HK1060360A1 - Somatostatin-dopamine chimeric analogs - Google Patents
Somatostatin-dopamine chimeric analogsInfo
- Publication number
- HK1060360A1 HK1060360A1 HK04102651.2A HK04102651A HK1060360A1 HK 1060360 A1 HK1060360 A1 HK 1060360A1 HK 04102651 A HK04102651 A HK 04102651A HK 1060360 A1 HK1060360 A1 HK 1060360A1
- Authority
- HK
- Hong Kong
- Prior art keywords
- somatostatin
- dopamine chimeric
- chimeric analogs
- analogs
- dopamine
- Prior art date
Links
- 229960003638 dopamine Drugs 0.000 title 1
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D457/00—Heterocyclic compounds containing indolo [4, 3-f, g] quinoline ring systems, e.g. derivatives of ergoline, of the formula:, e.g. lysergic acid
- C07D457/02—Heterocyclic compounds containing indolo [4, 3-f, g] quinoline ring systems, e.g. derivatives of ergoline, of the formula:, e.g. lysergic acid with hydrocarbon or substituted hydrocarbon radicals, attached in position 8
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
-
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- A61P1/18—Drugs for disorders of the alimentary tract or the digestive system for pancreatic disorders, e.g. pancreatic enzymes
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D457/00—Heterocyclic compounds containing indolo [4, 3-f, g] quinoline ring systems, e.g. derivatives of ergoline, of the formula:, e.g. lysergic acid
- C07D457/04—Heterocyclic compounds containing indolo [4, 3-f, g] quinoline ring systems, e.g. derivatives of ergoline, of the formula:, e.g. lysergic acid with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 8
- C07D457/06—Lysergic acid amides
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D457/00—Heterocyclic compounds containing indolo [4, 3-f, g] quinoline ring systems, e.g. derivatives of ergoline, of the formula:, e.g. lysergic acid
- C07D457/10—Heterocyclic compounds containing indolo [4, 3-f, g] quinoline ring systems, e.g. derivatives of ergoline, of the formula:, e.g. lysergic acid with hetero atoms directly attached in position 8
- C07D457/12—Nitrogen atoms
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/06—Peri-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- C07K14/575—Hormones
- C07K14/655—Somatostatins
- C07K14/6555—Somatostatins at least 1 amino acid in D-form
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Diabetes (AREA)
- Endocrinology (AREA)
- Immunology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Hematology (AREA)
- Molecular Biology (AREA)
- Genetics & Genomics (AREA)
- Biophysics (AREA)
- Biochemistry (AREA)
- Gastroenterology & Hepatology (AREA)
- Zoology (AREA)
- Obesity (AREA)
- Toxicology (AREA)
- Physical Education & Sports Medicine (AREA)
- Heart & Thoracic Surgery (AREA)
- Neurosurgery (AREA)
- Urology & Nephrology (AREA)
- Cardiology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Biomedical Technology (AREA)
- Rheumatology (AREA)
- Neurology (AREA)
- Epidemiology (AREA)
- Psychiatry (AREA)
- Nutrition Science (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US29705901P | 2001-06-08 | 2001-06-08 | |
PCT/US2002/017859 WO2002100888A1 (en) | 2001-06-08 | 2002-06-07 | Somatostatin-dopamine chimeric analogs |
Publications (1)
Publication Number | Publication Date |
---|---|
HK1060360A1 true HK1060360A1 (en) | 2004-08-06 |
Family
ID=23144680
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
HK04102651.2A HK1060360A1 (en) | 2001-06-08 | 2004-04-15 | Somatostatin-dopamine chimeric analogs |
Country Status (25)
Country | Link |
---|---|
US (4) | US7579435B2 (ru) |
EP (2) | EP2062914B1 (ru) |
JP (2) | JP3996897B2 (ru) |
KR (3) | KR100743212B1 (ru) |
CN (2) | CN101481405A (ru) |
AR (1) | AR037226A1 (ru) |
AT (1) | ATE424414T1 (ru) |
AU (1) | AU2002305845B2 (ru) |
BR (1) | BR0210915A (ru) |
CA (1) | CA2449634C (ru) |
CZ (1) | CZ305160B6 (ru) |
DE (1) | DE60231403D1 (ru) |
DK (2) | DK1401863T3 (ru) |
ES (2) | ES2325880T3 (ru) |
HK (1) | HK1060360A1 (ru) |
HU (1) | HUP0400245A3 (ru) |
IL (2) | IL158922A0 (ru) |
MX (1) | MXPA03011321A (ru) |
NO (2) | NO332042B1 (ru) |
NZ (1) | NZ530007A (ru) |
PL (1) | PL216217B1 (ru) |
PT (2) | PT1401863E (ru) |
RU (1) | RU2277539C2 (ru) |
TW (1) | TWI318214B (ru) |
WO (1) | WO2002100888A1 (ru) |
Families Citing this family (23)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AU2002341792B2 (en) * | 2001-09-21 | 2007-09-06 | The Administrators Of The Tulane Educational Fund | Diagnostic or therapeutic somatostatin or bombesin analog conjugates and uses thereof |
AU2004229437B2 (en) * | 2003-04-11 | 2007-12-06 | Ipsen Pharma S.A.S. | Somatostatin-dopamine chimeric analogs |
AU2008200694B2 (en) * | 2003-04-11 | 2011-04-14 | Ipsen Pharma S.A.S. | Method of treating acromegaly, hyperprolactinemia, portal hypertension and gastrointestinal bleeding with somatostatin-dopamine chimeric analogs |
EP2161037A3 (en) * | 2003-04-22 | 2010-05-26 | Ipsen Pharma | Camptothecin-Somatostatin conjugates |
DE10325813B4 (de) | 2003-06-06 | 2007-12-20 | Universitätsklinikum Freiburg | Prophylaxe und/oder Therapie bei der portalen Hypertonie |
US20100261796A1 (en) * | 2005-04-28 | 2010-10-14 | Ferring B.V. | Use of Novel Compounds for IBD Treatment |
US9098855B2 (en) * | 2006-05-23 | 2015-08-04 | Intelligent Clearing Network, Inc. | Intelligent clearing network |
WO2009139855A2 (en) * | 2008-05-14 | 2009-11-19 | Ipsen Pharma S.A.S. | Pharmaceutical compositions of somatostatin-dopamine conjugates |
FR2949469A1 (fr) * | 2009-08-25 | 2011-03-04 | Sanofi Aventis | Derives anticancereux, leur preparation et leur application en therapeutique |
WO2011104627A1 (en) * | 2010-02-24 | 2011-09-01 | Ipsen Pharma S.A.S. | Metabolites of dop2-d-lys(dop2)-cyclo[cys-tyr-d-trp-lys-abu-cys]-thr-nh2 |
KR20140027284A (ko) * | 2011-04-21 | 2014-03-06 | 쎄러테크놀로지스 인코포레이티드 | 성장 호르몬 방출 인자(grf) 유사체 및 이의 용도 |
UA115542C2 (uk) | 2011-12-23 | 2017-11-27 | Іпсен Мануфекчерінг Айрленд Лімітед | Процес синтезу терапевтичних пептидів |
US9620430B2 (en) | 2012-01-23 | 2017-04-11 | Taiwan Semiconductor Manufacturing Company, Ltd. | Sawing underfill in packaging processes |
TWI523863B (zh) | 2012-11-01 | 2016-03-01 | 艾普森藥品公司 | 體抑素-多巴胺嵌合體類似物 |
JP2016503402A (ja) | 2012-11-01 | 2016-02-04 | イプセン ファルマ ソシエテ パール アクシオン サンプリフィエIpsen Pharma S.A.S. | ソマトスタチン類似体及びそのダイマー |
US9096679B2 (en) | 2012-12-03 | 2015-08-04 | The Board Of Regents Of The University Of Oklahoma | Peptide compounds and methods of production and use thereof |
WO2014089088A1 (en) * | 2012-12-03 | 2014-06-12 | The Board Of Regents Of The University Of Oklahoma | Peptide compounds and methods of production and use thereof |
US20200157159A1 (en) | 2013-04-16 | 2020-05-21 | The Board Of Regents Of The University Of Oklahoma | Peptide compounds and compositions thereof |
EP3166967B1 (en) * | 2014-09-14 | 2023-03-08 | Tel Hashomer Medical Research Infrastructure and Services Ltd. | Synthetic somatostatin receptor ligands |
MX2017009406A (es) | 2015-01-20 | 2018-01-18 | Xoc Pharmaceuticals Inc | Compuestos de tipo isoergolina y usos de estos. |
EP3253753A4 (en) | 2015-01-20 | 2018-06-27 | Xoc Pharmaceuticals, Inc | Ergoline compounds and uses thereof |
BR112019025420A2 (pt) | 2017-06-01 | 2020-06-16 | Xoc Pharmaceuticals, Inc. | Compostos policíclicos e usos destes |
WO2023225043A1 (en) * | 2022-05-18 | 2023-11-23 | Kuleon Llc | Tricyclic and tetracyclic serotonin receptor modulators and methods of making and using the same |
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LU78191A1 (de) | 1977-09-28 | 1979-05-25 | Ciba Geigy Ag | Verfahren zur herstellung von neuen cyclopeptiden |
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CA1107273A (en) | 1978-05-19 | 1981-08-18 | Chester A. Meyers | Somatostatin analogs having a substituted tryptophyl residue in position eight |
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DD140044A1 (de) * | 1978-11-08 | 1980-02-06 | Guenter Losse | Verfahren zur herstellung von lysergyl-enkephalin-derivaten |
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US4316890A (en) | 1979-03-16 | 1982-02-23 | Ciba-Geigy Corporation | Peptides and processes for the manufacture thereof |
US4209426A (en) | 1979-05-29 | 1980-06-24 | American Home Products Corporation | Polypeptides related to somatostatin |
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