HK18184A - Fluorinated amino acids - Google Patents

Fluorinated amino acids

Info

Publication number
HK18184A
HK18184A HK181/84A HK18184A HK18184A HK 18184 A HK18184 A HK 18184A HK 181/84 A HK181/84 A HK 181/84A HK 18184 A HK18184 A HK 18184A HK 18184 A HK18184 A HK 18184A
Authority
HK
Hong Kong
Prior art keywords
rti
compound
formula
sep
fluoromethyl
Prior art date
Application number
HK181/84A
Other languages
English (en)
Inventor
Kollonitsch Janos
Allan Patchett Arthur
Marburg Stephen
Original Assignee
Merck & Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US05/802,391 external-priority patent/US4325961A/en
Application filed by Merck & Co Inc filed Critical Merck & Co Inc
Publication of HK18184A publication Critical patent/HK18184A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/64Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms, e.g. histidine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Indole Compounds (AREA)
HK181/84A 1977-06-01 1984-03-01 Fluorinated amino acids HK18184A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US80238977A 1977-06-01 1977-06-01
US05/802,391 US4325961A (en) 1977-06-01 1977-06-01 Fluorinated amino acids

Publications (1)

Publication Number Publication Date
HK18184A true HK18184A (en) 1984-03-09

Family

ID=27122442

Family Applications (1)

Application Number Title Priority Date Filing Date
HK181/84A HK18184A (en) 1977-06-01 1984-03-01 Fluorinated amino acids

Country Status (26)

Country Link
JP (1) JPS5416423A (en, 2012)
AR (1) AR223463A1 (en, 2012)
AT (1) AT360509B (en, 2012)
AU (1) AU518479B2 (en, 2012)
CA (1) CA1120040A (en, 2012)
CH (1) CH639639A5 (en, 2012)
DD (1) DD138651A5 (en, 2012)
DE (1) DE2824116A1 (en, 2012)
DK (1) DK149841C (en, 2012)
ES (1) ES470296A1 (en, 2012)
FI (1) FI66840C (en, 2012)
FR (1) FR2392958A1 (en, 2012)
GB (1) GB1602525A (en, 2012)
GR (1) GR64495B (en, 2012)
HK (1) HK18184A (en, 2012)
HU (1) HU181911B (en, 2012)
IE (1) IE46983B1 (en, 2012)
IT (1) IT1104709B (en, 2012)
LU (1) LU79750A1 (en, 2012)
NL (1) NL190485C (en, 2012)
NO (1) NO147382C (en, 2012)
NZ (1) NZ187377A (en, 2012)
PL (1) PL115731B1 (en, 2012)
PT (1) PT68102B (en, 2012)
SE (1) SE7806440L (en, 2012)
YU (1) YU129178A (en, 2012)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL59481A0 (en) * 1977-07-11 1980-05-30 Merrell Toraude & Co -halomethyl amino acids
CA1091661A (en) * 1977-07-11 1980-12-16 Philippe Bey .alpha.-HALOMETHYL DERIVATIVES OF .alpha.-AMINO ACIDS
ZA783273B (en) * 1977-07-11 1979-06-27 Merrell Toraude & Co A-halomethyl amino acids
US4315095A (en) * 1977-07-28 1982-02-09 Merrell Toraude Et Compagnie α-Halomethyl derivatives of amino acids
ATE3282T1 (de) * 1978-07-24 1983-05-15 Merck & Co. Inc. Alpha-difluormethyl-alpha-aminosaeuren und sie enthaltende pharmazeutische zusammensetzung.
IE49522B1 (en) * 1979-04-26 1985-10-16 Merrell Toraude & Co Alpha-halomethylaminoacids
CA1158657A (en) * 1979-07-26 1983-12-13 Philippe Bey Preparation of fluorinated methyl aminoalkanoic acids and novel process intermediates
ZA813018B (en) * 1980-05-09 1982-05-26 Merrell Toraude & Co Fluoromethylated tyrosine methyl ester
CA1174603A (en) * 1980-06-16 1984-09-18 Albert Sjoerdsma Method of inhibiting the growth of protozoa
US4421767A (en) * 1981-06-01 1983-12-20 Merrell Toraude Et Compagnie Compounds and methods for treating depression
GB9325368D0 (en) * 1993-12-10 1994-02-16 Univ Bristol Organic compounds

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3046300A (en) * 1960-10-21 1962-07-24 Merck & Co Inc alpha-trifluoromethyloxyphenylalanines

Also Published As

Publication number Publication date
NO781892L (no) 1978-12-04
PT68102A (en) 1978-06-01
NL190485C (nl) 1994-03-16
AR223463A1 (es) 1981-08-31
GR64495B (en) 1980-03-31
DD138651A5 (de) 1979-11-14
NO147382C (no) 1983-03-30
DE2824116C2 (en, 2012) 1989-04-27
NL190485B (nl) 1993-10-18
DK149841B (da) 1986-10-13
LU79750A1 (fr) 1979-02-02
CH639639A5 (en) 1983-11-30
JPS641474B2 (en, 2012) 1989-01-11
AU3658678A (en) 1979-12-06
FI66840B (fi) 1984-08-31
FR2392958B1 (en, 2012) 1980-10-24
IT7849637A0 (it) 1978-05-31
CA1120040A (en) 1982-03-16
DK149841C (da) 1987-04-21
NL7805981A (nl) 1978-12-05
AT360509B (de) 1981-01-12
GB1602525A (en) 1981-11-11
ES470296A1 (es) 1979-09-16
NO147382B (no) 1982-12-20
IE781078L (en) 1978-12-01
AU518479B2 (en) 1981-10-01
YU129178A (en) 1983-01-21
ATA393278A (de) 1980-06-15
FI66840C (fi) 1984-12-10
SE7806440L (sv) 1978-12-02
PL115731B1 (en) 1981-04-30
FR2392958A1 (fr) 1978-12-29
PT68102B (en) 1982-06-08
DE2824116A1 (de) 1978-12-14
IE46983B1 (en) 1983-11-16
FI781674A7 (fi) 1978-12-02
PL207242A1 (pl) 1979-04-23
IT1104709B (it) 1985-10-28
NZ187377A (en) 1981-05-15
HU181911B (en) 1983-11-28
JPS5416423A (en) 1979-02-07
DK237978A (da) 1979-01-19

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Legal Events

Date Code Title Description
PE Patent expired