HUE026549T2 - 1-N-azacikloalkil-3-fenoxipropán pszichotróp gyógyszerek elõállítására alkalmas származékai - Google Patents

1-N-azacikloalkil-3-fenoxipropán pszichotróp gyógyszerek elõállítására alkalmas származékai

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Publication number
HUE026549T2
HUE026549T2 HUE06744550A HUE06744550A HUE026549T2 HU E026549 T2 HUE026549 T2 HU E026549T2 HU E06744550 A HUE06744550 A HU E06744550A HU E06744550 A HUE06744550 A HU E06744550A HU E026549 T2 HUE026549 T2 HU E026549T2
Authority
HU
Hungary
Prior art keywords
phenoxypropane
azacycloalkyl
derivatives
useful
preparation
Prior art date
Application number
HUE06744550A
Other languages
English (en)
Inventor
Isabelle Bertrand
Marc Capet
Jeanne-Marie Lecomte
Nicolas Levoin
Xavier Ligneau
Olivia Poupardin-Olivier
Philippe Robert
Jean-Charles Schwartz
Olivier Labeeuw
Original Assignee
Bioprojet Soc Civ
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from EP05290950A external-priority patent/EP1717234A1/en
Application filed by Bioprojet Soc Civ filed Critical Bioprojet Soc Civ
Publication of HUE026549T2 publication Critical patent/HUE026549T2/hu

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    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
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    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
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    • C—CHEMISTRY; METALLURGY
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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links

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HUE06744550A 2005-04-29 2006-04-25 1-N-azacikloalkil-3-fenoxipropán pszichotróp gyógyszerek elõállítására alkalmas származékai HUE026549T2 (hu)

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EP05290950A EP1717234A1 (en) 2005-04-29 2005-04-29 Phenoxypropylpiperidines and -pyrrolidines and their use as histamine H3-receptor ligands
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ES2563065T3 (es) 2016-03-10
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AU2006242950B2 (en) 2013-01-10
BRPI0612957B8 (pt) 2021-05-25
US8076329B2 (en) 2011-12-13
SI1874746T1 (sl) 2016-03-31
NZ562873A (en) 2011-03-31
KR20080005997A (ko) 2008-01-15
BRPI0612957A2 (pt) 2010-12-07
US20090111808A1 (en) 2009-04-30
EA200702363A1 (ru) 2008-04-28
KR101291575B1 (ko) 2013-08-08
PL1874746T3 (pl) 2016-06-30
JP2008539218A (ja) 2008-11-13
EP1874746A2 (en) 2008-01-09
CN101258138B (zh) 2013-06-12
BRPI0612957B1 (pt) 2020-10-27
WO2006117609A3 (en) 2007-03-22
CA2606262A1 (en) 2006-11-09
EA019594B1 (ru) 2014-04-30
EP1717235A3 (en) 2007-02-28
NO20075624L (no) 2007-11-28
MA29399B1 (fr) 2008-04-01
TNSN07393A1 (fr) 2009-03-17
SG162732A1 (en) 2010-07-29
WO2006117609A2 (en) 2006-11-09
EP1874746B1 (en) 2015-11-18
CN101258138A (zh) 2008-09-03
PT1874746E (pt) 2016-03-22
DK1874746T3 (en) 2016-02-15
EP1717235A2 (en) 2006-11-02
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