HK1102021A1 - Pharmaceutical composition for oral administration of a pyrazol-3- carboxamide derivative - Google Patents

Pharmaceutical composition for oral administration of a pyrazol-3- carboxamide derivative

Info

Publication number
HK1102021A1
HK1102021A1 HK07106763.5A HK07106763A HK1102021A1 HK 1102021 A1 HK1102021 A1 HK 1102021A1 HK 07106763 A HK07106763 A HK 07106763A HK 1102021 A1 HK1102021 A1 HK 1102021A1
Authority
HK
Hong Kong
Prior art keywords
pyrazol
pharmaceutical composition
oral administration
carboxamide derivative
carboxamide
Prior art date
Application number
HK07106763.5A
Other languages
English (en)
Inventor
Thierry Breul
Jean Claude Gautier
Olivier Saslawski
Original Assignee
Sanofi Aventis
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi Aventis filed Critical Sanofi Aventis
Publication of HK1102021A1 publication Critical patent/HK1102021A1/xx

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/10Dispersions; Emulsions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4151,2-Diazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • A61K31/4523Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/454Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. pimozide, domperidone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/08Solutions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Dispersion Chemistry (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
HK07106763.5A 2003-11-10 2007-06-25 Pharmaceutical composition for oral administration of a pyrazol-3- carboxamide derivative HK1102021A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR0313259A FR2861992B1 (fr) 2003-11-10 2003-11-10 Composition pharmaceutique destinee a l'administration orale d'un derive de pyrazole-3-carboxamide.
PCT/FR2004/002875 WO2005046690A1 (fr) 2003-11-10 2004-11-09 Composition pharmaceutique destinee a l'administration orale d'un derive de pyrazole-3­carboxamide

Publications (1)

Publication Number Publication Date
HK1102021A1 true HK1102021A1 (en) 2007-11-02

Family

ID=34508418

Family Applications (1)

Application Number Title Priority Date Filing Date
HK07106763.5A HK1102021A1 (en) 2003-11-10 2007-06-25 Pharmaceutical composition for oral administration of a pyrazol-3- carboxamide derivative

Country Status (28)

Country Link
US (2) US20060264469A1 (es)
EP (1) EP1691808B1 (es)
JP (1) JP4767171B2 (es)
KR (1) KR20060108668A (es)
CN (1) CN100528158C (es)
AR (1) AR047237A1 (es)
AT (1) ATE429227T1 (es)
AU (1) AU2004289086A1 (es)
BR (1) BRPI0416341A (es)
CA (1) CA2544413A1 (es)
CY (1) CY1110478T1 (es)
DE (1) DE602004020797D1 (es)
DK (1) DK1691808T3 (es)
ES (1) ES2325373T3 (es)
FR (1) FR2861992B1 (es)
HK (1) HK1102021A1 (es)
HR (1) HRP20090393T1 (es)
IL (1) IL175556A (es)
MA (1) MA28419B1 (es)
NO (1) NO20062609L (es)
NZ (1) NZ547763A (es)
PL (1) PL1691808T3 (es)
PT (1) PT1691808E (es)
RU (1) RU2321404C1 (es)
SI (1) SI1691808T1 (es)
TW (1) TWI280129B (es)
WO (1) WO2005046690A1 (es)
ZA (1) ZA200604451B (es)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1880715A1 (en) * 2006-07-19 2008-01-23 Abbott GmbH & Co. KG Pharmaceutically acceptable solubilizing composition and pharmaceutical dosage form containing same
EP1920767A1 (en) * 2006-11-09 2008-05-14 Abbott GmbH & Co. KG Melt-processed imatinib dosage form
WO2009024590A2 (en) * 2007-08-21 2009-02-26 Basilea Pharmaceutica Ag Antifungal composition
MY158809A (en) * 2010-09-22 2016-11-15 Craun Res Sdn Bhd Pharmaceutical compositions for calanolides, their derivatives and analogues, and process for producing the same
WO2012071043A1 (en) * 2010-11-24 2012-05-31 Pharmaceutics International, Inc. Self micro-emulsifying drug delivery system with increased bioavailability

Family Cites Families (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5059691A (en) * 1990-01-22 1991-10-22 American Cyanamid Company N-((dialkylamino)methylene)-substituted pyrazolo (1,5-A)-pyrimidine-3-carboxamides and N-((dialkylamino)methylene)-substituted-4,5-dihydropyrazolo-(1,5-A)-pyrimidine-3-carboxamides
FR2692575B1 (fr) * 1992-06-23 1995-06-30 Sanofi Elf Nouveaux derives du pyrazole, procede pour leur preparation et compositions pharmaceutiques les contenant.
EP1033128B2 (en) * 1993-09-28 2011-11-23 R.P. Scherer GmbH Soft gelatin capsule manufacture
GB9405304D0 (en) * 1994-03-16 1994-04-27 Scherer Ltd R P Delivery systems for hydrophobic drugs
JPH11504028A (ja) * 1995-04-24 1999-04-06 イースム リサーチ ディベロップメント カンパニー オブ ザ ヒーブル ユニバーシティ オブ エルサレム 油/水エマルジョンを作り出す自己乳化性配合物
JPH11505257A (ja) * 1995-05-19 1999-05-18 アボツト・ラボラトリーズ 親油性薬物の自己乳化性製剤
US5993858A (en) * 1996-06-14 1999-11-30 Port Systems L.L.C. Method and formulation for increasing the bioavailability of poorly water-soluble drugs
TW495509B (en) * 1997-03-14 2002-07-21 Otsuka Pharma Co Ltd Novel pyrimidine derivative
FR2761265B1 (fr) * 1997-03-28 1999-07-02 Sanofi Sa Composition pharmaceutique pour l'administration orale d'un derive du n-piperidino-3-pyrazolecarboxamide, de ses sels et de leurs solvates
FR2761266B1 (fr) * 1997-03-28 1999-07-02 Sanofi Sa Composition pharmaceutique formee par granulation humide pour l'administration orale d'un derive du n-piperidino-3- pyrazolecarboxamide, de ses sels et de leurs solvates
US6617426B1 (en) * 1999-06-22 2003-09-09 Merck & Co Inc Cysteinyl protease inhibitors
JP2001151669A (ja) * 1999-11-24 2001-06-05 Nippon Kayaku Co Ltd 経口用自己乳化製剤
YU43702A (sh) * 1999-12-23 2004-11-25 Pfizer Products Inc. Farmaceutske kompozicije koje obezbeđuju povećanje koncentracije leka
GB0001928D0 (en) * 2000-01-27 2000-03-22 Novartis Ag Organic compounds
FR2831883B1 (fr) * 2001-11-08 2004-07-23 Sanofi Synthelabo Forme polymorphe du rimonabant, son procede de preparation et les compositions pharmaceutiques en contenant
JP2005523295A (ja) * 2002-03-01 2005-08-04 ノバガリ、ファルマ、エスアー 難溶性薬剤の自己乳化型薬物送達システム
GB0216700D0 (en) * 2002-07-18 2002-08-28 Astrazeneca Ab Process

Also Published As

Publication number Publication date
AR047237A1 (es) 2006-01-11
CA2544413A1 (fr) 2005-05-26
JP4767171B2 (ja) 2011-09-07
US20060264469A1 (en) 2006-11-23
RU2006120447A (ru) 2007-12-20
AU2004289086A1 (en) 2005-05-26
KR20060108668A (ko) 2006-10-18
DE602004020797D1 (de) 2009-06-04
RU2321404C1 (ru) 2008-04-10
NZ547763A (en) 2009-08-28
FR2861992B1 (fr) 2007-07-20
WO2005046690A1 (fr) 2005-05-26
TWI280129B (en) 2007-05-01
PL1691808T3 (pl) 2009-09-30
DK1691808T3 (da) 2009-08-03
IL175556A0 (en) 2008-04-13
CN100528158C (zh) 2009-08-19
CY1110478T1 (el) 2015-04-29
EP1691808B1 (fr) 2009-04-22
FR2861992A1 (fr) 2005-05-13
HRP20090393T1 (en) 2009-08-31
SI1691808T1 (sl) 2009-10-31
ZA200604451B (en) 2007-10-31
ES2325373T3 (es) 2009-09-02
EP1691808A1 (fr) 2006-08-23
CN1925856A (zh) 2007-03-07
ATE429227T1 (de) 2009-05-15
IL175556A (en) 2010-11-30
PT1691808E (pt) 2009-07-14
NO20062609L (no) 2006-06-06
JP2007516960A (ja) 2007-06-28
TW200524597A (en) 2005-08-01
US20090004261A1 (en) 2009-01-01
BRPI0416341A (pt) 2007-02-27
MA28419B1 (fr) 2007-02-01

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Legal Events

Date Code Title Description
PC Patent ceased (i.e. patent has lapsed due to the failure to pay the renewal fee)

Effective date: 20131109