HU176452B - Process for preparing beta-daunosaminyl-nucleosides and pharmaceutical preparations containing thereof - Google Patents

Process for preparing beta-daunosaminyl-nucleosides and pharmaceutical preparations containing thereof Download PDF

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Publication number
HU176452B
HU176452B HU76FA995A HUFA000995A HU176452B HU 176452 B HU176452 B HU 176452B HU 76FA995 A HU76FA995 A HU 76FA995A HU FA000995 A HUFA000995 A HU FA000995A HU 176452 B HU176452 B HU 176452B
Authority
HU
Hungary
Prior art keywords
daunosaminyl
formula
pharmaceutical composition
compound
trifluoroacetyl
Prior art date
Application number
HU76FA995A
Other languages
English (en)
Hungarian (hu)
Inventor
Ettore Lazzari
Marco Aurelio Di
Federico Arcamone
Original Assignee
Farmaceutici Italia
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Farmaceutici Italia filed Critical Farmaceutici Italia
Publication of HU176452B publication Critical patent/HU176452B/hu

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/06—Pyrimidine radicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/16—Purine radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Glass Compositions (AREA)
HU76FA995A 1975-12-18 1976-12-13 Process for preparing beta-daunosaminyl-nucleosides and pharmaceutical preparations containing thereof HU176452B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB51967/75A GB1531469A (en) 1975-12-18 1975-12-18 Daunosamine nucleosides

Publications (1)

Publication Number Publication Date
HU176452B true HU176452B (en) 1981-03-28

Family

ID=10462134

Family Applications (1)

Application Number Title Priority Date Filing Date
HU76FA995A HU176452B (en) 1975-12-18 1976-12-13 Process for preparing beta-daunosaminyl-nucleosides and pharmaceutical preparations containing thereof

Country Status (8)

Country Link
US (1) US4067968A (en:Method)
JP (1) JPS5277074A (en:Method)
CH (1) CH629220A5 (en:Method)
DE (1) DE2657376A1 (en:Method)
FR (1) FR2335233A1 (en:Method)
GB (1) GB1531469A (en:Method)
HU (1) HU176452B (en:Method)
SU (2) SU683629A3 (en:Method)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4201773A (en) * 1978-07-26 1980-05-06 The United States Of America As Represented By The Department Of Health, Education And Welfare 7-O-(2,6-Dideoxy-α-L-lyxo-hexopyranosyl)-daunomycinone, desmethoxy daunomycinone, adriamycinone, and carminomycinone
US4562177A (en) * 1982-08-17 1985-12-31 The Ohio State University Research Foundation 3'-Amino-2' halo-anthracycline antibiotics

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3803124A (en) * 1968-04-12 1974-04-09 Farmaceutici It Soc Process for the preparation of adriamycin and adriamycinone and adriamycin derivatives
SU452961A3 (ru) * 1969-04-11 1974-12-05 Шеринг Аг. (Фирма) Способ получени пиримидиннуклеозидов
US3654262A (en) * 1969-08-21 1972-04-04 Merck & Co Inc 3-deoxy-3-c-lower alkyl glycosides and nucleosides
US3721664A (en) * 1970-01-27 1973-03-20 Hoffmann La Roche Preparation of 5-cytosine nucleosides
DE2012888C3 (de) * 1970-03-14 1981-04-02 Schering Ag, 1000 Berlin Und 4619 Bergkamen Verfahren zur Herstellung von 5-Azapyrimidinnucleosiden

Also Published As

Publication number Publication date
JPS5277074A (en) 1977-06-29
US4067968A (en) 1978-01-10
SU683629A3 (ru) 1979-08-30
DE2657376A1 (de) 1977-06-30
CH629220A5 (de) 1982-04-15
SU715024A3 (ru) 1980-02-05
FR2335233B1 (en:Method) 1980-03-14
GB1531469A (en) 1978-11-08
FR2335233A1 (fr) 1977-07-15

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