HK1203814A1 - 用於治療 型糖尿病、 型糖尿病、葡萄糖耐量降低或高血糖症的 抑制劑 - Google Patents

用於治療 型糖尿病、 型糖尿病、葡萄糖耐量降低或高血糖症的 抑制劑

Info

Publication number
HK1203814A1
HK1203814A1 HK15104259.1A HK15104259A HK1203814A1 HK 1203814 A1 HK1203814 A1 HK 1203814A1 HK 15104259 A HK15104259 A HK 15104259A HK 1203814 A1 HK1203814 A1 HK 1203814A1
Authority
HK
Hong Kong
Prior art keywords
sglt
diabetes mellitus
type
hyperglycemia
inhibitor
Prior art date
Application number
HK15104259.1A
Other languages
English (en)
Inventor
.埃克爾曼
.馬克
.西曼
.托馬斯
.布羅伊德爾
.格里姆普勒
Original Assignee
Boehringer Ingelheim Int
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=42008536&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=HK1203814(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Boehringer Ingelheim Int filed Critical Boehringer Ingelheim Int
Publication of HK1203814A1 publication Critical patent/HK1203814A1/zh

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    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7028Compounds having saccharide radicals attached to non-saccharide compounds by glycosidic linkages
    • A61K31/7034Compounds having saccharide radicals attached to non-saccharide compounds by glycosidic linkages attached to a carbocyclic compound, e.g. phloridzin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7048Compounds having saccharide radicals and heterocyclic rings having oxygen as a ring hetero atom, e.g. leucoglucosan, hesperidin, erythromycin, nystatin, digitoxin or digoxin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/26Carbohydrates, e.g. sugar alcohols, amino sugars, nucleic acids, mono-, di- or oligo-saccharides; Derivatives thereof, e.g. polysorbates, sorbitan fatty acid esters or glycyrrhizin
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    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0019Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
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    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2013Organic compounds, e.g. phospholipids, fats
    • A61K9/2018Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
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    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/2027Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
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    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
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    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/48Drugs for disorders of the endocrine system of the pancreatic hormones
    • A61P5/50Drugs for disorders of the endocrine system of the pancreatic hormones for increasing or potentiating the activity of insulin
    • AHUMAN NECESSITIES
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    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
HK15104259.1A 2009-02-13 2012-03-13 用於治療 型糖尿病、 型糖尿病、葡萄糖耐量降低或高血糖症的 抑制劑 HK1203814A1 (zh)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US15231809P 2009-02-13 2009-02-13

Publications (1)

Publication Number Publication Date
HK1203814A1 true HK1203814A1 (zh) 2015-11-06

Family

ID=42008536

Family Applications (1)

Application Number Title Priority Date Filing Date
HK15104259.1A HK1203814A1 (zh) 2009-02-13 2012-03-13 用於治療 型糖尿病、 型糖尿病、葡萄糖耐量降低或高血糖症的 抑制劑

Country Status (28)

Country Link
US (8) US20110046087A1 (zh)
EP (1) EP2396005A1 (zh)
JP (3) JP5896276B2 (zh)
KR (2) KR20110118668A (zh)
CN (2) CN104138370A (zh)
AP (1) AP2011005795A0 (zh)
AR (1) AR075424A1 (zh)
AU (1) AU2010212865A1 (zh)
BR (1) BRPI1013640A2 (zh)
CA (1) CA2751833C (zh)
CL (1) CL2011001757A1 (zh)
CO (1) CO6410306A2 (zh)
EA (1) EA021796B1 (zh)
EC (1) ECSP11011275A (zh)
GE (1) GEP20146120B (zh)
HK (1) HK1203814A1 (zh)
IL (1) IL213723A0 (zh)
MA (1) MA33043B1 (zh)
MX (1) MX344264B (zh)
MY (1) MY161472A (zh)
NZ (1) NZ594485A (zh)
PE (1) PE20120002A1 (zh)
PH (1) PH12016501607A1 (zh)
SG (2) SG10201600204YA (zh)
TN (1) TN2011000413A1 (zh)
TW (1) TWI478935B (zh)
UA (1) UA106365C2 (zh)
WO (1) WO2010092123A1 (zh)

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