priority Date Filing Date
IDW00200101769A ID30057A (id) 1999-02-18 2000-02-12 Turunan fenilalaninol

Country Status (29)

Country Link
US (1) US6420600B1 (no)
EP (1) EP1154987B1 (no)
JP (1) JP2002537283A (no)
KR (1) KR100636458B1 (no)
CN (1) CN1213020C (no)
AT (1) ATE264835T1 (no)
AU (1) AU771938B2 (no)
BR (1) BR0008368A (no)
CA (1) CA2362833C (no)
CZ (1) CZ20012984A3 (no)
DE (1) DE60010049T2 (no)
DK (1) DK1154987T3 (no)
ES (1) ES2218116T3 (no)
HK (1) HK1043589A1 (no)
HR (1) HRP20010594B1 (no)
HU (1) HUP0200343A3 (no)
ID (1) ID30057A (no)
IL (2) IL144641A0 (no)
MA (1) MA26772A1 (no)
MX (1) MXPA01008178A (no)
NO (1) NO20013946D0 (no)
PL (1) PL349463A1 (no)
PT (1) PT1154987E (no)
RU (1) RU2238265C2 (no)
SI (1) SI1154987T1 (no)
TR (1) TR200102395T2 (no)
WO (1) WO2000048988A1 (no)
YU (1) YU58601A (no)
ZA (1) ZA200106075B (no)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6939855B2 (en) * 1997-07-31 2005-09-06 Elan Pharmaceuticals, Inc. Anti-inflammatory compositions and method
KR100720907B1 (ko) * 1999-08-13 2007-05-25 바이오겐 아이덱 엠에이 인코포레이티드 세포 유착 억제제
US6388084B1 (en) 1999-12-06 2002-05-14 Hoffmann-La Roche Inc. 4-pyridinyl-n-acyl-l-phenylalanines
US6380387B1 (en) 1999-12-06 2002-04-30 Hoffmann-La Roche Inc. 4-Pyrimidinyl-n-acyl-l phenylalanines
US7015323B2 (en) 2003-05-20 2006-03-21 Genentech, Inc. Thiocarbamate inhibitors of alpha-4 integrins
WO2006081986A1 (en) * 2005-02-07 2006-08-10 F.Hoffmann-La Roche Ag Bambuterol and integrin inhibitor combination
WO2006094640A2 (en) * 2005-03-04 2006-09-14 F.Hoffmann-La Roche Ag Roflumilast and integrin inhibitor combination and method of treatment
IL172896A0 (en) * 2005-12-29 2006-06-11 Yeda Res & Dev Cxcr4 inhibition
US8877815B2 (en) 2010-11-16 2014-11-04 Novartis Ag Substituted carbamoylcycloalkyl acetic acid derivatives as NEP

Family Cites Families (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE584914A (no) 1958-11-24
US3527793A (en) 1967-08-18 1970-09-08 Bristol Myers Co Phenylglycine derivatives
IT1190378B (it) 1985-06-21 1988-02-16 Isf Spa Derivati pirrolidonici
US5039805A (en) 1988-12-08 1991-08-13 Hoffmann-La Roche Inc. Novel benzoic and phenylacetic acid derivatives
US5463116A (en) 1991-07-30 1995-10-31 Ajinomoto Co., Inc. Crystals of N- (trans-4-isopropylcyclohexlycarbonyl)-D-phenylalanine and methods for preparing them
CA2191979A1 (en) 1994-06-20 1995-12-28 Muneo Takatani Condensed imidazole compounds, their production and use
US6306840B1 (en) 1995-01-23 2001-10-23 Biogen, Inc. Cell adhesion inhibitors
US5804595A (en) 1995-12-05 1998-09-08 Regents Of The University Of Minnesota Kappa opioid receptor agonists
PT891325E (pt) * 1996-03-29 2002-07-31 Searle & Co Derivados do acido fenilpropanoico para-substituido como antagonistas de integrina
DE69706407T2 (de) 1996-03-29 2002-05-29 Searle & Co META-SUBSTITUIERTE PHENYLENDERIVATE UND IHRE VERWENDUNG ALS ALPHAvBETA3 INTERGRIN-ANTAGONISTEN ODER INHIBITOREN
ID19155A (id) * 1996-12-13 1998-06-18 Tanabe Seiyaku Co Turunan-turunan piridin, pembuatannya dan intermediet untuk pembuatannya
EP1001764A4 (en) * 1997-05-29 2005-08-24 Merck & Co Inc Heterocyclic amides as cell adhesion inhibitors
TR200000482T2 (tr) * 1997-08-22 2000-06-21 F. Hoffmann-La Roche Ag. N-Aroilfenilalanin türevleri.
PT1005446E (pt) * 1997-08-22 2004-06-30 Hoffmann La Roche Derivados de n-aroilfenilalanina
US6555562B1 (en) 1998-02-26 2003-04-29 Celltech R&D Limited Phenylalanine derivatives
US6521626B1 (en) 1998-03-24 2003-02-18 Celltech R&D Limited Thiocarboxamide derivatives
GB9811159D0 (en) 1998-05-22 1998-07-22 Celltech Therapeutics Ltd Chemical compounds

Also Published As

Publication number Publication date
HRP20010594A2 (en) 2002-08-31
CN1340043A (zh) 2002-03-13
TR200102395T2 (tr) 2001-12-21
EP1154987B1 (en) 2004-04-21
HRP20010594B1 (en) 2006-02-28
PL349463A1 (en) 2002-07-29
EP1154987A1 (en) 2001-11-21
ES2218116T3 (es) 2004-11-16
HUP0200343A2 (en) 2002-06-29
CZ20012984A3 (cs) 2002-02-13
ZA200106075B (en) 2002-10-24
CA2362833C (en) 2009-04-07
CN1213020C (zh) 2005-08-03
ATE264835T1 (de) 2004-05-15
HK1043589A1 (en) 2002-09-20
IL144641A0 (en) 2002-05-23
US6420600B1 (en) 2002-07-16
DE60010049D1 (de) 2004-05-27
NO20013946L (no) 2001-08-14
AU771938B2 (en) 2004-04-08
SI1154987T1 (en) 2004-08-31
YU58601A (sh) 2004-05-12
KR20010102260A (ko) 2001-11-15
JP2002537283A (ja) 2002-11-05
DK1154987T3 (da) 2004-08-09
IL144641A (en) 2006-09-05
CA2362833A1 (en) 2000-08-24
AU2548600A (en) 2000-09-04
NO20013946D0 (no) 2001-08-14
WO2000048988A1 (en) 2000-08-24
PT1154987E (pt) 2004-08-31
HUP0200343A3 (en) 2005-04-28
DE60010049T2 (de) 2005-03-31
RU2238265C2 (ru) 2004-10-20
KR100636458B1 (ko) 2006-10-18
MXPA01008178A (es) 2002-03-13
MA26772A1 (fr) 2004-12-20
BR0008368A (pt) 2001-11-06

Similar Documents

Publication Publication Date Title
US6426348B1 (en) Diphenyl heterocyclic thioamide derivatives
ID30057A (id) Turunan fenilalaninol
EA200000427A1 (ru) Терапевтические применения хинолиновых производных
MY144184A (en) Disposable wearing article
PL315030A1 (en) Method of bonding a flexible material with its associated substrate and product obtained thereby
NO20000413L (no) Karbamyloksyforbindelser som inhiberer leukocytt adhesjon mediert av VLA-4
DE69928226T8 (de) Chemokin rezeptor antagonisten und verwendung
NZ505089A (en) PPAR-gamma receptor activators, useful for the treatment of skin disorders
EP1329459A3 (en) Monoclonal antibodies against the interferon receptor, with neutralizing activity against type I interferon
ATE204471T1 (de) Pyrimidin- oder triazincarbonsäurederivate zur verwendung als arzneimittel
BR9609092A (pt) Prendedores de aba de fita para artigos absorventes descartáveis
HU9303009D0 (en) New 2-saccharinyl-methyl-aryl-carboxylat derivatives and pharmaceutical preparations containing said compounds
DE59100797D1 (de) Windel mit Dichtungsklappen.
DE3880499D1 (de) Cyanhydrinderivate und deren verwendung in fluessigkristallmaterialien und vorrichtungen.
NZ335318A (en) (o-acyl-p-N-acylamino-phenyl)-O-phosphoethanolamines with anti-inflammatory activity
HUP0302440A2 (hu) Amino-kinolin származékok, eljárás előállításukra és ezeket hatóanyagként tartalmazó gyógyszerkészítmények