HUE035553T2 - Aminopirimidinil-vegyületek mint JAK-inhibitorok - Google Patents

Aminopirimidinil-vegyületek mint JAK-inhibitorok Download PDF

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Publication number
HUE035553T2
HUE035553T2 HUE15766627A HUE15766627A HUE035553T2 HU E035553 T2 HUE035553 T2 HU E035553T2 HU E15766627 A HUE15766627 A HU E15766627A HU E15766627 A HUE15766627 A HU E15766627A HU E035553 T2 HUE035553 T2 HU E035553T2
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HU
Hungary
Prior art keywords
alkyl
group
carbon atoms
rti
aryl
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HUE15766627A
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English (en)
Hungarian (hu)
Inventor
Andrew Fensome
Ariamala Gopalsamy
Brian S Gerstenberger
Ivan Viktorovich Efremov
Zhao-Kui Wan
Betsy PIERCE
Jean-Baptiste Telliez
John I Trujillo
Liying Zhang
Li Xing
Eddine Saiah
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Pfizer
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=54148580&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=HUE035553(T2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pfizer filed Critical Pfizer
Publication of HUE035553T2 publication Critical patent/HUE035553T2/hu

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    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
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    • C07D401/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
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    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
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HUE15766627A 2014-08-21 2015-08-07 Aminopirimidinil-vegyületek mint JAK-inhibitorok HUE035553T2 (hu)

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US201462039969P 2014-08-21 2014-08-21

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US (5) US9663526B2 (enrdf_load_stackoverflow)
EP (1) EP3183247B9 (enrdf_load_stackoverflow)
JP (1) JP6218260B2 (enrdf_load_stackoverflow)
KR (1) KR101877189B1 (enrdf_load_stackoverflow)
CN (1) CN107074867B (enrdf_load_stackoverflow)
AP (1) AP2017009748A0 (enrdf_load_stackoverflow)
AR (1) AR101599A1 (enrdf_load_stackoverflow)
AU (1) AU2015304883B2 (enrdf_load_stackoverflow)
BR (1) BR112017003054B1 (enrdf_load_stackoverflow)
CA (1) CA2900855C (enrdf_load_stackoverflow)
CL (1) CL2017000406A1 (enrdf_load_stackoverflow)
CO (1) CO2017001603A2 (enrdf_load_stackoverflow)
CR (1) CR20170066A (enrdf_load_stackoverflow)
CU (1) CU24435B1 (enrdf_load_stackoverflow)
CY (1) CY1119771T1 (enrdf_load_stackoverflow)
DK (1) DK3183247T3 (enrdf_load_stackoverflow)
DO (1) DOP2017000048A (enrdf_load_stackoverflow)
EA (1) EA032609B1 (enrdf_load_stackoverflow)
EC (1) ECSP17010156A (enrdf_load_stackoverflow)
ES (1) ES2655971T3 (enrdf_load_stackoverflow)
GE (1) GEP20197003B (enrdf_load_stackoverflow)
GT (1) GT201700035A (enrdf_load_stackoverflow)
HR (1) HRP20171913T1 (enrdf_load_stackoverflow)
HU (1) HUE035553T2 (enrdf_load_stackoverflow)
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