HRP20170653T1 - Postupak za pripremanje 1-([1,3]dioksolan-4-ilmetil)-1h-pirazol-3-ilamina - Google Patents
Postupak za pripremanje 1-([1,3]dioksolan-4-ilmetil)-1h-pirazol-3-ilamina Download PDFInfo
- Publication number
- HRP20170653T1 HRP20170653T1 HRP20170653TT HRP20170653T HRP20170653T1 HR P20170653 T1 HRP20170653 T1 HR P20170653T1 HR P20170653T T HRP20170653T T HR P20170653TT HR P20170653 T HRP20170653 T HR P20170653T HR P20170653 T1 HRP20170653 T1 HR P20170653T1
- Authority
- HR
- Croatia
- Prior art keywords
- formula
- image
- compound
- phenyl
- lithium
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/38—Nitrogen atoms
- C07D231/40—Acylated on said nitrogen atom
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/06—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Preparation Of Compounds By Using Micro-Organisms (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CN2012087380 | 2012-12-25 | ||
| EP13811542.3A EP2938609B1 (en) | 2012-12-25 | 2013-12-20 | Process for the preparation of 1-([1,3]dioxolan-4-ylmethyl)-1h-pyrazol-3-ylamine |
| PCT/EP2013/077563 WO2014102164A1 (en) | 2012-12-25 | 2013-12-20 | Process for the preparation of 1-([1,3]dioxolan-4-ylmethyl)-1h-pyrazol-3-ylamine |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| HRP20170653T1 true HRP20170653T1 (hr) | 2017-06-30 |
Family
ID=49876646
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| HRP20170653TT HRP20170653T1 (hr) | 2012-12-25 | 2013-12-20 | Postupak za pripremanje 1-([1,3]dioksolan-4-ilmetil)-1h-pirazol-3-ilamina |
Country Status (23)
| Country | Link |
|---|---|
| US (1) | US9388168B2 (enExample) |
| EP (1) | EP2938609B1 (enExample) |
| JP (1) | JP6297590B2 (enExample) |
| KR (1) | KR102122569B1 (enExample) |
| CN (1) | CN105051031B (enExample) |
| AU (1) | AU2013369473B2 (enExample) |
| BR (1) | BR112015015229B1 (enExample) |
| CA (1) | CA2896155C (enExample) |
| CY (1) | CY1119040T1 (enExample) |
| DK (1) | DK2938609T3 (enExample) |
| ES (1) | ES2629313T3 (enExample) |
| HR (1) | HRP20170653T1 (enExample) |
| HU (1) | HUE032621T2 (enExample) |
| IL (1) | IL239558A (enExample) |
| LT (1) | LT2938609T (enExample) |
| NZ (1) | NZ709362A (enExample) |
| PL (1) | PL2938609T3 (enExample) |
| PT (1) | PT2938609T (enExample) |
| RU (1) | RU2621725C2 (enExample) |
| SG (1) | SG11201504951TA (enExample) |
| SI (1) | SI2938609T1 (enExample) |
| WO (1) | WO2014102164A1 (enExample) |
| ZA (1) | ZA201504601B (enExample) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US11266630B2 (en) * | 2016-12-15 | 2022-03-08 | Hua Medicine (Shanghai) Ltd. | Oral preparation of glucokinase activator and preparation method therefor |
| CN113493442B (zh) * | 2020-04-03 | 2024-11-08 | 天津药物研究院有限公司 | 作为葡萄糖激酶活化剂的吡咯烷酮衍生物及其制备方法和用途 |
| US11813274B2 (en) | 2020-04-22 | 2023-11-14 | Hua Medicine (Shanghai) Ltd. | Treating untreated or treatment-resistant diabetes with glucokinase activator and sodium-glucose cotransporter-2 inhibitor |
| WO2021212360A1 (en) * | 2020-04-22 | 2021-10-28 | Hua Medicine (Shanghai) Ltd. | Treating untreated or treatment-resistant diabetes with glucokinase activator and sodium-glucose cotransporter-2 inhibitor |
| CN111732543A (zh) * | 2020-08-14 | 2020-10-02 | 浙江鼎龙科技有限公司 | 一种4,5-二氨基-1-(2-羟乙基)吡唑硫酸盐的制备方法 |
| CN113750100B (zh) * | 2021-08-31 | 2022-12-30 | 海南中济医药科技有限公司 | 一种含有多扎格列艾汀与西格列汀的药物组合物及其制备方法 |
| AR127064A1 (es) * | 2021-09-15 | 2023-12-13 | Hua Medicine Shanghai Ltd | Prodroga de derivados de pirrolidona como activador de glucoquinasa |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4160841A (en) * | 1977-01-31 | 1979-07-10 | Janssen Pharmaceutica, N.V. | Heterocyclic derivatives of 1-(1,3-dioxolan-2-ylmethyl)-1H-imidazoles |
| FR2748274B1 (fr) * | 1996-05-03 | 1998-06-12 | Oreal | Nouveaux diamino pyrazoles, leur synthese, compositions de teinture des fibres keratiniques les contenant, procede de teinture des fibres keratiniques |
| KR20100113518A (ko) * | 2008-01-18 | 2010-10-21 | 아스텔라스세이야쿠 가부시키가이샤 | 페닐아세트아미드 유도체 |
| US7741327B2 (en) * | 2008-04-16 | 2010-06-22 | Hoffmann-La Roche Inc. | Pyrrolidinone glucokinase activators |
| US8178689B2 (en) * | 2010-06-17 | 2012-05-15 | Hoffman-La Roche Inc. | Tricyclic compounds |
-
2013
- 2013-12-20 HU HUE13811542A patent/HUE032621T2/en unknown
- 2013-12-20 SI SI201330684A patent/SI2938609T1/sl unknown
- 2013-12-20 AU AU2013369473A patent/AU2013369473B2/en active Active
- 2013-12-20 NZ NZ709362A patent/NZ709362A/en unknown
- 2013-12-20 CN CN201380068179.8A patent/CN105051031B/zh active Active
- 2013-12-20 PT PT138115423T patent/PT2938609T/pt unknown
- 2013-12-20 ES ES13811542.3T patent/ES2629313T3/es active Active
- 2013-12-20 KR KR1020157019691A patent/KR102122569B1/ko active Active
- 2013-12-20 US US14/655,287 patent/US9388168B2/en active Active
- 2013-12-20 JP JP2015550041A patent/JP6297590B2/ja active Active
- 2013-12-20 DK DK13811542.3T patent/DK2938609T3/en active
- 2013-12-20 RU RU2015126911A patent/RU2621725C2/ru active
- 2013-12-20 PL PL13811542T patent/PL2938609T3/pl unknown
- 2013-12-20 LT LTEP13811542.3T patent/LT2938609T/lt unknown
- 2013-12-20 SG SG11201504951TA patent/SG11201504951TA/en unknown
- 2013-12-20 BR BR112015015229-5A patent/BR112015015229B1/pt active IP Right Grant
- 2013-12-20 HR HRP20170653TT patent/HRP20170653T1/hr unknown
- 2013-12-20 CA CA2896155A patent/CA2896155C/en active Active
- 2013-12-20 WO PCT/EP2013/077563 patent/WO2014102164A1/en not_active Ceased
- 2013-12-20 EP EP13811542.3A patent/EP2938609B1/en active Active
-
2015
- 2015-06-21 IL IL239558A patent/IL239558A/en active IP Right Grant
- 2015-06-25 ZA ZA2015/04601A patent/ZA201504601B/en unknown
-
2017
- 2017-07-10 CY CY20171100727T patent/CY1119040T1/el unknown
Also Published As
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| HRP20170653T1 (hr) | Postupak za pripremanje 1-([1,3]dioksolan-4-ilmetil)-1h-pirazol-3-ilamina | |
| JP2015509939A5 (enExample) | ||
| RU2014137470A (ru) | Способы и соединения, которые можно использовать для синтеза антагонистов рецепторов орексина-2 | |
| AR082891A1 (es) | Di-azetidinil diamidas como inhibidores de monoacilglicerol lipasas | |
| AR073892A1 (es) | Proceso de preparacion de inhibidores de sglt | |
| JP2015500335A5 (enExample) | ||
| HRP20140668T1 (hr) | Postupak proizvodnje prasugrel hidroklorida visoke äśistoä†e | |
| JP2017522357A5 (enExample) | ||
| ES2512591T3 (es) | Método de producción de 2'-desoxi-5-azacitidina (decitabina) | |
| BR112014004210B1 (pt) | processo para a preparação de derivados de diamida do ácido antranílico substituídos com tetrazole por reação de benzoxazinonas com aminas | |
| HRP20150885T1 (hr) | Postupak za pripremu 4-{4-[({[4-kloro-3-(trifluorometil)-fenil]amino}karbonil)amino]-3-fluorofenoksi}-n-metilpiridin-2-karboksamida, njegovih soli i monohidrata | |
| BR112014000471B1 (pt) | processo para preparo de derivados de diamida de ácido antranílico substituídos com tetrazol por meio da reação de ácidos pirazóis com ésteres antranílicos | |
| RU2014128826A (ru) | Дисоли малоновой кислоты и способ получения малонилдигалогенидов | |
| JP2016503812A5 (enExample) | ||
| RU2012122367A (ru) | Способ получения простагландинов и промежуточные соединения для их получения | |
| EP2275415A2 (en) | Method for producing aminothiazole derivative and production intermediate | |
| CA2761399C (en) | Process for the production of bendamustine alkyl ester, bendamustine, and derivatives thereof | |
| WO2012174685A1 (zh) | 一种2-取代-2h-1,2,3-三氮唑衍生物的制备方法 | |
| HRP20161563T1 (hr) | Postupak za dobivanje 5-fluor-1h-pirazola | |
| AR092070A1 (es) | Proceso para la preparacion de inhibidores de quinasa c-fms | |
| RU2004139100A (ru) | Способ получения производных пенама из производных цефама | |
| CN109232428A (zh) | 一种吡唑基偶氮苯酚化合物及其合成、衍生 | |
| JP2010516779A5 (enExample) | ||
| ES2546059T3 (es) | Procedimiento para la preparación de 2,4-dioxotetrahidrofurano-3-carboxilatos | |
| PH12014501704B1 (en) | Method for preparing compound by novel michael addition reaction using water or various acids as additive |