HUE056051T2 - Fúzionált biciklikus sGC stimulátorok - Google Patents

Fúzionált biciklikus sGC stimulátorok

Info

Publication number
HUE056051T2
HUE056051T2 HUE17768311A HUE17768311A HUE056051T2 HU E056051 T2 HUE056051 T2 HU E056051T2 HU E17768311 A HUE17768311 A HU E17768311A HU E17768311 A HUE17768311 A HU E17768311A HU E056051 T2 HUE056051 T2 HU E056051T2
Authority
HU
Hungary
Prior art keywords
fused bicyclic
sgc stimulators
sgc
stimulators
bicyclic
Prior art date
Application number
HUE17768311A
Other languages
English (en)
Hungarian (hu)
Inventor
Glen Rennie
Rajesh Iyengar
Thomas Lee
Takashi Nakai
Ara Mermerian
Lei Jia
G-Yoon Im
Paul Renhowe
Joon Jung
Peter Germano
Karthik Iyer
Timothy Barden
Kim Tang
Original Assignee
Cyclerion Therapeutics Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Cyclerion Therapeutics Inc filed Critical Cyclerion Therapeutics Inc
Publication of HUE056051T2 publication Critical patent/HUE056051T2/hu

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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
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    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/4985—Pyrazines or piperazines ortho- or peri-condensed with heterocyclic ring systems
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    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
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    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
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HUE17768311A 2016-09-02 2017-09-01 Fúzionált biciklikus sGC stimulátorok HUE056051T2 (hu)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US201662382942P 2016-09-02 2016-09-02
US201662423445P 2016-11-17 2016-11-17
US201762468598P 2017-03-08 2017-03-08
US201762482486P 2017-04-06 2017-04-06

Publications (1)

Publication Number Publication Date
HUE056051T2 true HUE056051T2 (hu) 2022-01-28

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HUE17768311A HUE056051T2 (hu) 2016-09-02 2017-09-01 Fúzionált biciklikus sGC stimulátorok

Country Status (29)

Country Link
US (4) US10472363B2 (fr)
EP (2) EP3872080B1 (fr)
JP (2) JP7050759B2 (fr)
KR (2) KR20230124760A (fr)
CN (2) CN109790167B (fr)
AU (2) AU2017321810B2 (fr)
BR (1) BR112019004468A2 (fr)
CA (1) CA3035210A1 (fr)
CL (1) CL2019000486A1 (fr)
CO (1) CO2019001760A2 (fr)
CR (2) CR20220309A (fr)
CY (1) CY1124612T1 (fr)
DK (1) DK3507291T3 (fr)
ES (2) ES2885003T3 (fr)
HR (1) HRP20211355T1 (fr)
HU (1) HUE056051T2 (fr)
IL (2) IL292968A (fr)
LT (1) LT3507291T (fr)
MA (1) MA53999A (fr)
MX (3) MX2019002313A (fr)
PE (1) PE20190607A1 (fr)
PH (1) PH12019500461A1 (fr)
PL (1) PL3507291T3 (fr)
PT (1) PT3507291T (fr)
RS (1) RS62256B1 (fr)
SG (1) SG11201901729YA (fr)
SI (1) SI3507291T1 (fr)
TW (2) TWI813078B (fr)
WO (1) WO2018045276A1 (fr)

Families Citing this family (27)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
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