CO5370677A1 - Nuevos derivados heterociclicos de carbonil sustituido y su uso como ligantes receptores d3 de dopamina - Google Patents

Nuevos derivados heterociclicos de carbonil sustituido y su uso como ligantes receptores d3 de dopamina

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Publication number
CO5370677A1
CO5370677A1 CO02013028A CO02013028A CO5370677A1 CO 5370677 A1 CO5370677 A1 CO 5370677A1 CO 02013028 A CO02013028 A CO 02013028A CO 02013028 A CO02013028 A CO 02013028A CO 5370677 A1 CO5370677 A1 CO 5370677A1
Authority
CO
Colombia
Prior art keywords
disorders
dopamine
compounds
receptors
disease
Prior art date
Application number
CO02013028A
Other languages
English (en)
Spanish (es)
Inventor
James A Hendrix
Original Assignee
Aventis Pharma Inc
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Filing date
Publication date
Application filed by Aventis Pharma Inc filed Critical Aventis Pharma Inc
Publication of CO5370677A1 publication Critical patent/CO5370677A1/es

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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
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    • A61P25/20—Hypnotics; Sedatives
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    • C07D295/14—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
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    • C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
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CO02013028A 2001-02-16 2002-02-15 Nuevos derivados heterociclicos de carbonil sustituido y su uso como ligantes receptores d3 de dopamina CO5370677A1 (es)

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