HN2002000197A - Proceso para la produccion de quinazolinas - Google Patents

Proceso para la produccion de quinazolinas

Info

Publication number
HN2002000197A
HN2002000197A HN2002000197A HN2002000197A HN2002000197A HN 2002000197 A HN2002000197 A HN 2002000197A HN 2002000197 A HN2002000197 A HN 2002000197A HN 2002000197 A HN2002000197 A HN 2002000197A HN 2002000197 A HN2002000197 A HN 2002000197A
Authority
HN
Honduras
Prior art keywords
quinazolins
production
useful
compounds
quinazoline compounds
Prior art date
Application number
HN2002000197A
Other languages
English (en)
Original Assignee
Inc Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Inc Pfizer filed Critical Inc Pfizer
Publication of HN2002000197A publication Critical patent/HN2002000197A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/08Drugs for disorders of the urinary system of the prostate
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D213/00Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/24Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D213/54Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D213/57Nitriles

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Urology & Nephrology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Pyridine Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)

Abstract

LA PRESENTE INVENCION SE REFIERE A UN NUEVO PROCESO PARA PRODUCIR COMPUESTOS DE QUINAZOLINA QUE SON UTILES EN TERAPIA.- MAS ESPECIFICAMENTE, LOS COMPUESTOS SON ÚTILES EN EL TRATAMIENTO DE LA HIPERPLASIA PROSTATICA BENIGNA. COMPUESTOS DE QUINOLINA Y QUINAZOLINA SUSTITUTIDAS (VER FORMULA)
HN2002000197A 2001-08-01 2002-07-29 Proceso para la produccion de quinazolinas HN2002000197A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB0118752.5A GB0118752D0 (en) 2001-08-01 2001-08-01 Process for the production of quinazolines

Publications (1)

Publication Number Publication Date
HN2002000197A true HN2002000197A (es) 2003-02-27

Family

ID=9919612

Family Applications (1)

Application Number Title Priority Date Filing Date
HN2002000197A HN2002000197A (es) 2001-08-01 2002-07-29 Proceso para la produccion de quinazolinas

Country Status (27)

Country Link
US (1) US7026479B2 (es)
EP (1) EP1412331B1 (es)
JP (1) JP2005501054A (es)
KR (1) KR20040019097A (es)
CN (1) CN1533378A (es)
AP (1) AP1299A (es)
AR (1) AR036204A1 (es)
AT (1) ATE323677T1 (es)
BR (1) BR0211670A (es)
CA (1) CA2451075A1 (es)
CZ (1) CZ2004151A3 (es)
DE (1) DE60210778T2 (es)
DO (1) DOP2002000443A (es)
EG (1) EG23204A (es)
ES (1) ES2260457T3 (es)
GB (1) GB0118752D0 (es)
HN (1) HN2002000197A (es)
HU (1) HUP0401573A3 (es)
IL (1) IL158998A0 (es)
MX (1) MXPA04000978A (es)
PA (1) PA8550301A1 (es)
PE (1) PE20030346A1 (es)
PL (1) PL368520A1 (es)
RU (1) RU2261861C1 (es)
UY (1) UY27399A1 (es)
WO (1) WO2003011829A1 (es)
ZA (1) ZA200309043B (es)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2400339T3 (es) * 2002-07-15 2013-04-09 Symphony Evolution, Inc. Compuestos, composiciones farmacéuticas de los mismos y su uso en el tratamiento del cáncer
JP4638436B2 (ja) 2003-09-26 2011-02-23 エグゼリクシス, インコーポレイテッド c−Metモジュレーターおよびその使用
CA2565812C (en) * 2004-05-06 2012-03-13 Warner-Lambert Company Llc 4-phenylamino-quinazolin-6-yl-amides
WO2008015270A1 (en) * 2006-08-04 2008-02-07 Merz Pharma Gmbh & Co. Kgaa Pyrazolopyrimidines, a process for their preparation and their use as medicine
TWI577664B (zh) 2009-01-16 2017-04-11 艾克塞里克斯公司 N-(4-{〔6,7-雙(甲氧基)喹啉-4-基〕氧基}苯基)-n’-(4-氟苯基)環丙烷-1,1-二甲醯胺蘋果酸鹽、包含其之醫藥組合物及其用途
JP5795304B2 (ja) 2009-03-18 2015-10-14 レスバーロジックス コーポレイション 新規抗炎症剤
IN2012DN00352A (es) * 2009-06-16 2015-08-21 Bikam Pharmaceuticals Inc
UA108618C2 (uk) 2009-08-07 2015-05-25 Застосування c-met-модуляторів в комбінації з темозоломідом та/або променевою терапією для лікування раку
US9353063B2 (en) 2011-11-30 2016-05-31 Bikam Pharmaceuticals, Inc. Opsin-binding ligands, compositions and methods of use
CN104884427B (zh) * 2012-10-15 2016-09-07 雷斯韦洛吉克斯公司 可用于合成苯甲酰胺化合物的化合物
KR102662814B1 (ko) 2015-03-13 2024-05-03 리스버로직스 코퍼레이션 보체 관련 질환을 치료하기 위한 조성물 및 치료 방법

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8719378D0 (en) * 1987-08-15 1987-09-23 Pfizer Ltd Antiarrythmic agents
EP0894797A4 (en) * 1997-01-09 2001-08-16 Terumo Corp NEW AMID DERIVATIVES AND INTERMEDIATES ON YOUR SYNTHESIS

Also Published As

Publication number Publication date
EG23204A (en) 2004-07-31
GB0118752D0 (en) 2001-09-26
BR0211670A (pt) 2004-07-13
AR036204A1 (es) 2004-08-18
IL158998A0 (en) 2004-05-12
RU2261861C1 (ru) 2005-10-10
DE60210778T2 (de) 2007-01-04
AP2002002602A0 (en) 2002-09-30
ES2260457T3 (es) 2006-11-01
PE20030346A1 (es) 2003-04-05
AP1299A (en) 2004-09-06
ATE323677T1 (de) 2006-05-15
JP2005501054A (ja) 2005-01-13
CZ2004151A3 (cs) 2005-01-12
EP1412331B1 (en) 2006-04-19
CA2451075A1 (en) 2003-02-13
PL368520A1 (en) 2005-04-04
KR20040019097A (ko) 2004-03-04
PA8550301A1 (es) 2003-09-05
DE60210778D1 (de) 2006-05-24
US20030100753A1 (en) 2003-05-29
RU2004102692A (ru) 2005-07-10
EP1412331A1 (en) 2004-04-28
US7026479B2 (en) 2006-04-11
HUP0401573A3 (en) 2005-06-28
CN1533378A (zh) 2004-09-29
UY27399A1 (es) 2003-02-28
WO2003011829A1 (en) 2003-02-13
MXPA04000978A (es) 2004-04-20
ZA200309043B (en) 2004-11-22
DOP2002000443A (es) 2003-02-15
HUP0401573A2 (hu) 2005-01-28

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