HK1212232A1 - Formulations pharmacokinetics of deuterated benzoquinoline inhibitors of vesicular monoamine transporter 2 - Google Patents

Formulations pharmacokinetics of deuterated benzoquinoline inhibitors of vesicular monoamine transporter 2 Download PDF

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Publication number
HK1212232A1
HK1212232A1 HK16100273.0A HK16100273A HK1212232A1 HK 1212232 A1 HK1212232 A1 HK 1212232A1 HK 16100273 A HK16100273 A HK 16100273A HK 1212232 A1 HK1212232 A1 HK 1212232A1
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HK
Hong Kong
Prior art keywords
pharmacokinetics
formulations
monoamine transporter
vesicular monoamine
deuterated
Prior art date
Application number
HK16100273.0A
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English (en)
Chinese (zh)
Inventor
Andreas Sommer
Chengzhi Zhang
John Carter
John Arthur
Margaret BRADBURY
Thomas Gant
Manouchehr Shahbaz
Original Assignee
Auspex Pharmaceuticals, Inc.
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=50341905&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=HK1212232(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Auspex Pharmaceuticals, Inc. filed Critical Auspex Pharmaceuticals, Inc.
Publication of HK1212232A1 publication Critical patent/HK1212232A1/xx

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    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A61K31/473—Quinolines; Isoquinolines ortho- or peri-condensed with carbocyclic ring systems, e.g. acridines, phenanthridines
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    • A61K31/4738—Quinolines; Isoquinolines ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/4745—Quinolines; Isoquinolines ortho- or peri-condensed with heterocyclic ring systems condensed with ring systems having nitrogen as a ring hetero atom, e.g. phenantrolines
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HK16100273.0A 2012-09-18 2013-09-18 Formulations pharmacokinetics of deuterated benzoquinoline inhibitors of vesicular monoamine transporter 2 HK1212232A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201261702586P 2012-09-18 2012-09-18
US61/702,586 2012-09-18
PCT/US2013/060387 WO2014047167A1 (en) 2012-09-18 2013-09-18 Formulations pharmacokinetics of deuterated benzoquinoline inhibitors of vesicular monoamine transporter 2

Related Parent Applications (1)

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HK42024096455.1A Division HK40109792A (en) 2012-09-18 2016-01-12 Formulations pharmacokinetics of deuterated benzoquinoline inhibitors of vesicular monoamine transporter 2

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HK42024096455.1A Addition HK40109792A (en) 2012-09-18 2016-01-12 Formulations pharmacokinetics of deuterated benzoquinoline inhibitors of vesicular monoamine transporter 2

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HK1212232A1 true HK1212232A1 (en) 2016-06-10

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US (10) US9346800B2 (enExample)
EP (2) EP2897615A4 (enExample)
JP (4) JP6362601B2 (enExample)
CN (3) CN111728971A (enExample)
AU (3) AU2013318182C1 (enExample)
BR (1) BR112015005894B1 (enExample)
CA (2) CA3124804C (enExample)
HK (1) HK1212232A1 (enExample)
IN (1) IN2015DN01662A (enExample)
NZ (1) NZ705372A (enExample)
WO (1) WO2014047167A1 (enExample)

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WO2014047167A1 (en) 2012-09-18 2014-03-27 Auspex Pharmaceuticals, Inc. Formulations pharmacokinetics of deuterated benzoquinoline inhibitors of vesicular monoamine transporter 2
US9550780B2 (en) 2012-09-18 2017-01-24 Auspex Pharmaceuticals, Inc. Formulations pharmacokinetics of deuterated benzoquinoline inhibitors of vesicular monoamine transporter 2
HK1224222A1 (zh) 2013-12-03 2017-08-18 Auspex Pharmaceuticals, Inc. 制造苯并喹啉化合物的方法
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WO2015175505A1 (en) * 2014-05-15 2015-11-19 Lundbeck Llc Tetrabenazine modified release formulation
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MA41557A (fr) 2015-02-18 2017-12-26 Auspex Pharmaceuticals Inc Inhibiteurs diméthoxyphényles du transporteur vésiculaire des monoamines 2
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JP6919099B2 (ja) * 2015-06-23 2021-08-18 ニューロクライン バイオサイエンシーズ，インコーポレイテッド 神経学的疾患または障害を処置するためのｖｍａｔ２阻害剤
HUE053872T2 (hu) 2015-10-30 2021-07-28 Neurocrine Biosciences Inc Valbenazin-ditozilát és polimorfjai
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