HUP0001613A2 - Eljárás tercier nitrillel szubsztituált aromás vegyület előállítására - Google Patents
Eljárás tercier nitrillel szubsztituált aromás vegyület előállításáraInfo
- Publication number
- HUP0001613A2 HUP0001613A2 HU0001613A HUP0001613A HUP0001613A2 HU P0001613 A2 HUP0001613 A2 HU P0001613A2 HU 0001613 A HU0001613 A HU 0001613A HU P0001613 A HUP0001613 A HU P0001613A HU P0001613 A2 HUP0001613 A2 HU P0001613A2
- Authority
- HU
- Hungary
- Prior art keywords
- aromatic compound
- formula
- nitrile
- tertiary
- producing
- Prior art date
Links
- 150000001491 aromatic compounds Chemical group 0.000 title abstract 4
- 125000002560 nitrile group Chemical group 0.000 title 1
- 150000002825 nitriles Chemical group 0.000 abstract 2
- 239000000010 aprotic solvent Substances 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 125000000962 organic group Chemical group 0.000 abstract 1
Classifications
-
- G—PHYSICS
- G02—OPTICS
- G02C—SPECTACLES; SUNGLASSES OR GOGGLES INSOFAR AS THEY HAVE THE SAME FEATURES AS SPECTACLES; CONTACT LENSES
- G02C3/00—Special supporting arrangements for lens assemblies or monocles
- G02C3/003—Arrangements for fitting and securing to the head in the position of use
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D213/54—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
- C07D213/57—Nitriles
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C253/00—Preparation of carboxylic acid nitriles
- C07C253/30—Preparation of carboxylic acid nitriles by reactions not involving the formation of cyano groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/54—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings condensed with carbocyclic rings or ring systems
- C07D231/56—Benzopyrazoles; Hydrogenated benzopyrazoles
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Physics & Mathematics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Health & Medical Sciences (AREA)
- General Physics & Mathematics (AREA)
- Ophthalmology & Optometry (AREA)
- Optics & Photonics (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pyridine Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Abstract
A találmány tárgya eljárás (1.0.0) általános képletű tercier nitrillelszubsztituált aromás vegyület előállítására oly módon, hogy egy(2.0.0) képletű szubsztituált aromás vegyületet (3.0.0) képletűszekunder nitrillel reagáltatják bázis jelenlétében, amelynek pKa-értéke körülbelül 17-30, feltéve, hogy a bázis és a (3.0.0) képletűmegfelelő tercier nitril pKa-értéke közötti különbség nem haladja mega körülbelül 6-ot, aprotikus oldószerben, melynek dielektromosállandója (e) körülbelül 20-nál kevesebb; körülbelül 0-120 °C-on, ésígy (1.0.0) képletű tercier nitrillel szubsztituált aromás vegyületetkapnak, ahol W1, W2, W3, W4 és W5 és R1, R2, R4, R5, R6 és R7 az(1.0.0), (2.0.0) és (3.0.0) képletű vegyületekben ismert szervescsoport, illetve ezek részletezése a bejelentésben található. Ó
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US13017599P | 1999-04-20 | 1999-04-20 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| HU0001613D0 HU0001613D0 (en) | 2000-06-28 |
| HUP0001613A2 true HUP0001613A2 (hu) | 2000-11-28 |
| HUP0001613A3 HUP0001613A3 (en) | 2003-03-28 |
Family
ID=22443407
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| HU0001613A HUP0001613A3 (en) | 1999-04-20 | 2000-04-20 | Process for producing an aromatic compound substituted by a tertiary nitrile |
Country Status (24)
| Country | Link |
|---|---|
| US (1) | US6303782B1 (hu) |
| EP (1) | EP1046635B1 (hu) |
| JP (1) | JP3420553B2 (hu) |
| KR (1) | KR100352111B1 (hu) |
| CN (1) | CN1138756C (hu) |
| AR (1) | AR023571A1 (hu) |
| AT (1) | ATE286019T1 (hu) |
| AU (1) | AU771854B2 (hu) |
| BR (1) | BR0001628A (hu) |
| CA (1) | CA2306004C (hu) |
| DE (1) | DE60017001T2 (hu) |
| DK (1) | DK1046635T3 (hu) |
| ES (1) | ES2233286T3 (hu) |
| HK (1) | HK1032041A1 (hu) |
| HU (1) | HUP0001613A3 (hu) |
| ID (1) | ID25689A (hu) |
| IL (1) | IL135633A (hu) |
| PL (1) | PL339832A1 (hu) |
| PT (1) | PT1046635E (hu) |
| RU (1) | RU2182572C2 (hu) |
| TR (1) | TR200001053A2 (hu) |
| TW (1) | TW552256B (hu) |
| YU (1) | YU19700A (hu) |
| ZA (1) | ZA200001962B (hu) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20040186310A1 (en) * | 2001-06-22 | 2004-09-23 | Kim Keun-Sik | Process for preparation of cyclohexanol derivatives |
| BRPI0608221A2 (pt) * | 2005-04-29 | 2009-11-24 | Wyeth Corp | métodos para preparação de um composto, e para preparar seletivamente um composto de nitrila, e, composto |
| CN101486676B (zh) * | 2008-12-23 | 2010-12-08 | 南京航空航天大学 | 氰甲基吡啶化合物的制备方法 |
| CN102911080B (zh) * | 2012-09-12 | 2015-01-21 | 衢州学院 | 一种制备2,6-二氯-α-(4-氯苯基)-4-硝基苯乙腈的方法 |
| RS58961B1 (sr) | 2015-01-22 | 2019-08-30 | Sanofi Aventis Deutschland | Proces proizvodnje 2-[4-(ciklopropankarbonil)fenil]-2-metil-propannitrila |
| CN107114183B (zh) * | 2017-05-03 | 2019-11-19 | 滨州学院 | 一种提高冬枣果实品质的土壤管理方法 |
-
2000
- 2000-03-01 US US09/516,417 patent/US6303782B1/en not_active Expired - Fee Related
- 2000-03-31 PT PT00302766T patent/PT1046635E/pt unknown
- 2000-03-31 EP EP00302766A patent/EP1046635B1/en not_active Expired - Lifetime
- 2000-03-31 ES ES00302766T patent/ES2233286T3/es not_active Expired - Lifetime
- 2000-03-31 AT AT00302766T patent/ATE286019T1/de not_active IP Right Cessation
- 2000-03-31 DK DK00302766T patent/DK1046635T3/da active
- 2000-03-31 DE DE60017001T patent/DE60017001T2/de not_active Expired - Fee Related
- 2000-04-03 YU YU19700A patent/YU19700A/sh unknown
- 2000-04-06 AU AU26449/00A patent/AU771854B2/en not_active Ceased
- 2000-04-12 IL IL13563300A patent/IL135633A/xx not_active IP Right Cessation
- 2000-04-17 TW TW089107165A patent/TW552256B/zh not_active IP Right Cessation
- 2000-04-17 BR BR0001628-4A patent/BR0001628A/pt not_active IP Right Cessation
- 2000-04-18 CN CNB001067516A patent/CN1138756C/zh not_active Expired - Fee Related
- 2000-04-18 ID IDP20000306D patent/ID25689A/id unknown
- 2000-04-18 CA CA002306004A patent/CA2306004C/en not_active Expired - Fee Related
- 2000-04-18 ZA ZA200001962A patent/ZA200001962B/xx unknown
- 2000-04-18 TR TR2000/01053A patent/TR200001053A2/xx unknown
- 2000-04-19 AR ARP000101874A patent/AR023571A1/es unknown
- 2000-04-19 RU RU2000110186/04A patent/RU2182572C2/ru not_active IP Right Cessation
- 2000-04-19 KR KR1020000020556A patent/KR100352111B1/ko not_active IP Right Cessation
- 2000-04-20 JP JP2000119372A patent/JP3420553B2/ja not_active Expired - Fee Related
- 2000-04-20 PL PL00339832A patent/PL339832A1/xx not_active Application Discontinuation
- 2000-04-20 HU HU0001613A patent/HUP0001613A3/hu unknown
-
2001
- 2001-04-12 HK HK01102636A patent/HK1032041A1/xx not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| ES2233286T3 (es) | 2005-06-16 |
| RU2182572C2 (ru) | 2002-05-20 |
| ID25689A (id) | 2000-10-26 |
| TW552256B (en) | 2003-09-11 |
| ZA200001962B (en) | 2002-03-20 |
| JP2000344725A (ja) | 2000-12-12 |
| TR200001053A2 (tr) | 2001-01-22 |
| IL135633A0 (en) | 2001-05-20 |
| AU771854B2 (en) | 2004-04-01 |
| ATE286019T1 (de) | 2005-01-15 |
| YU19700A (sh) | 2003-01-31 |
| US6303782B1 (en) | 2001-10-16 |
| KR100352111B1 (ko) | 2002-09-12 |
| HU0001613D0 (en) | 2000-06-28 |
| CN1138756C (zh) | 2004-02-18 |
| AR023571A1 (es) | 2002-09-04 |
| CA2306004C (en) | 2005-11-29 |
| DK1046635T3 (da) | 2005-03-14 |
| CN1271723A (zh) | 2000-11-01 |
| DE60017001D1 (de) | 2005-02-03 |
| EP1046635A1 (en) | 2000-10-25 |
| IL135633A (en) | 2005-09-25 |
| EP1046635B1 (en) | 2004-12-29 |
| CA2306004A1 (en) | 2000-10-20 |
| HK1032041A1 (en) | 2001-07-06 |
| DE60017001T2 (de) | 2005-12-15 |
| PL339832A1 (en) | 2000-10-23 |
| BR0001628A (pt) | 2001-01-02 |
| KR20000071731A (ko) | 2000-11-25 |
| PT1046635E (pt) | 2005-04-29 |
| HUP0001613A3 (en) | 2003-03-28 |
| AU2644900A (en) | 2000-10-26 |
| JP3420553B2 (ja) | 2003-06-23 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FD9A | Lapse of provisional protection due to non-payment of fees |