HK1085658A1 - Pharmaceutical compositions comprising 1-aminocyclohexane derivatives and acetylcholinesterase inhibitors - Google Patents

Pharmaceutical compositions comprising 1-aminocyclohexane derivatives and acetylcholinesterase inhibitors

Info

Publication number
HK1085658A1
HK1085658A1 HK06105633A HK06105633A HK1085658A1 HK 1085658 A1 HK1085658 A1 HK 1085658A1 HK 06105633 A HK06105633 A HK 06105633A HK 06105633 A HK06105633 A HK 06105633A HK 1085658 A1 HK1085658 A1 HK 1085658A1
Authority
HK
Hong Kong
Prior art keywords
pharmaceutical compositions
acetylcholinesterase inhibitors
aminocyclohexane derivatives
aminocyclohexane
derivatives
Prior art date
Application number
HK06105633A
Other languages
English (en)
Inventor
Hans-Joerg Moebius
Original Assignee
Merz Pharma Gmbh & Co Kgaa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merz Pharma Gmbh & Co Kgaa filed Critical Merz Pharma Gmbh & Co Kgaa
Publication of HK1085658A1 publication Critical patent/HK1085658A1/xx

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/16Amides, e.g. hydroxamic acids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/21Esters, e.g. nitroglycerine, selenocyanates
    • A61K31/27Esters, e.g. nitroglycerine, selenocyanates of carbamic or thiocarbamic acids, meprobamate, carbachol, neostigmine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/325Carbamic acids; Thiocarbamic acids; Anhydrides or salts thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • A61K31/473Quinolines; Isoquinolines ortho- or peri-condensed with carbocyclic ring systems, e.g. acridines, phenanthridines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0053Mouth and digestive tract, i.e. intraoral and peroral administration
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biomedical Technology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Organic Chemistry (AREA)
  • Emergency Medicine (AREA)
  • Psychiatry (AREA)
  • Hospice & Palliative Care (AREA)
  • Nutrition Science (AREA)
  • Physiology (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicinal Preparation (AREA)
HK06105633A 2002-10-24 2006-05-16 Pharmaceutical compositions comprising 1-aminocyclohexane derivatives and acetylcholinesterase inhibitors HK1085658A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US42091802P 2002-10-24 2002-10-24
PCT/GB2003/004549 WO2004037234A2 (en) 2002-10-24 2003-10-23 Combination therapy using 1-aminocyclohexane derivatives and acetylcholinesterase inhibitors

Publications (1)

Publication Number Publication Date
HK1085658A1 true HK1085658A1 (en) 2006-09-01

Family

ID=32176649

Family Applications (1)

Application Number Title Priority Date Filing Date
HK06105633A HK1085658A1 (en) 2002-10-24 2006-05-16 Pharmaceutical compositions comprising 1-aminocyclohexane derivatives and acetylcholinesterase inhibitors

Country Status (17)

Country Link
US (6) US20040087658A1 (ja)
EP (2) EP1556019A2 (ja)
JP (2) JP2006506378A (ja)
KR (2) KR100852834B1 (ja)
CN (1) CN100339070C (ja)
AU (1) AU2003274353B2 (ja)
CA (1) CA2502432A1 (ja)
EA (1) EA008863B1 (ja)
GE (1) GEP20094759B (ja)
HK (1) HK1085658A1 (ja)
MX (1) MXPA04006900A (ja)
NO (1) NO20052462L (ja)
PL (1) PL376476A1 (ja)
TW (1) TW200418446A (ja)
UA (1) UA83645C2 (ja)
WO (1) WO2004037234A2 (ja)
ZA (1) ZA200503204B (ja)

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EP2260839A2 (en) 2010-12-15
CN100339070C (zh) 2007-09-26
AU2003274353A1 (en) 2004-05-13
JP2006506378A (ja) 2006-02-23
UA83645C2 (ru) 2008-08-11
KR100852834B1 (ko) 2008-08-18
PL376476A1 (en) 2005-12-27
KR100777904B1 (ko) 2007-11-28
TW200418446A (en) 2004-10-01
CA2502432A1 (en) 2004-05-06
EA200500699A1 (ru) 2005-10-27
JP2011246491A (ja) 2011-12-08
US20040087658A1 (en) 2004-05-06
KR20070087161A (ko) 2007-08-27
CN1720035A (zh) 2006-01-11
WO2004037234A3 (en) 2004-08-05
KR20050072770A (ko) 2005-07-12
US20100227852A1 (en) 2010-09-09
US20160136144A1 (en) 2016-05-19
US20210169864A1 (en) 2021-06-10
ZA200503204B (en) 2006-07-26
MXPA04006900A (es) 2004-10-15
EP1556019A2 (en) 2005-07-27
WO2004037234A2 (en) 2004-05-06
NO20052462D0 (no) 2005-05-23
US20140371260A1 (en) 2014-12-18
GEP20094759B (en) 2009-08-25
US20090124659A1 (en) 2009-05-14
AU2003274353B2 (en) 2007-04-05
EA008863B1 (ru) 2007-08-31
EP2260839A3 (en) 2012-05-02

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