HRP20080440B1 - Postupak za proizvodnju spoja 5-alkoksi-4-hidroksimetilpirazola - Google Patents

Postupak za proizvodnju spoja 5-alkoksi-4-hidroksimetilpirazola

Info

Publication number
HRP20080440B1
HRP20080440B1 HRP20080440AA HRP20080440A HRP20080440B1 HR P20080440 B1 HRP20080440 B1 HR P20080440B1 HR P20080440A A HRP20080440A A HR P20080440AA HR P20080440 A HRP20080440 A HR P20080440A HR P20080440 B1 HRP20080440 B1 HR P20080440B1
Authority
HR
Croatia
Prior art keywords
alkoxy
production
group
compound
substituent
Prior art date
Application number
HRP20080440AA
Other languages
English (en)
Inventor
Yukio Uchida
Naoya Atsumi
Original Assignee
Ihara Chemical Industry Co., Ltd.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ihara Chemical Industry Co., Ltd. filed Critical Ihara Chemical Industry Co., Ltd.
Publication of HRP20080440A2 publication Critical patent/HRP20080440A2/hr
Publication of HRP20080440B1 publication Critical patent/HRP20080440B1/hr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/18—One oxygen or sulfur atom
    • C07D231/20—One oxygen atom attached in position 3 or 5
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/18—One oxygen or sulfur atom
    • C07D231/20—One oxygen atom attached in position 3 or 5
    • C07D231/22—One oxygen atom attached in position 3 or 5 with aryl radicals attached to ring nitrogen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Predloženi izum odnosi se na postupak za proizvodnju spoja 5-alkoksi-4-hidroksimetilpirazola na jednostavan način i s dobrom učinkovitošću. Postupak za proizvodnju spoja 5-alkoksi-4-hidroksi-metilpirazola kojeg prikazuje opća formula (3)(u kojoj Rje supstituent kao što je alkilna skupina, supstituirana ili nesupstituirana skupina, ili slično, i Rje skupina koja privlači elektron) sa spojem kojeg prikazuje opća formula (2)L-R(2)(u kojoj L je izlazna skupina i Rje supstituent kao što je supstituirana ili nesupstituirana alkilna skupina ili slično) u prisutnosti baze i formaldehida.
HRP20080440AA 2006-02-14 2008-09-10 Postupak za proizvodnju spoja 5-alkoksi-4-hidroksimetilpirazola HRP20080440B1 (hr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2006037245 2006-02-14
PCT/JP2007/052184 WO2007094225A1 (ja) 2006-02-14 2007-02-08 ５－アルコキシ－４－ヒドロキシメチルピラゾール化合物の製造方法

Publications (2)

Publication Number Publication Date
HRP20080440A2 HRP20080440A2 (hr) 2009-02-28
HRP20080440B1 true HRP20080440B1 (hr) 2014-11-21

Family

ID=38371412

Family Applications (1)

Application Number Title Priority Date Filing Date
HRP20080440AA HRP20080440B1 (hr) 2006-02-14 2008-09-10 Postupak za proizvodnju spoja 5-alkoksi-4-hidroksimetilpirazola

Country Status (20)

Country Link
US (1) US7812175B2 (hr)
EP (1) EP1990336B1 (hr)
JP (1) JP5052495B2 (hr)
KR (1) KR101401139B1 (hr)
CN (2) CN101384556B (hr)
AR (1) AR059375A1 (hr)
AT (1) ATE544755T1 (hr)
AU (1) AU2007216034B2 (hr)
BR (1) BRPI0707801B1 (hr)
CA (1) CA2642308C (hr)
CR (1) CR10155A (hr)
ES (1) ES2381695T3 (hr)
HR (1) HRP20080440B1 (hr)
IL (1) IL192702A (hr)
NZ (2) NZ595579A (hr)
PL (1) PL1990336T3 (hr)
RU (1) RU2451677C2 (hr)
TW (1) TWI385155B (hr)
UA (1) UA90940C2 (hr)
WO (1) WO2007094225A1 (hr)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
UY34585A (es) 2012-01-24 2013-09-02 Aicuris Gmbh & Co Kg Compuestos b-lactámicos sustituidos con amidina, su preparación y uso
US20180230103A1 (en) 2015-11-16 2018-08-16 Lonza Ltd Method for preparation of 1-methyl-3-(trifluoromethyl)-1h-pyrazol-5-ol
TW201835036A (zh) 2017-02-27 2018-10-01 瑞士商隆薩有限公司 製備1-甲基-3-(三氟甲基)-1h-吡唑-5-醇的方法
KR20230053729A (ko) 2019-10-31 2023-04-21 구미아이 가가쿠 고교 가부시키가이샤 제초제 및 그 중간체의 제조방법
CN111574511A (zh) * 2020-06-28 2020-08-25 安徽久易农业股份有限公司 一种砜吡草唑的合成方法及其应用
CN114989142A (zh) * 2022-05-09 2022-09-02 沈阳万菱生物技术有限公司 一种吡唑类化合物的制备方法

Citations (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2004013106A1 (ja) * 2002-08-01 2004-02-12 Ihara Chemical Industry Co., Ltd. ピラゾール誘導体及びその製造方法
WO2004099157A1 (en) * 2003-05-07 2004-11-18 Pfizer Products Inc. Cannabinoid receptor ligands and uses thereof
WO2005085205A1 (ja) * 2004-03-05 2005-09-15 Nissan Chemical Industries, Ltd. 置換ピラゾール化合物および除草剤
WO2005095352A1 (ja) * 2004-03-31 2005-10-13 Ihara Chemical Industry Co., Ltd. ５－ヒドロキシ－４－チオメチルピラゾール化合物の製造方法
WO2006123088A2 (en) * 2005-05-18 2006-11-23 Syngenta Limited 4- (thiazol-2-ylthioalkyl) -pyrazoles and their use as herbicides

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5133556B2 (hr) 1974-03-01 1976-09-20
JPH10287654A (ja) 1997-04-11 1998-10-27 Nissan Chem Ind Ltd ピラゾロン誘導体及び除草剤
TW200423930A (en) * 2003-02-18 2004-11-16 Hoffmann La Roche Non-nucleoside reverse transcriptase inhibitors

Patent Citations (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2004013106A1 (ja) * 2002-08-01 2004-02-12 Ihara Chemical Industry Co., Ltd. ピラゾール誘導体及びその製造方法
WO2004099157A1 (en) * 2003-05-07 2004-11-18 Pfizer Products Inc. Cannabinoid receptor ligands and uses thereof
WO2005085205A1 (ja) * 2004-03-05 2005-09-15 Nissan Chemical Industries, Ltd. 置換ピラゾール化合物および除草剤
WO2005095352A1 (ja) * 2004-03-31 2005-10-13 Ihara Chemical Industry Co., Ltd. ５－ヒドロキシ－４－チオメチルピラゾール化合物の製造方法
WO2006123088A2 (en) * 2005-05-18 2006-11-23 Syngenta Limited 4- (thiazol-2-ylthioalkyl) -pyrazoles and their use as herbicides

Also Published As

Publication number Publication date
AU2007216034A1 (en) 2007-08-23
IL192702A0 (en) 2009-02-11
US20090036688A1 (en) 2009-02-05
HRP20080440A2 (hr) 2009-02-28
NZ570495A (en) 2011-10-28
EP1990336B1 (en) 2012-02-08
EP1990336A4 (en) 2010-12-29
NZ595579A (en) 2013-03-28
ES2381695T3 (es) 2012-05-30
RU2008136892A (ru) 2010-03-20
CN102659683B (zh) 2014-11-12
PL1990336T3 (pl) 2012-07-31
KR101401139B1 (ko) 2014-05-29
TW200804296A (en) 2008-01-16
WO2007094225A1 (ja) 2007-08-23
TWI385155B (zh) 2013-02-11
UA90940C2 (ru) 2010-06-10
JP5052495B2 (ja) 2012-10-17
AR059375A1 (es) 2008-03-26
JPWO2007094225A1 (ja) 2009-07-02
WO2007094225A9 (ja) 2007-09-27
CA2642308C (en) 2013-12-17
CN101384556B (zh) 2012-06-20
AU2007216034B2 (en) 2011-08-04
KR20080093445A (ko) 2008-10-21
IL192702A (en) 2012-08-30
CA2642308A1 (en) 2007-08-23
US7812175B2 (en) 2010-10-12
RU2451677C2 (ru) 2012-05-27
CN102659683A (zh) 2012-09-12
BRPI0707801B1 (pt) 2018-01-16
BRPI0707801A2 (pt) 2011-05-10
ATE544755T1 (de) 2012-02-15
CR10155A (es) 2008-09-23
EP1990336A1 (en) 2008-11-12
CN101384556A (zh) 2009-03-11

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