HN2002000197A - Proceso para la produccion de quinazolinas - Google Patents

Proceso para la produccion de quinazolinas

Info

Publication number
HN2002000197A
HN2002000197A HN2002000197A HN2002000197A HN2002000197A HN 2002000197 A HN2002000197 A HN 2002000197A HN 2002000197 A HN2002000197 A HN 2002000197A HN 2002000197 A HN2002000197 A HN 2002000197A HN 2002000197 A HN2002000197 A HN 2002000197A
Authority
HN
Honduras
Prior art keywords
quinazolins
production
useful
compounds
quinazoline compounds
Prior art date
Application number
HN2002000197A
Other languages
English (en)
Original Assignee
Inc Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Inc Pfizer filed Critical Inc Pfizer
Publication of HN2002000197A publication Critical patent/HN2002000197A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/08Drugs for disorders of the urinary system of the prostate
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D213/00Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/24Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D213/54Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D213/57Nitriles

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Urology & Nephrology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pyridine Compounds (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)

Abstract

LA PRESENTE INVENCION SE REFIERE A UN NUEVO PROCESO PARA PRODUCIR COMPUESTOS DE QUINAZOLINA QUE SON UTILES EN TERAPIA.- MAS ESPECIFICAMENTE, LOS COMPUESTOS SON ÚTILES EN EL TRATAMIENTO DE LA HIPERPLASIA PROSTATICA BENIGNA. COMPUESTOS DE QUINOLINA Y QUINAZOLINA SUSTITUTIDAS (VER FORMULA)
HN2002000197A 2001-08-01 2002-07-29 Proceso para la produccion de quinazolinas HN2002000197A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB0118752.5A GB0118752D0 (en) 2001-08-01 2001-08-01 Process for the production of quinazolines

Publications (1)

Publication Number Publication Date
HN2002000197A true HN2002000197A (es) 2003-02-27

Family

ID=9919612

Family Applications (1)

Application Number Title Priority Date Filing Date
HN2002000197A HN2002000197A (es) 2001-08-01 2002-07-29 Proceso para la produccion de quinazolinas

Country Status (27)

Country Link
US (1) US7026479B2 (es)
EP (1) EP1412331B1 (es)
JP (1) JP2005501054A (es)
KR (1) KR20040019097A (es)
CN (1) CN1533378A (es)
AP (1) AP1299A (es)
AR (1) AR036204A1 (es)
AT (1) ATE323677T1 (es)
BR (1) BR0211670A (es)
CA (1) CA2451075A1 (es)
CZ (1) CZ2004151A3 (es)
DE (1) DE60210778T2 (es)
DO (1) DOP2002000443A (es)
EG (1) EG23204A (es)
ES (1) ES2260457T3 (es)
GB (1) GB0118752D0 (es)
HN (1) HN2002000197A (es)
HU (1) HUP0401573A3 (es)
IL (1) IL158998A0 (es)
MX (1) MXPA04000978A (es)
PA (1) PA8550301A1 (es)
PE (1) PE20030346A1 (es)
PL (1) PL368520A1 (es)
RU (1) RU2261861C1 (es)
UY (1) UY27399A1 (es)
WO (1) WO2003011829A1 (es)
ZA (1) ZA200309043B (es)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2280003B1 (en) * 2002-07-15 2014-04-02 Symphony Evolution, Inc. Process for preparing receptor-type kinase modulators
SI2392564T1 (sl) * 2003-09-26 2014-02-28 Exelixis, Inc. c-Met modulatorji in postopki uporabe
JP4205757B2 (ja) 2004-05-06 2009-01-07 ワーナー−ランバート カンパニー リミテッド ライアビリティー カンパニー 4−フェニルアミノ−キナゾリン−6−イル−アミド
BRPI0714622A2 (pt) * 2006-08-04 2013-04-30 Merz Pharma Gmbh & Co Kgaa pirazolopirimidinas substituÍdas, processo para sua preparaÇço e seu uso como medicamento
CA2995880C (en) 2009-01-16 2021-01-05 Exelixis, Inc. Processes for preparing n-(4-{[6,7-bis(methyloxy)quinolin-4-yl]oxy}phenyl)-n'-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide
US9238640B2 (en) 2009-03-18 2016-01-19 Resverlogix Corp. Anti-inflammatory agents
IN2012DN00352A (es) * 2009-06-16 2015-08-21 Bikam Pharmaceuticals Inc
UA108618C2 (uk) 2009-08-07 2015-05-25 Застосування c-met-модуляторів в комбінації з темозоломідом та/або променевою терапією для лікування раку
EP2785346A4 (en) 2011-11-30 2015-04-29 Bikam Pharmaceuticals Inc OPSINBINDING LIGANDS, COMPOSITIONS THEREOF, AND METHOD OF USE THEREOF
PT2906531T (pt) * 2012-10-15 2018-02-06 Resverlogix Corp Compostos úteis na síntese de compostos de benzamida
JP6903585B2 (ja) 2015-03-13 2021-07-14 レスバーロジックス コーポレイション 補体関連疾患の治療のための組成物および治療方法

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8719378D0 (en) * 1987-08-15 1987-09-23 Pfizer Ltd Antiarrythmic agents
EP0894797A4 (en) * 1997-01-09 2001-08-16 Terumo Corp NEW AMID DERIVATIVES AND INTERMEDIATES ON YOUR SYNTHESIS

Also Published As

Publication number Publication date
ES2260457T3 (es) 2006-11-01
PE20030346A1 (es) 2003-04-05
PL368520A1 (en) 2005-04-04
MXPA04000978A (es) 2004-04-20
BR0211670A (pt) 2004-07-13
IL158998A0 (en) 2004-05-12
AP2002002602A0 (en) 2002-09-30
US7026479B2 (en) 2006-04-11
CN1533378A (zh) 2004-09-29
JP2005501054A (ja) 2005-01-13
CA2451075A1 (en) 2003-02-13
DE60210778D1 (de) 2006-05-24
DE60210778T2 (de) 2007-01-04
HUP0401573A2 (hu) 2005-01-28
EP1412331B1 (en) 2006-04-19
AP1299A (en) 2004-09-06
US20030100753A1 (en) 2003-05-29
EG23204A (en) 2004-07-31
AR036204A1 (es) 2004-08-18
UY27399A1 (es) 2003-02-28
RU2261861C1 (ru) 2005-10-10
DOP2002000443A (es) 2003-02-15
RU2004102692A (ru) 2005-07-10
ZA200309043B (en) 2004-11-22
GB0118752D0 (en) 2001-09-26
ATE323677T1 (de) 2006-05-15
EP1412331A1 (en) 2004-04-28
WO2003011829A1 (en) 2003-02-13
CZ2004151A3 (cs) 2005-01-12
KR20040019097A (ko) 2004-03-04
HUP0401573A3 (en) 2005-06-28
PA8550301A1 (es) 2003-09-05

Similar Documents

Publication Publication Date Title
UY27234A1 (es) Inhibidores novedosos de tirosina cinasa
LU92338I2 (fr) Enzalutamide et ses sels pharmaceutiquement acceptables (XTANDI)
NO20091661L (no) Anvendelse av pegylert IL-10 for a behandle kreft
HN2002000197A (es) Proceso para la produccion de quinazolinas
WO2008046083A3 (en) Use of oxindole compounds as therapeutic agents
CR7182A (es) Benzoilsufanamidas y sulfonilbenzamidinas que se usan como agentes antitumorales
CR7332A (es) INHIBIDORES DEL FACTOR Xa Y DE OTRAS PROTEASAS DE SERINA IMPLICADAS EN LA CASCADA DE LA COAGULACION
HRP20070567B1 (hr) Heliks 12 usmjereni ne-steroidni antiandrogeni
ECSP024382A (es) Inhibidores de proteasa de serina
HK1087613A1 (en) Quinazoline derivatives and their use in the treatment of cancer
CY1107674T1 (el) Φαρμακευτικος συνδυασμος για τη θεραπευτικη αντιμετωπιση της καλοηθους υπερπλασιας του προστατη ή για την μακροπροθεσμη προληψη της οξειας επισχεσης ουρων
BR122018009866B8 (pt) métodos para preparar compostos de éter aminocicloexílico e compostos intermediários
WO2008046082A3 (en) Use of heterocyclic compounds as therapeutic agents
HN2001000277A (es) PIRROLO [2,1 - a] DIHIDROISOQUINOLINAS
BRPI0407913A (pt) antagonistas receptores de ccr-3
GT200100251A (es) Procedimiento para la preparacion de imidazotriazinonas substituidas con sulfonamida
MX2007006927A (es) Combinacion de inhibidor de tirosina cinasa y her-2/neu para terapia de cancer.
BR0109512A (pt) Imidazopiridinas tricìclicas
BRPI0415678A (pt) compostos de pirimidina para o tratamento de inflamação
DE602006020585D1 (de) Neue cysteinproteasehemmer und ihre therapeutische anwendung
MX2008001838A (es) Sales y polimorfos de un inhibidor de vegf-r.
HK1074840A1 (en) Novel dithiolopyrrolones with therapeutic activity
EA200401100A1 (ru) 1α-ФТОР-25-ГИДРОКСИ-16,23E-ДИЕН-26,27-БИСГОМО-20-ЭПИХОЛЕКАЛЬЦИФЕРОЛ И ЕГО ПРИМЕНЕНИЕ ДЛЯ ЛЕЧЕНИЯ
DK1521752T3 (da) Makrocykliske forbindelser til behandling af cancer
ATE319707T1 (de) Verfahren zur herstellung von chinazolinen