HRP20000653A2 - Azabicyclic 5ht1 receptor ligands - Google Patents
Azabicyclic 5ht1 receptor ligands Download PDFInfo
- Publication number
- HRP20000653A2 HRP20000653A2 HR20000653A HRP20000653A HRP20000653A2 HR P20000653 A2 HRP20000653 A2 HR P20000653A2 HR 20000653 A HR20000653 A HR 20000653A HR P20000653 A HRP20000653 A HR P20000653A HR P20000653 A2 HRP20000653 A2 HR P20000653A2
- Authority
- HR
- Croatia
- Prior art keywords
- octahydro
- benzo
- pyrido
- isoxazol
- cis
- Prior art date
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- 239000003446 ligand Substances 0.000 title description 3
- 102000035038 5-HT1 receptors Human genes 0.000 title description 2
- 108091005478 5-HT1 receptors Proteins 0.000 title description 2
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Classifications
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- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
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Landscapes
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- Gynecology & Obstetrics (AREA)
- Urology & Nephrology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Luminescent Compositions (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US8123798P | 1998-04-09 | 1998-04-09 | |
| PCT/IB1999/000457 WO1999052907A1 (en) | 1998-04-09 | 1999-03-18 | Azabicyclic 5ht1 receptor ligands |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| HRP20000653A2 true HRP20000653A2 (en) | 2001-04-30 |
Family
ID=22162936
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| HR20000653A HRP20000653A2 (en) | 1998-04-09 | 2000-10-04 | Azabicyclic 5ht1 receptor ligands |
Country Status (41)
| Country | Link |
|---|---|
| US (2) | US6525048B1 (zh) |
| EP (1) | EP1070065B1 (zh) |
| JP (1) | JP3496759B2 (zh) |
| KR (1) | KR100378931B1 (zh) |
| CN (1) | CN1117092C (zh) |
| AP (1) | AP1175A (zh) |
| AR (1) | AR015751A1 (zh) |
| AT (1) | ATE248838T1 (zh) |
| AU (1) | AU749254B2 (zh) |
| BG (1) | BG104915A (zh) |
| BR (1) | BR9909522A (zh) |
| CA (1) | CA2327782A1 (zh) |
| CO (1) | CO5080727A1 (zh) |
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| DZ (1) | DZ2756A1 (zh) |
| EA (1) | EA003400B1 (zh) |
| ES (1) | ES2204154T3 (zh) |
| HK (1) | HK1035719A1 (zh) |
| HR (1) | HRP20000653A2 (zh) |
| HU (1) | HUP0102400A3 (zh) |
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| TR (1) | TR200002932T2 (zh) |
| TW (1) | TW555758B (zh) |
| WO (1) | WO1999052907A1 (zh) |
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Families Citing this family (15)
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|---|---|---|---|---|
| US6231833B1 (en) * | 1999-08-05 | 2001-05-15 | Pfizer Inc | 2,7-substituted octahydro-1H-pyrido[1,2-A]pyrazine derivatives as ligands for serotonin receptors |
| UA62015C2 (en) * | 1998-12-28 | 2003-12-15 | Pfizer Prod Inc | Benzoizoxazol derivatives, a pharmaceutical composition (variants) based thereon (variants) and a method for treatment (variants) |
| BR0014166A (pt) * | 1999-09-03 | 2002-05-14 | Lilly Co Eli | Método de utilização de inibidores de reabsorção de serotonina seletivo de rápido ataque para tratamento de disfunção sexual |
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| US6855729B2 (en) * | 2001-02-20 | 2005-02-15 | Timothy G. Dinan | Treatment of fibromyalgia and related fatigue syndromes using antagonists or partial agonists of 5HT1a receptors |
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| US5106849A (en) * | 1988-05-24 | 1992-04-21 | American Home Products Corporation | Use of aryl- and heteroaryl piperazinyl carboxamides in the treatment of various central nervous system disorders |
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| HUT71488A (en) * | 1991-09-25 | 1995-11-28 | Pfizer | Process for the production of neuroleptic 2-substituted perhydro-1-h-pyrido[1,2a]pyrazines and pharmaceuticals compositions containing the same |
| US5262428A (en) * | 1992-03-13 | 1993-11-16 | Wake Forest University | Biologically active tropane derivatives |
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| US5614523A (en) * | 1995-01-17 | 1997-03-25 | Eli Lilly And Company | Compounds having effects on serotonin-related systems |
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