GT200200250A - Compuestos hexaciclicos - Google Patents

Compuestos hexaciclicos

Info

Publication number
GT200200250A
GT200200250A GT200200250A GT200200250A GT200200250A GT 200200250 A GT200200250 A GT 200200250A GT 200200250 A GT200200250 A GT 200200250A GT 200200250 A GT200200250 A GT 200200250A GT 200200250 A GT200200250 A GT 200200250A
Authority
GT
Guatemala
Prior art keywords
hexaciclic
compounds
record
cases
useful
Prior art date
Application number
GT200200250A
Other languages
English (en)
Spanish (es)
Inventor
Takeshi Murata
Satoshi Niizuma
Nobuo Shimma
Hitomi Suda
Masso Tsukazaki
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Publication of GT200200250A publication Critical patent/GT200200250A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D491/00Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/22Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains four or more hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
GT200200250A 2001-11-30 2002-11-29 Compuestos hexaciclicos GT200200250A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP01128361 2001-11-30

Publications (1)

Publication Number Publication Date
GT200200250A true GT200200250A (es) 2004-01-15

Family

ID=8179394

Family Applications (1)

Application Number Title Priority Date Filing Date
GT200200250A GT200200250A (es) 2001-11-30 2002-11-29 Compuestos hexaciclicos

Country Status (28)

Country Link
US (2) US6825194B2 (https=)
EP (1) EP1480984B9 (https=)
JP (1) JP4305909B2 (https=)
KR (1) KR100895746B1 (https=)
CN (1) CN100338066C (https=)
AT (1) ATE398131T1 (https=)
AU (1) AU2002356720B2 (https=)
BR (1) BR0214615A (https=)
CA (1) CA2468824C (https=)
DE (1) DE60227113D1 (https=)
ES (1) ES2307830T3 (https=)
GT (1) GT200200250A (https=)
HU (1) HUP0500062A3 (https=)
IL (1) IL162058A0 (https=)
MX (1) MXPA04005185A (https=)
MY (1) MY136138A (https=)
NO (1) NO329005B1 (https=)
NZ (1) NZ533568A (https=)
PA (1) PA8558901A1 (https=)
PE (1) PE20030725A1 (https=)
PL (1) PL207510B1 (https=)
RS (1) RS51051B (https=)
RU (1) RU2299212C2 (https=)
TW (1) TWI258481B (https=)
UA (1) UA80409C2 (https=)
UY (1) UY27560A1 (https=)
WO (1) WO2003045952A2 (https=)
ZA (1) ZA200404522B (https=)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7595400B2 (en) 2003-02-21 2009-09-29 Chugai Seiyaku Kabushiki Kaisha Process for the preparation of hexacyclic compounds
TWI351284B (en) 2004-04-09 2011-11-01 Chugai Pharmaceutical Co Ltd Novel water-soluble prodrugs
TW200744603A (en) * 2005-08-22 2007-12-16 Chugai Pharmaceutical Co Ltd Novel anticancer concomitant drug
US20090118271A1 (en) * 2005-10-19 2009-05-07 Chugai Seiyaku Kabushiki Kaisha Preventive or Therapeutic Agents for Pancreatic Cancer, Ovarian Cancer, or Liver Cancer Comprising a Novel Water-Soluble Prodrug
RU2439073C1 (ru) * 2010-07-13 2012-01-10 Государственное образовательное учреждение высшего профессионального образования "Кубанский государственный технологический университет" (ГОУ ВПО "КубГТУ") СПОСОБ ПОЛУЧЕНИЯ ПРОИЗВОДНЫХ ИНДОЛИЗИНО[7,6-b]ИНДОЛА
MX2021011812A (es) 2019-03-29 2021-10-22 Medimmune Ltd Compuestos y conjugados de estos.

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4473692A (en) 1981-09-04 1984-09-25 Kabushiki Kaisha Yakult Honsha Camptothecin derivatives and process for preparing same
US4939255A (en) * 1987-06-24 1990-07-03 Daiichi Pharmaceutical Co., Ltd. Hexa-cyclic camptothecin derivatives
HU213136B (en) * 1990-08-14 1997-02-28 Kyorin Seiyaku Kk Process for producing fluoroethyl camptothecin derivatives and pharmaceutical compositions containing them
JP3008226B2 (ja) * 1991-01-16 2000-02-14 第一製薬株式会社 六環性化合物
JP3359955B2 (ja) * 1992-07-16 2002-12-24 第一製薬株式会社 抗腫瘍剤
GB9402934D0 (en) * 1994-02-16 1994-04-06 Erba Carlo Spa Camptothecin derivatives and process for their preparation
US5663177A (en) * 1995-05-31 1997-09-02 Smithkline Beecham Corporation Water soluble camptothecin analogs
ES2262223T3 (es) 1997-02-14 2006-11-16 Bionumerik Pharmaceuticals, Inc. Derivados de camptotecina altamente lipofilos.
GB9715821D0 (en) * 1997-07-25 1997-10-01 Pharmacia & Upjohn Spa Amidino-camptothecin derivatives

Also Published As

Publication number Publication date
CN100338066C (zh) 2007-09-19
AU2002356720B2 (en) 2009-01-29
CA2468824A1 (en) 2003-06-05
RS51051B (sr) 2010-10-31
US20050059679A1 (en) 2005-03-17
BR0214615A (pt) 2004-09-14
JP4305909B2 (ja) 2009-07-29
NZ533568A (en) 2006-01-27
US6825194B2 (en) 2004-11-30
MXPA04005185A (es) 2004-08-11
ES2307830T3 (es) 2008-12-01
MY136138A (en) 2008-08-29
ZA200404522B (en) 2005-01-04
NO329005B1 (no) 2010-07-19
WO2003045952A3 (en) 2003-10-16
RS47004A (sr) 2007-02-05
IL162058A0 (en) 2005-11-20
RU2004119841A (ru) 2005-03-27
AU2002356720A1 (en) 2003-06-10
TWI258481B (en) 2006-07-21
KR20040062976A (ko) 2004-07-09
US20030144304A1 (en) 2003-07-31
CA2468824C (en) 2011-01-11
TW200408642A (en) 2004-06-01
HK1077303A1 (en) 2006-02-10
HUP0500062A2 (hu) 2005-04-28
DE60227113D1 (de) 2008-07-24
WO2003045952A2 (en) 2003-06-05
JP2005511643A (ja) 2005-04-28
CN1617874A (zh) 2005-05-18
EP1480984B1 (en) 2008-06-11
UY27560A1 (es) 2003-05-30
ATE398131T1 (de) 2008-07-15
HK1072935A1 (en) 2005-09-16
PA8558901A1 (es) 2003-06-30
NO20042729L (no) 2004-08-27
PE20030725A1 (es) 2003-08-28
RU2299212C2 (ru) 2007-05-20
EP1480984B9 (en) 2009-03-11
PL370479A1 (en) 2005-05-30
HUP0500062A3 (en) 2012-12-28
PL207510B1 (pl) 2010-12-31
UA80409C2 (en) 2007-09-25
KR100895746B1 (ko) 2009-04-30
EP1480984A2 (en) 2004-12-01
US7109195B2 (en) 2006-09-19

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