GR3015430T3 - 3-[2-(dimethylamino)ethyl]-N-methyl-1H-indole-5-methanesulphonamide sulphate (2:1). - Google Patents

3-[2-(dimethylamino)ethyl]-N-methyl-1H-indole-5-methanesulphonamide sulphate (2:1).

Info

Publication number
GR3015430T3
GR3015430T3 GR940403944T GR940403944T GR3015430T3 GR 3015430 T3 GR3015430 T3 GR 3015430T3 GR 940403944 T GR940403944 T GR 940403944T GR 940403944 T GR940403944 T GR 940403944T GR 3015430 T3 GR3015430 T3 GR 3015430T3
Authority
GR
Greece
Prior art keywords
indole
dimethylamino
ethyl
methyl
methanesulphonamide sulphate
Prior art date
Application number
GR940403944T
Other languages
Greek (el)
English (en)
Inventor
Joanne Craig
Derek Leslie Crookes
Stephen John Skittrall
Original Assignee
Glaxo Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Publication of GR3015430T3 publication Critical patent/GR3015430T3/el

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
    • C07D209/14—Radicals substituted by nitrogen atoms, not forming part of a nitro radical
    • C07D209/16—Tryptamines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/06—Antimigraine agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A61P29/02—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID] without antiinflammatory effect

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pain & Pain Management (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Engineering & Computer Science (AREA)
  • Biomedical Technology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Indole Compounds (AREA)
GR940403944T 1990-12-12 1995-03-16 3-[2-(dimethylamino)ethyl]-N-methyl-1H-indole-5-methanesulphonamide sulphate (2:1). GR3015430T3 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB909026998A GB9026998D0 (en) 1990-12-12 1990-12-12 Medicaments

Publications (1)

Publication Number Publication Date
GR3015430T3 true GR3015430T3 (en) 1995-06-30

Family

ID=10686904

Family Applications (1)

Application Number Title Priority Date Filing Date
GR940403944T GR3015430T3 (en) 1990-12-12 1995-03-16 3-[2-(dimethylamino)ethyl]-N-methyl-1H-indole-5-methanesulphonamide sulphate (2:1).

Country Status (36)

Country Link
US (2) US5554639A (de)
EP (1) EP0490689B1 (de)
JP (1) JP2994037B2 (de)
KR (1) KR100211479B1 (de)
CN (2) CN1030890C (de)
AP (1) AP230A (de)
AT (1) ATE119881T1 (de)
AU (1) AU650706B2 (de)
BE (1) BE1005085A3 (de)
CA (1) CA2098302C (de)
CH (1) CH684192A5 (de)
CY (1) CY2005A (de)
CZ (1) CZ281931B6 (de)
DE (1) DE69108200T2 (de)
DK (1) DK0490689T3 (de)
EG (1) EG20219A (de)
ES (1) ES2069836T3 (de)
FR (1) FR2670487B1 (de)
GB (2) GB9026998D0 (de)
GR (1) GR3015430T3 (de)
HK (1) HK82697A (de)
HU (1) HU211937A9 (de)
IE (1) IE62894B1 (de)
IL (1) IL100330A (de)
IS (1) IS1706B (de)
IT (1) IT1252868B (de)
MX (1) MX9102501A (de)
MY (1) MY109265A (de)
NL (1) NL9102071A (de)
NZ (1) NZ240942A (de)
PT (1) PT99757B (de)
RU (1) RU2108328C1 (de)
TW (2) TW300886B (de)
WO (1) WO1992010477A1 (de)
YU (1) YU48926B (de)
ZA (1) ZA919750B (de)

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US20040176359A1 (en) * 2001-02-20 2004-09-09 University Of Kentucky Research Foundation Intranasal Benzodiazepine compositions
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US7208628B2 (en) * 2002-05-13 2007-04-24 Kansas State University Research Foundation Compositions and methods for the treatment of hepatitis C virus infection
US7074893B2 (en) * 2002-06-03 2006-07-11 Regents Of The University Of Michigan Methods and compositions for the treatment of diseases associated with signal transduction aberrations
US20040068000A1 (en) * 2002-10-02 2004-04-08 Mintong Guo Compression coated tablets
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US20080213363A1 (en) * 2003-01-23 2008-09-04 Singh Nikhilesh N Methods and compositions for delivering 5-HT3 antagonists across the oral mucosa
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WO2004112723A2 (en) 2003-06-20 2004-12-29 Ronald Aung-Din Tropical therapy for the treatment of migraines, muscle sprains, muscle spasm, spasticity and related conditions
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MY147767A (en) 2004-06-16 2013-01-31 Janssen Pharmaceutica Nv Novel sulfamate and sulfamide derivatives useful for the treatment of epilepsy and related disorders
JP2008545650A (ja) 2005-05-20 2008-12-18 ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ スルファミド誘導体の製造方法
US20070166336A1 (en) * 2005-12-13 2007-07-19 David Delmarre Stable and palatable oral liquid sumatriptan compositions
US8497298B2 (en) 2005-12-19 2013-07-30 Janssen Pharmaceutica Nv Use of benzo-fused heterocycle sulfamide derivatives for lowering lipids and lowering blood glucose levels
US8716231B2 (en) 2005-12-19 2014-05-06 Janssen Pharmaceutica Nv Use of benzo-fused heterocycle sulfamide derivatives for the treatment of pain
US8691867B2 (en) 2005-12-19 2014-04-08 Janssen Pharmaceutica Nv Use of benzo-fused heterocycle sulfamide derivatives for the treatment of substance abuse and addiction
US8937096B2 (en) 2005-12-19 2015-01-20 Janssen Pharmaceutica Nv Use of benzo-fused heterocyle sulfamide derivatives for the treatment of mania and bipolar disorder
US8492431B2 (en) 2005-12-19 2013-07-23 Janssen Pharmaceutica, N.V. Use of benzo-fused heterocycle sulfamide derivatives for the treatment of obesity
US20070191461A1 (en) * 2006-02-15 2007-08-16 Smith-Swintosky Virginia L Use of benzo-heteroaryl sulfamide derivatives for the treatment of migraine
EP2026790A2 (de) 2006-05-19 2009-02-25 Janssen Pharmaceutica, N.V. Kombinationstherapie zur behandlung von epilepsie und assoziierten erkrankungen
US8653066B2 (en) 2006-10-09 2014-02-18 Charleston Laboratories, Inc. Pharmaceutical compositions
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US8815939B2 (en) 2008-07-22 2014-08-26 Janssen Pharmaceutica Nv Substituted sulfamide derivatives
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US10383816B2 (en) 2015-03-02 2019-08-20 Afgin Pharma, Llc Topical regional neuro-affective therapy with cannabinoid combination products
US10494405B2 (en) 2015-05-15 2019-12-03 The Regents Of The University Of Michigan Methods and compositions for the treatment of arthritis
WO2017152130A1 (en) 2016-03-04 2017-09-08 Charleston Laboratories, Inc. Pharmaceutical compositions
US20180049994A1 (en) 2016-08-16 2018-02-22 Afgin Pharma, Llc Topical regional neuro-affective therapy with caryophyllene
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US11364225B2 (en) * 2019-08-21 2022-06-21 Bn Intellectual Properties, Inc. Pharmaceutical formulation for treating symptoms of migraine and cluster headaches, and method of using the same
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GB8615599D0 (en) * 1986-06-26 1986-07-30 Glaxo Group Ltd Chemical compounds
GB8928208D0 (en) * 1989-12-13 1990-02-14 Glaxo Group Ltd Medicaments

Also Published As

Publication number Publication date
AP230A (en) 1993-01-27
CH684192A5 (fr) 1994-07-29
EG20219A (en) 1997-11-30
GB2251614A (en) 1992-07-15
ATE119881T1 (de) 1995-04-15
ITRM910922A1 (it) 1993-06-11
CA2098302A1 (en) 1992-06-13
JPH06503560A (ja) 1994-04-21
CA2098302C (en) 2001-10-16
EP0490689B1 (de) 1995-03-15
HU211937A9 (en) 1996-01-29
GB9126297D0 (en) 1992-02-12
YU191491A (sh) 1994-04-05
PT99757B (pt) 1999-05-31
FR2670487B1 (fr) 1993-08-20
MX9102501A (es) 1992-09-01
CN1050831C (zh) 2000-03-29
TW300886B (de) 1997-03-21
CN1128259A (zh) 1996-08-07
PT99757A (pt) 1992-12-31
ES2069836T3 (es) 1995-05-16
YU48926B (sh) 2002-12-10
NZ240942A (en) 1994-03-25
IE62894B1 (en) 1995-03-08
AU650706B2 (en) 1994-06-30
DE69108200T2 (de) 1995-07-20
CZ281931B6 (cs) 1997-04-16
AP9100339A0 (en) 1992-01-31
US5705520A (en) 1998-01-06
IT1252868B (it) 1995-06-28
IS1706B (is) 1998-12-10
CY2005A (en) 1997-12-05
GB2251614B (en) 1994-12-14
US5554639A (en) 1996-09-10
MY109265A (en) 1996-12-31
GB9026998D0 (en) 1991-01-30
CN1063099A (zh) 1992-07-29
ZA919750B (en) 1992-10-28
IL100330A0 (en) 1992-09-06
HK82697A (en) 1997-06-27
NL9102071A (nl) 1992-07-01
IE914317A1 (en) 1992-06-17
TW205035B (de) 1993-05-01
DE69108200D1 (de) 1995-04-20
JP2994037B2 (ja) 1999-12-27
EP0490689A1 (de) 1992-06-17
BE1005085A3 (fr) 1993-04-13
ITRM910922A0 (it) 1991-12-11
CN1030890C (zh) 1996-02-07
DK0490689T3 (da) 1995-05-22
WO1992010477A1 (en) 1992-06-25
CZ114093A3 (en) 1994-02-16
FR2670487A1 (fr) 1992-06-19
KR100211479B1 (ko) 1999-08-02
RU2108328C1 (ru) 1998-04-10
IL100330A (en) 1996-06-18
AU9072091A (en) 1992-07-08
IS3790A7 (is) 1992-06-13

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