HU190507B - Process for production of azetidinil sulpfon acids and analogic substances - Google Patents

Process for production of azetidinil sulpfon acids and analogic substances Download PDF

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Publication number
HU190507B
HU190507B HU833460A HU346083A HU190507B HU 190507 B HU190507 B HU 190507B HU 833460 A HU833460 A HU 833460A HU 346083 A HU346083 A HU 346083A HU 190507 B HU190507 B HU 190507B
Authority
HU
Hungary
Prior art keywords
salt
acid
mmol
amino
formula
Prior art date
Application number
HU833460A
Other languages
German (de)
English (en)
Hungarian (hu)
Inventor
William A Slusarchyk
David R Kronenthal
Original Assignee
E.R.Squibb And Sons Inc,Us
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by E.R.Squibb And Sons Inc,Us filed Critical E.R.Squibb And Sons Inc,Us
Publication of HU190507B publication Critical patent/HU190507B/hu

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D205/00Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
    • C07D205/02Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
    • C07D205/06Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D205/08Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D205/00Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
    • C07D205/02Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
    • C07D205/06Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D205/08Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams
    • C07D205/085Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams with a nitrogen atom directly attached in position 3
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02ATECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Cephalosporin Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
HU833460A 1982-10-06 1983-10-06 Process for production of azetidinil sulpfon acids and analogic substances HU190507B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US43317582A 1982-10-06 1982-10-06

Publications (1)

Publication Number Publication Date
HU190507B true HU190507B (en) 1986-09-29

Family

ID=23719123

Family Applications (1)

Application Number Title Priority Date Filing Date
HU833460A HU190507B (en) 1982-10-06 1983-10-06 Process for production of azetidinil sulpfon acids and analogic substances

Country Status (27)

Country Link
JP (1) JPS5988462A (ru)
KR (1) KR900005132B1 (ru)
AU (1) AU568312B2 (ru)
BE (1) BE897883A (ru)
CA (1) CA1253501A (ru)
CH (1) CH658858A5 (ru)
DD (1) DD222016A5 (ru)
DE (1) DE3336262A1 (ru)
DK (1) DK457983A (ru)
ES (1) ES8504814A1 (ru)
FI (1) FI833631A (ru)
FR (1) FR2534253B1 (ru)
GB (1) GB2129428B (ru)
GR (1) GR79704B (ru)
HU (1) HU190507B (ru)
IE (1) IE56600B1 (ru)
IL (1) IL69917A (ru)
IT (1) IT1171722B (ru)
LU (1) LU85033A1 (ru)
NL (1) NL8303410A (ru)
NO (1) NO833626L (ru)
NZ (1) NZ205642A (ru)
PH (1) PH24175A (ru)
PT (1) PT77458B (ru)
SE (1) SE8305509L (ru)
SU (1) SU1318146A3 (ru)
ZA (1) ZA837491B (ru)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0135194A1 (en) * 1983-09-16 1985-03-27 Takeda Chemical Industries, Ltd. Azetidinones and their production
WO1985004876A1 (en) * 1984-04-24 1985-11-07 Takeda Chemical Industries, Ltd. 2-azetidinone derivatives and process for their preparation
US4581170A (en) * 1984-08-03 1986-04-08 E. R. Squibb & Sons, Inc. N-hydroxyl protecting groups and process and intermediates for the preparation of 3-acylamino-1-hydroxy-2-azetidinones
EP0171064B1 (en) * 1984-08-06 1995-07-12 Fujisawa Pharmaceutical Co., Ltd. Azetidinone derivative and processes for production thereof
UY34585A (es) 2012-01-24 2013-09-02 Aicuris Gmbh & Co Kg Compuestos b-lactámicos sustituidos con amidina, su preparación y uso

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4337197A (en) * 1980-10-31 1982-06-29 E. R. Squibb & Sons, Inc. O-sulfated β-lactam hydroxamic acids and intermediates

Also Published As

Publication number Publication date
IL69917A (en) 1987-10-20
AU568312B2 (en) 1987-12-24
GR79704B (ru) 1984-10-31
KR900005132B1 (ko) 1990-07-20
SE8305509D0 (sv) 1983-10-06
BE897883A (fr) 1984-03-30
ES526282A0 (es) 1985-04-16
FI833631A0 (fi) 1983-10-06
JPS5988462A (ja) 1984-05-22
IE832354L (en) 1984-04-06
IE56600B1 (en) 1991-10-09
AU1993983A (en) 1984-04-12
LU85033A1 (fr) 1984-05-10
FR2534253A1 (fr) 1984-04-13
PH24175A (en) 1990-03-22
SU1318146A3 (ru) 1987-06-15
DE3336262A1 (de) 1984-04-12
NO833626L (no) 1984-04-09
CH658858A5 (fr) 1986-12-15
ES8504814A1 (es) 1985-04-16
KR840006337A (ko) 1984-11-29
PT77458A (en) 1983-11-01
ZA837491B (en) 1984-06-27
DK457983D0 (da) 1983-10-04
GB8326626D0 (en) 1983-11-09
NL8303410A (nl) 1984-05-01
DK457983A (da) 1984-04-07
IT8323172A0 (it) 1983-10-06
FI833631A (fi) 1984-04-07
SE8305509L (sv) 1984-04-07
NZ205642A (en) 1986-08-08
IL69917A0 (en) 1984-01-31
GB2129428B (en) 1986-03-19
FR2534253B1 (fr) 1985-07-26
IT1171722B (it) 1987-06-10
CA1253501A (en) 1989-05-02
DD222016A5 (de) 1985-05-08
GB2129428A (en) 1984-05-16
PT77458B (en) 1986-02-26

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Legal Events

Date Code Title Description
HU90 Patent valid on 900628
HMM4 Cancellation of final prot. due to non-payment of fee