DE60229673D1 - Heterocyclische substituierte carbonyl derivate und ihre verwendung als dopamin d3 rezeptor liganden - Google Patents

Heterocyclische substituierte carbonyl derivate und ihre verwendung als dopamin d3 rezeptor liganden

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Publication number
DE60229673D1
DE60229673D1 DE60229673T DE60229673T DE60229673D1 DE 60229673 D1 DE60229673 D1 DE 60229673D1 DE 60229673 T DE60229673 T DE 60229673T DE 60229673 T DE60229673 T DE 60229673T DE 60229673 D1 DE60229673 D1 DE 60229673D1
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Germany
Prior art keywords
dopamine
receptor ligands
substituted carbonyl
heterocyclic substituted
carbonyl derivatives
Prior art date
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Expired - Lifetime
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DE60229673T
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German (de)
English (en)
Inventor
James A Hendrix
Horst Hemmerle
Matthias Urmann
Gregory M Shutske
Joseph T Strupczewski
Kenneth J Bordeau
John G Jurcak
Thaddeus Nieduzak
Sharon Anne Jackson
Paul Angell
James P Carey
George E Lee
David M Fink
Jean-Francois Sabuco
Yulin Chiang
Nicola Collar
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Aventis Pharmaceuticals Inc
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Aventis Pharmaceuticals Inc
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Publication of DE60229673D1 publication Critical patent/DE60229673D1/de
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    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
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    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
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    • C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
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DE60229673T 2001-02-16 2002-02-15 Heterocyclische substituierte carbonyl derivate und ihre verwendung als dopamin d3 rezeptor liganden Expired - Lifetime DE60229673D1 (de)

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US7521445B2 (en) 2009-04-21
US7772252B2 (en) 2010-08-10
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