FR2625200A1 - 7-(1-Azetidinyl)-1,4-dihydro-4-oxoquinoline-3-carboxylic acid derivatives, their preparation and their application as medicaments - Google Patents

7-(1-Azetidinyl)-1,4-dihydro-4-oxoquinoline-3-carboxylic acid derivatives, their preparation and their application as medicaments Download PDF

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Publication number
FR2625200A1
FR2625200A1 FR8718289A FR8718289A FR2625200A1 FR 2625200 A1 FR2625200 A1 FR 2625200A1 FR 8718289 A FR8718289 A FR 8718289A FR 8718289 A FR8718289 A FR 8718289A FR 2625200 A1 FR2625200 A1 FR 2625200A1
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FR
France
Prior art keywords
radical
formula
sep
hydrogen atom
dihydro
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
FR8718289A
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English (en)
French (fr)
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FR2625200B1 (enExample
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Esteve Pharmaceuticals SA
Original Assignee
Laboratorios del Dr Esteve SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Laboratorios del Dr Esteve SA filed Critical Laboratorios del Dr Esteve SA
Priority to FR8718289A priority Critical patent/FR2625200A1/fr
Priority to FR888809816A priority patent/FR2634483B2/fr
Priority to US07/290,315 priority patent/US4927926A/en
Priority to JP63335712A priority patent/JPH0813811B2/ja
Priority to DE8888403352T priority patent/DE3876969T2/de
Priority to AT88403352T priority patent/ATE83774T1/de
Priority to EP88403352A priority patent/EP0324298B1/fr
Priority to DD88324257A priority patent/DD283385A5/de
Priority to ES8900318A priority patent/ES2010114A6/es
Priority to SU884613206A priority patent/SU1731055A3/ru
Priority to NO885797A priority patent/NO176605C/no
Priority to DK726188A priority patent/DK726188A/da
Priority to YU237088A priority patent/YU47124B/sh
Priority to PT89352A priority patent/PT89352B/pt
Priority to KR1019880017747A priority patent/KR920004136B1/ko
Priority to AU27578/88A priority patent/AU617735B2/en
Priority to HU886648A priority patent/HU206206B/hu
Priority to ZA889705A priority patent/ZA889705B/xx
Publication of FR2625200A1 publication Critical patent/FR2625200A1/fr
Application granted granted Critical
Publication of FR2625200B1 publication Critical patent/FR2625200B1/fr
Priority to GR920403018T priority patent/GR3006664T3/el
Granted legal-status Critical Current

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D455/00—Heterocyclic compounds containing quinolizine ring systems, e.g. emetine alkaloids, protoberberine; Alkylenedioxy derivatives of dibenzo [a, g] quinolizines, e.g. berberine
    • C07D455/03—Heterocyclic compounds containing quinolizine ring systems, e.g. emetine alkaloids, protoberberine; Alkylenedioxy derivatives of dibenzo [a, g] quinolizines, e.g. berberine containing quinolizine ring systems directly condensed with at least one six-membered carbocyclic ring, e.g. protoberberine; Alkylenedioxy derivatives of dibenzo [a, g] quinolizines, e.g. berberine
    • C07D455/04—Heterocyclic compounds containing quinolizine ring systems, e.g. emetine alkaloids, protoberberine; Alkylenedioxy derivatives of dibenzo [a, g] quinolizines, e.g. berberine containing quinolizine ring systems directly condensed with at least one six-membered carbocyclic ring, e.g. protoberberine; Alkylenedioxy derivatives of dibenzo [a, g] quinolizines, e.g. berberine containing a quinolizine ring system condensed with only one six-membered carbocyclic ring, e.g. julolidine

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
FR8718289A 1987-12-29 1987-12-29 7-(1-Azetidinyl)-1,4-dihydro-4-oxoquinoline-3-carboxylic acid derivatives, their preparation and their application as medicaments Granted FR2625200A1 (en)

Priority Applications (19)

Application Number Priority Date Filing Date Title
FR8718289A FR2625200A1 (en) 1987-12-29 1987-12-29 7-(1-Azetidinyl)-1,4-dihydro-4-oxoquinoline-3-carboxylic acid derivatives, their preparation and their application as medicaments
FR888809816A FR2634483B2 (fr) 1987-12-29 1988-07-20 Derives des acides 7-(1-azetidinyl)-1,4-dihydro-4-oxoquinoleine-3-carboxyliques, leur preparation et leur application en tant que medicaments
US07/290,315 US4927926A (en) 1987-12-29 1988-12-27 Derivatives of 7-(1-azetidinyl)-1,4-dihydro-4-oxo-3-quinolinecarboxylic acids, their preparation and application as medicines
YU237088A YU47124B (sh) 1987-12-29 1988-12-28 Postupak za dobijanje novih derivata 7-(1-azetidinil)-1,4-dihidro-4-oksokinolein-3-karboks ilnih kiselina
AT88403352T ATE83774T1 (de) 1987-12-29 1988-12-28 7-(1-azetidinyl)-1,4-dihydro-4-oxochinolin-3carbons|ure-derivate, ihre herstellung und ihre verwendung als arzneimittel.
EP88403352A EP0324298B1 (fr) 1987-12-29 1988-12-28 Dérivés des acides 7-(1-azétidinyl)-1,4-dihydro-4-oxoquinoléine-3-carboxyliques, leur préparation et leur application en tant que médicaments
DD88324257A DD283385A5 (de) 1987-12-29 1988-12-28 Verfahren zur herstellung von derivaten der 7-(1-azetidinyl)-1,4-dihydro-4-oxoquinolein-3-carboxylsaeure
ES8900318A ES2010114A6 (es) 1987-12-29 1988-12-28 Procedimiento de preparacion de derivados de los acidos 1,4-dihidro-4-oxoquinolein-3-carboxilicos.
SU884613206A SU1731055A3 (ru) 1987-12-29 1988-12-28 Способ получени азетидиновых производных 1,4-дигидро-4-оксохинолин-3-карбоновых кислот
NO885797A NO176605C (no) 1987-12-29 1988-12-28 Analogifremgangsmåte til fremstilling av terapeutisk aktive 7-(1-azetidinyl)-1,4-dihydro-4-okso-3-kinolinkarboksylsyrederivater
JP63335712A JPH0813811B2 (ja) 1987-12-29 1988-12-28 ７―（１―アセチジニル）―１、４―ジヒドロ―４―オキソキノリン―３―カルボン酸の誘導体、その製造法、およびその医薬としての用途
DE8888403352T DE3876969T2 (de) 1987-12-29 1988-12-28 7-(1-azetidinyl)-1,4-dihydro-4-oxochinolin-3-carbonsaeure-derivate, ihre herstellung und ihre verwendung als arzneimittel.
PT89352A PT89352B (pt) 1987-12-29 1988-12-28 Processo para a preparacao de derivados dos acidos 7-(1-azetidinil)-1,4-dihidro-4-oxoquinoleina-3-carboxilicos e de composicoes farmaceuticas que os contem
DK726188A DK726188A (da) 1987-12-29 1988-12-28 Quinolinderivater
KR1019880017747A KR920004136B1 (ko) 1987-12-29 1988-12-29 7-(1-아제티디닐)-1,4-디히드로-4-옥소-3-퀴놀린카르복실산의 유도체 및 그의 제조방법
AU27578/88A AU617735B2 (en) 1987-12-29 1988-12-29 Derivatives of 7-(1-azetidinyl)-1,4-dihydro-4-oxo-3- guinolinecarboxylic acids, their preparation and application as medicines
HU886648A HU206206B (en) 1987-12-29 1988-12-29 Process for producing 7-/1-azetidinyl/-1,4-dihydro-4-oxo-3-quinoline- carboxylic acid derivatives and pharmaceutical compositions comprising same as active ingredient
ZA889705A ZA889705B (en) 1987-12-29 1988-12-29 Derivatives of 7-(1-azetidinyl)-1,4-dihydro-4-oxo-3-quinoline-carboxylic acids,their preparation and application as medicines
GR920403018T GR3006664T3 (enExample) 1987-12-29 1992-12-24

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR8718289A FR2625200A1 (en) 1987-12-29 1987-12-29 7-(1-Azetidinyl)-1,4-dihydro-4-oxoquinoline-3-carboxylic acid derivatives, their preparation and their application as medicaments

Publications (2)

Publication Number Publication Date
FR2625200A1 true FR2625200A1 (en) 1989-06-30
FR2625200B1 FR2625200B1 (enExample) 1991-04-12

Family

ID=9358387

Family Applications (1)

Application Number Title Priority Date Filing Date
FR8718289A Granted FR2625200A1 (en) 1987-12-29 1987-12-29 7-(1-Azetidinyl)-1,4-dihydro-4-oxoquinoline-3-carboxylic acid derivatives, their preparation and their application as medicaments

Country Status (4)

Country Link
DD (1) DD283385A5 (enExample)
FR (1) FR2625200A1 (enExample)
SU (1) SU1731055A3 (enExample)
ZA (1) ZA889705B (enExample)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2005026146A1 (en) * 2003-09-12 2005-03-24 Warner-Lambert Company Llc Azetidinyl quinolones as antibacterial agents

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5527910A (en) * 1992-12-30 1996-06-18 Cheil Foods & Chemicals, Inc. Pyridone carboxylic acid compounds and their uses for treating infectious diseases caused by bacteria
EP1015445B1 (en) * 1997-09-15 2009-02-25 The Procter & Gamble Company Antimicrobial quinolones, their compositions and uses

Citations (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0106489A2 (en) * 1982-09-09 1984-04-25 Warner-Lambert Company Antibacterial agents
EP0047005B1 (en) * 1980-09-02 1984-11-14 Daiichi Seiyaku Co., Ltd. Benzoxazine derivatives
US4617308A (en) * 1985-01-25 1986-10-14 Warner-Lambert Company 7-substituted amino-1-aryl-6,8-difluoro-1,4-dihydro-4-oxo-3-quinolinecarboxylic acids and derivatives thereof as antibacterial agents
EP0241206A2 (en) * 1986-03-31 1987-10-14 Sankyo Company Limited Quinoline-3-carboxylic acid derivatives, their preparation and use

Patent Citations (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0047005B1 (en) * 1980-09-02 1984-11-14 Daiichi Seiyaku Co., Ltd. Benzoxazine derivatives
EP0106489A2 (en) * 1982-09-09 1984-04-25 Warner-Lambert Company Antibacterial agents
US4617308A (en) * 1985-01-25 1986-10-14 Warner-Lambert Company 7-substituted amino-1-aryl-6,8-difluoro-1,4-dihydro-4-oxo-3-quinolinecarboxylic acids and derivatives thereof as antibacterial agents
EP0241206A2 (en) * 1986-03-31 1987-10-14 Sankyo Company Limited Quinoline-3-carboxylic acid derivatives, their preparation and use

Non-Patent Citations (1)

* Cited by examiner, † Cited by third party
Title
CHEMICAL & PHARMACEUTICAL BULLETIN, vol. 32, no. 12, décembre 1984, page 4907; I.HAYAKAWA et al.: "Synthesis and antibacterial activities of substituted 7-Oxo-2,3-dihydro-7H-pyrido[1,2,3-deÜ[1,4Übenzoxazine-6-carboxylic acids" *

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2005026146A1 (en) * 2003-09-12 2005-03-24 Warner-Lambert Company Llc Azetidinyl quinolones as antibacterial agents

Also Published As

Publication number Publication date
DD283385A5 (de) 1990-10-10
FR2625200B1 (enExample) 1991-04-12
SU1731055A3 (ru) 1992-04-30
ZA889705B (en) 1989-10-25

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