HRP20181710T1 - Uporaba derivata benzimidazol-prolina - Google Patents

Uporaba derivata benzimidazol-prolina

Info

Publication number
HRP20181710T1
HRP20181710T1 HRP20181710TT HRP20181710T HRP20181710T1 HR P20181710 T1 HRP20181710 T1 HR P20181710T1 HR P20181710T T HRP20181710T T HR P20181710TT HR P20181710 T HRP20181710 T HR P20181710T HR P20181710 T1 HRP20181710 T1 HR P20181710T1
Authority
HR
Croatia
Prior art keywords
benzimidazole
proline derivatives
proline
derivatives
Prior art date
Application number
HRP20181710TT
Other languages
English (en)
Inventor
Christoph Boss
Catherine Roch
Christine Brotschi
Markus Gude
Bibia Heidmann
Francois Jenck
Thierry Sifferlen
Michel Steiner
Jodi T. Williams
Original Assignee
Idorsia Pharmaceuticals Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Idorsia Pharmaceuticals Ltd filed Critical Idorsia Pharmaceuticals Ltd
Publication of HRP20181710T1 publication Critical patent/HRP20181710T1/hr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4164—1,3-Diazoles
    • A61K31/4178—1,3-Diazoles not condensed 1,3-diazoles and containing further heterocyclic rings, e.g. pilocarpine, nitrofurantoin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4192—1,2,3-Triazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
HRP20181710TT 2013-12-04 2018-10-18 Uporaba derivata benzimidazol-prolina HRP20181710T1 (hr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
IB2013060630 2013-12-04
PCT/IB2014/066548 WO2015083094A1 (en) 2013-12-04 2014-12-03 Use of benzimidazole-proline derivatives
EP14827273.5A EP3077391B1 (en) 2013-12-04 2014-12-03 Use of benzimidazole-proline derivatives

Publications (1)

Publication Number Publication Date
HRP20181710T1 true HRP20181710T1 (hr) 2018-12-28

Family

ID=52347368

Family Applications (1)

Application Number Title Priority Date Filing Date
HRP20181710TT HRP20181710T1 (hr) 2013-12-04 2018-10-18 Uporaba derivata benzimidazol-prolina

Country Status (29)

Country Link
US (1) US9914721B2 (hr)
EP (1) EP3077391B1 (hr)
JP (1) JP6421185B2 (hr)
KR (1) KR102330133B1 (hr)
CN (1) CN105873921B (hr)
AU (1) AU2014358766B2 (hr)
CA (1) CA2930053A1 (hr)
CL (1) CL2016001349A1 (hr)
CY (1) CY1121089T1 (hr)
DK (1) DK3077391T3 (hr)
EA (1) EA029725B1 (hr)
ES (1) ES2696708T3 (hr)
HK (1) HK1225734B (hr)
HR (1) HRP20181710T1 (hr)
HU (1) HUE040555T2 (hr)
IL (1) IL245914B (hr)
LT (1) LT3077391T (hr)
MA (1) MA39165A1 (hr)
MX (1) MX366642B (hr)
MY (1) MY179605A (hr)
PH (1) PH12016500985A1 (hr)
PL (1) PL3077391T3 (hr)
PT (1) PT3077391T (hr)
SA (1) SA516371253B1 (hr)
SI (1) SI3077391T1 (hr)
TR (1) TR201815342T4 (hr)
UA (1) UA116053C2 (hr)
WO (1) WO2015083094A1 (hr)
ZA (1) ZA201604502B (hr)

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Also Published As

Publication number Publication date
AU2014358766B2 (en) 2019-01-17
IL245914A0 (en) 2016-08-02
CA2930053A1 (en) 2015-06-11
MX2016007313A (es) 2016-09-07
ES2696708T3 (es) 2019-01-17
MA39165A1 (fr) 2017-10-31
SA516371253B1 (ar) 2018-07-24
LT3077391T (lt) 2018-10-25
JP6421185B2 (ja) 2018-11-07
AU2014358766A1 (en) 2016-07-21
PL3077391T3 (pl) 2019-01-31
US9914721B2 (en) 2018-03-13
EA201600434A1 (ru) 2016-11-30
PH12016500985B1 (en) 2016-06-20
CN105873921B (zh) 2019-03-15
UA116053C2 (uk) 2018-01-25
HUE040555T2 (hu) 2019-03-28
IL245914B (en) 2019-09-26
HK1225734B (zh) 2017-09-15
PH12016500985A1 (en) 2016-06-20
ZA201604502B (en) 2019-07-31
CN105873921A (zh) 2016-08-17
EA029725B1 (ru) 2018-05-31
NZ721697A (en) 2021-09-24
PT3077391T (pt) 2018-11-26
EP3077391B1 (en) 2018-08-15
CL2016001349A1 (es) 2017-01-27
SI3077391T1 (sl) 2018-11-30
KR20160093686A (ko) 2016-08-08
MX366642B (es) 2019-07-17
DK3077391T3 (en) 2018-10-22
EP3077391A1 (en) 2016-10-12
TR201815342T4 (tr) 2018-11-21
CY1121089T1 (el) 2019-12-11
WO2015083094A1 (en) 2015-06-11
MY179605A (en) 2020-11-11
JP2016539157A (ja) 2016-12-15
US20170001985A1 (en) 2017-01-05
KR102330133B1 (ko) 2021-11-23

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