GB0117577D0 - Novel heterocyclic substituted carbonyl derivatives and their use as dopamine D receptor ligands - Google Patents

Novel heterocyclic substituted carbonyl derivatives and their use as dopamine D receptor ligands

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Publication number
GB0117577D0
GB0117577D0 GBGB0117577.7A GB0117577A GB0117577D0 GB 0117577 D0 GB0117577 D0 GB 0117577D0 GB 0117577 A GB0117577 A GB 0117577A GB 0117577 D0 GB0117577 D0 GB 0117577D0
Authority
GB
United Kingdom
Prior art keywords
dopamine
receptor ligands
substituted carbonyl
heterocyclic substituted
novel heterocyclic
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
GBGB0117577.7A
Other languages
English (en)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Aventis Pharmaceuticals Inc
Original Assignee
Aventis Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aventis Pharmaceuticals Inc filed Critical Aventis Pharmaceuticals Inc
Publication of GB0117577D0 publication Critical patent/GB0117577D0/en
Priority to AT05018120T priority Critical patent/ATE412638T1/de
Priority to ES05018120T priority patent/ES2317116T3/es
Priority to DK05018120T priority patent/DK1632483T3/da
Priority to MXPA03006943A priority patent/MXPA03006943A/es
Priority to AU2002250107A priority patent/AU2002250107B8/en
Priority to EP02718999A priority patent/EP1362039B1/en
Priority to EP08004461A priority patent/EP1935887B1/en
Priority to CA002438264A priority patent/CA2438264A1/en
Priority to DE60235130T priority patent/DE60235130D1/de
Priority to EP05018120A priority patent/EP1632483B1/en
Priority to ES02718999T priority patent/ES2253526T3/es
Priority to IL15741302A priority patent/IL157413A0/xx
Priority to AT02718999T priority patent/ATE313534T1/de
Priority to AT08004461T priority patent/ATE455108T1/de
Priority to PT05018120T priority patent/PT1632483E/pt
Priority to DE60208157T priority patent/DE60208157T2/de
Priority to JP2002565962A priority patent/JP4685331B2/ja
Priority to PCT/US2002/004713 priority patent/WO2002066446A1/en
Priority to DE60229673T priority patent/DE60229673D1/de
Priority to DK02718999T priority patent/DK1362039T3/da
Priority to US10/819,037 priority patent/US7186724B2/en
Priority to US11/714,047 priority patent/US7521445B2/en
Priority to JP2009097550A priority patent/JP2009185055A/ja
Priority to JP2009097547A priority patent/JP2009185054A/ja
Priority to US12/425,731 priority patent/US7772252B2/en
Ceased legal-status Critical Current

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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
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AT08004461T ATE455108T1 (de) 2001-02-16 2002-02-15 Heterocyclische substituierte carbonyl derivate und ihre verwendung als dopamin d3 rezeptor liganden
DK02718999T DK1362039T3 (da) 2001-02-16 2002-02-15 Heterocykliske, substituerede carbonylderivater og deres anvendelse som dopamin D3-receptorligander
AT02718999T ATE313534T1 (de) 2001-02-16 2002-02-15 Heterocyclische substituierte carbonyl derivate und ihre verwendung als dopamin d3 rezeptor liganden
DK05018120T DK1632483T3 (da) 2001-02-16 2002-02-15 Heterocykliske, substituerede carbonylderivater og deres anvendelse som dopamin-D3-receptorligander
MXPA03006943A MXPA03006943A (es) 2001-02-16 2002-02-15 Derivados de carbonilo sustituidos heterocicliclos y su uso como ligandos para el receptor d3 de la dopamina.
AU2002250107A AU2002250107B8 (en) 2001-02-16 2002-02-15 Heterocyclic substituted carbonyl derivatives and their use as dopamine D3 receptor ligands
EP02718999A EP1362039B1 (en) 2001-02-16 2002-02-15 Heterocyclic substituted carbonyl derivatives and their use as dopamine d3 receptor ligands
EP08004461A EP1935887B1 (en) 2001-02-16 2002-02-15 Heterocyclic substituted carbonyl derivatives and their use as dopamine D3 receptor ligands
CA002438264A CA2438264A1 (en) 2001-02-16 2002-02-15 Heterocyclic substituted carbonyl derivatives and their use as dopamine d3 receptor ligands
DE60235130T DE60235130D1 (de) 2001-02-16 2002-02-15 Heterocyclische substituierte carbonyl Derivate und ihre Verwendung als Dopamin D3 rezeptor Liganden
ES05018120T ES2317116T3 (es) 2001-02-16 2002-02-15 Derivados de carbonilos sustituidos heterociclicos y su uso como ligandos del receptor de dopamina d3.
ES02718999T ES2253526T3 (es) 2001-02-16 2002-02-15 Derivados de carbonilo sustituidos heterociclicos y su uso como ligandos de receptores d3 de dopamina.
IL15741302A IL157413A0 (en) 2001-02-16 2002-02-15 Heterocyclic substituted carbonyl derivatives and their use as dopamine d3 receptor ligands
AT05018120T ATE412638T1 (de) 2001-02-16 2002-02-15 Heterocyclische substituierte carbonyl derivate und ihre verwendung als dopamin d3 rezeptor liganden
EP05018120A EP1632483B1 (en) 2001-02-16 2002-02-15 Heterocyclic substituted carbonyl derivatives and their use as dopamine d3 receptor ligands
DE60229673T DE60229673D1 (de) 2001-02-16 2002-02-15 Heterocyclische substituierte carbonyl derivate und ihre verwendung als dopamin d3 rezeptor liganden
DE60208157T DE60208157T2 (de) 2001-02-16 2002-02-15 Heterocyclische substituierte carbonyl derivate und ihre verwendung als dopamin d3 rezeptor liganden
JP2002565962A JP4685331B2 (ja) 2001-02-16 2002-02-15 複素環置換カルボニル誘導体およびドーパミンｄ３受容体リガンドとしてのその使用
PCT/US2002/004713 WO2002066446A1 (en) 2001-02-16 2002-02-15 Heterocyclic substituted carbonyl derivatives and their use as dopamine d3 receptor ligands
PT05018120T PT1632483E (pt) 2001-02-16 2002-02-15 Derivados heterocíclicos de carbonilo substituídos e sua utilização como ligandos do receptor de dopamina d3
US10/819,037 US7186724B2 (en) 2001-02-16 2004-04-06 Heterocyclic substituted carbonyl derivatives and their use as dopamine D3 receptor ligands
US11/714,047 US7521445B2 (en) 2001-02-16 2007-03-05 Heterocyclic substituted carbonyl derivatives and their use as dopamine D3 receptor ligands
JP2009097550A JP2009185055A (ja) 2001-02-16 2009-04-14 複素環置換カルボニル誘導体およびドーパミンｄ３受容体リガンドとしてのその使用
JP2009097547A JP2009185054A (ja) 2001-02-16 2009-04-14 複素環置換カルボニル誘導体およびドーパミンｄ３受容体リガンドとしてのその使用
US12/425,731 US7772252B2 (en) 2001-02-16 2009-04-17 Heterocyclic substituted carbonyl derivatives and their use as dopamine D3 receptor ligands

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