FI974180A0 - Spirosyklisiä ja bisyklisiä diatsinyyli- ja karbatsinyylioksatsolidinoneja - Google Patents
Spirosyklisiä ja bisyklisiä diatsinyyli- ja karbatsinyylioksatsolidinonejaInfo
- Publication number
- FI974180A0 FI974180A0 FI974180A FI974180A FI974180A0 FI 974180 A0 FI974180 A0 FI 974180A0 FI 974180 A FI974180 A FI 974180A FI 974180 A FI974180 A FI 974180A FI 974180 A0 FI974180 A0 FI 974180A0
- Authority
- FI
- Finland
- Prior art keywords
- pct
- carbazinyloxazolidinones
- spirocyclic
- date nov
- sec
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/54—Spiro-condensed
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Communicable Diseases (AREA)
- Pharmacology & Pharmacy (AREA)
- Oncology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US43870595A | 1995-05-11 | 1995-05-11 | |
PCT/US1996/005202 WO1996035691A1 (en) | 1995-05-11 | 1996-04-18 | Spirocyclic and bicyclic diazinyl and carbazinyl oxazolidinones |
Publications (2)
Publication Number | Publication Date |
---|---|
FI974180A0 true FI974180A0 (fi) | 1997-11-10 |
FI974180A FI974180A (fi) | 1997-11-10 |
Family
ID=23741700
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
FI974180A FI974180A (fi) | 1995-05-11 | 1997-11-10 | Spirosyklisiä ja bisyklisiä diatsinyyli- ja karbatsinyylioksatsolidinoneja |
Country Status (18)
Country | Link |
---|---|
US (1) | US6090820A (fi) |
EP (1) | EP0828741B1 (fi) |
JP (1) | JPH11506430A (fi) |
KR (1) | KR100463771B1 (fi) |
CN (2) | CN1068328C (fi) |
AT (1) | ATE204874T1 (fi) |
AU (1) | AU702752B2 (fi) |
CA (1) | CA2218088A1 (fi) |
DE (1) | DE69614847T2 (fi) |
DK (1) | DK0828741T3 (fi) |
ES (1) | ES2162047T3 (fi) |
FI (1) | FI974180A (fi) |
HK (2) | HK1009449A1 (fi) |
MX (1) | MX9708627A (fi) |
NO (1) | NO311298B1 (fi) |
NZ (1) | NZ306310A (fi) |
PT (1) | PT828741E (fi) |
WO (1) | WO1996035691A1 (fi) |
Families Citing this family (46)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6277985B1 (en) * | 1995-09-15 | 2001-08-21 | Pharmacia & Upjohn Company | Aminoaryl oxazolidinone N-oxides |
GB9601666D0 (en) * | 1996-01-27 | 1996-03-27 | Zeneca Ltd | Chemical compounds |
GB9702213D0 (en) | 1996-02-24 | 1997-03-26 | Zeneca Ltd | Chemical compounds |
SG85683A1 (en) * | 1996-04-11 | 2002-01-15 | Upjohn Co | Process to prepare oxazolidinones |
GB9609919D0 (en) * | 1996-05-11 | 1996-07-17 | Zeneca Ltd | Chemical compounds |
GB9717804D0 (en) | 1997-08-22 | 1997-10-29 | Zeneca Ltd | Chemical compounds |
GB9717807D0 (en) | 1997-08-22 | 1997-10-29 | Zeneca Ltd | Chemical compounds |
KR100467309B1 (ko) * | 1997-09-04 | 2005-07-18 | 씨제이 주식회사 | 옥사졸리디논유도체및그의제조방법및항균제조성물 |
KR100463111B1 (ko) * | 1997-10-30 | 2005-06-13 | 씨제이 주식회사 | 신규한옥사졸리디논유도체및제조방법및그를함유하는항균제조성물 |
GB9725244D0 (en) | 1997-11-29 | 1998-01-28 | Zeneca Ltd | Chemical compounds |
HUP0103082A3 (en) | 1998-06-05 | 2002-12-28 | Astrazeneca Ab | Oxazolidinone derivatives, process for their preparation and pharmaceutical compositions containing them |
US6413981B1 (en) | 1999-08-12 | 2002-07-02 | Ortho-Mcneil Pharamceutical, Inc. | Bicyclic heterocyclic substituted phenyl oxazolidinone antibacterials, and related compositions and methods |
US6608081B2 (en) | 1999-08-12 | 2003-08-19 | Ortho-Mcneil Pharmaceutical, Inc. | Bicyclic heterocyclic substituted phenyl oxazolidinone antibacterials, and related compositions and methods |
US6297242B1 (en) | 1999-08-12 | 2001-10-02 | Ortho-Mcneil Pharmaceutical, Inc. | N-substituted amidine and guanidine oxazolidinone antibacterials and methods of use thereof |
GB9928568D0 (en) | 1999-12-03 | 2000-02-02 | Zeneca Ltd | Chemical compounds |
US6518285B2 (en) | 1999-12-21 | 2003-02-11 | Ortho Mcneil Pharmaceutical, Inc. | Piperidinyloxy and pyrrolidinyloxy oxazolidinone antibacterials |
GB0009803D0 (en) * | 2000-04-25 | 2000-06-07 | Astrazeneca Ab | Chemical compounds |
ITVA20000023A1 (it) * | 2000-07-19 | 2002-01-19 | Lamberti Spa | Composizioni di pvc stabili al calore. |
SE0100326D0 (sv) * | 2001-02-02 | 2001-02-02 | Astrazeneca Ab | New compounds |
BR0207952A (pt) | 2001-03-07 | 2004-07-27 | Pfizer Prod Inc | Moduladores da atividade de receptores de quimiocina |
CA2463794A1 (en) * | 2001-11-29 | 2003-06-12 | Merck & Co., Inc. | Cyclopropyl hexane containing oxazolidinone antibiotics and derivatives thereof |
AR038536A1 (es) | 2002-02-25 | 2005-01-19 | Upjohn Co | N-aril-2-oxazolidinona-5- carboxamidas y sus derivados |
US7141588B2 (en) | 2002-02-25 | 2006-11-28 | Pfizer, Inc. | N-aryl-2-oxazolidinone-5-carboxamides and their derivatives |
EP1539745B1 (en) | 2002-08-12 | 2006-03-29 | Pharmacia & Upjohn Company LLC | N-aryl-2-oxazolidinones and their derivatives |
KR100454099B1 (ko) * | 2002-08-22 | 2004-10-26 | 한국화학연구원 | 제초활성을 갖는9-(5-이속사졸린메톡시페닐)이미노-8-치아-1,6-디아자비시클로[4.3.0]노난-7-온 유도체 |
ATE344036T1 (de) | 2002-11-21 | 2006-11-15 | Pharmacia & Upjohn Co Llc | N-(4-(piperazin-1-yl)-phenyl-2-oxazolidinon-5- carbonsäureamid-derivate und verwandte verbindungen als antibakterielle mittel |
DE602004027811D1 (de) | 2003-07-02 | 2010-08-05 | Kyorin Seiyaku Kk | Cyclopropylgruppensubstituierte oxazolidinonantibiotika und derivate davon |
US7304050B2 (en) | 2003-09-16 | 2007-12-04 | Pfizer Inc. | Antibacterial agents |
EP1671972A1 (en) * | 2004-11-24 | 2006-06-21 | Pfizer Limited | Octahydropyrrolo[3,4-c]pyrrole derivatives |
EP1846409A1 (en) * | 2004-11-24 | 2007-10-24 | Pfizer Limited | Octahydropyrrolo[3,4-c]pyrrole derivatives |
KR100729344B1 (ko) * | 2006-02-16 | 2007-06-15 | 스마텍(주) | 차량용 사방 감지 카메라의 보호 및 작동 구조 |
US7728031B2 (en) | 2006-02-24 | 2010-06-01 | Abbott Laboratories | Octahydro-pyrrolo[3,4-b]pyrrole derivatives |
EP2188288A1 (en) | 2007-09-11 | 2010-05-26 | Abbott Laboratories | Octahydro-pyrrolo[3,4-b]pyrrole n-oxides |
US8841306B2 (en) | 2008-11-20 | 2014-09-23 | Panacea Biotec Ltd. | Antimicrobials |
CN102803224A (zh) | 2009-06-26 | 2012-11-28 | 万能药生物有限公司 | 新的氮杂双环己烷类化合物 |
US20130296569A1 (en) | 2010-11-03 | 2013-11-07 | Vijaykumar Jagdishwar Patil | Process for the preparation of phosphoric acid mono-(1--4-methoxymethyl-piperidin-4-yl) ester |
KR101271224B1 (ko) | 2011-07-05 | 2013-06-10 | 한국과학기술연구원 | 항균활성을 갖는 신규 이중고리를 포함하는 옥사졸리디논 유도체 및 이의 제조방법 |
US9487545B2 (en) | 2011-09-30 | 2016-11-08 | Xuanzhu Pharma Co., Ltd. | Fused ring-containing oxazolidinones antibiotics |
WO2015173664A1 (en) | 2014-05-14 | 2015-11-19 | Wockhardt Limited | Process for the preparation of (5s)-n-{3-[3,5-difluoro-4-(4-hydroxy-4-methoxymethyl-piperidin-1-yl)-phenyl]-2-oxo-oxazolidin-5-ylmethyl}-acetamide |
KR20180022826A (ko) | 2015-07-02 | 2018-03-06 | 얀센 사이언시즈 아일랜드 유씨 | 항균 화합물 |
EP3932917A3 (en) | 2015-07-17 | 2022-03-30 | The Global Alliance for TB Drug Development, Inc. | Substituted phenyloxazolidinones for antimicrobial therapy |
CN107400126A (zh) * | 2016-05-19 | 2017-11-28 | 陕西合成药业股份有限公司 | 新型噁唑烷酮类化合物及其制备方法和在医学上的应用 |
CA3026010A1 (en) | 2016-06-16 | 2017-12-21 | Janssen Sciences Ireland Unlimited Company | Heterocyclic compounds as antibacterials |
JP7307682B2 (ja) | 2017-03-01 | 2023-07-12 | ヤンセン・サイエンシズ・アイルランド・アンリミテッド・カンパニー | 併用療法 |
CN108727406B (zh) | 2017-03-28 | 2021-12-07 | 北京协和制药二厂 | 含氮杂环取代的苯并噁嗪噁唑烷酮类化合物及其制备方法和用途 |
WO2020234636A1 (en) | 2019-05-17 | 2020-11-26 | Cadila Healthcare Limited | Novel compounds for the treatment of mammalian infections |
Family Cites Families (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4921869A (en) * | 1987-10-09 | 1990-05-01 | E. I. Du Pont De Nemours And Company | Aminomethyl oxooxazolidinyl cycloalkylbenzene derivatives useful as antibacterial agents |
US4801600A (en) * | 1987-10-09 | 1989-01-31 | E. I. Du Pont De Nemours And Company | Aminomethyl oxooxazolidinyl cycloalkylbenzene derivatives useful as antibacterial agents |
CA1320730C (en) * | 1987-10-16 | 1993-07-27 | The Du Pont Merck Pharmaceutical Company | Aminomethyl oxooxazolidinyl aroylbenzene derivatives useful as antibacterial agents |
DE3884563T2 (de) * | 1987-10-21 | 1994-02-17 | Du Pont Merck Pharma | Aminomethyl-oxo-oxazolidinyl-ethenylbenzen-Derivate, nützlich als antibakterielles Mittel. |
US4948801A (en) * | 1988-07-29 | 1990-08-14 | E. I. Du Pont De Nemours And Company | Aminomethyloxooxazolidinyl arylbenzene derivatives useful as antibacterial agents |
ATE201870T1 (de) * | 1988-09-15 | 2001-06-15 | Upjohn Co | 3-(stickstoff substituierte)phenyl-5-beta- amidomethyloxazoliden-2-one |
DK0610265T3 (da) * | 1991-11-01 | 1997-06-09 | Upjohn Co | Substituerede aryl- og heteroarylphenyloxazolidioner, som kan anvendes som antibakterielle midler |
SK283420B6 (sk) * | 1992-05-08 | 2003-07-01 | Pharmacia & Upjohn Company | Antimikrobiálne oxazolidinóny obsahujúce substituované diazínové skupiny |
MY115155A (en) * | 1993-09-09 | 2003-04-30 | Upjohn Co | Substituted oxazine and thiazine oxazolidinone antimicrobials. |
JPH0873455A (ja) * | 1994-03-15 | 1996-03-19 | Upjohn Co:The | オキサゾリジノン誘導体及びこれを有効成分とする医薬組成物 |
-
1996
- 1996-04-18 DK DK96911768T patent/DK0828741T3/da active
- 1996-04-18 ES ES96911768T patent/ES2162047T3/es not_active Expired - Lifetime
- 1996-04-18 US US09/202,195 patent/US6090820A/en not_active Expired - Fee Related
- 1996-04-18 AT AT96911768T patent/ATE204874T1/de not_active IP Right Cessation
- 1996-04-18 PT PT96911768T patent/PT828741E/pt unknown
- 1996-04-18 WO PCT/US1996/005202 patent/WO1996035691A1/en active IP Right Grant
- 1996-04-18 DE DE69614847T patent/DE69614847T2/de not_active Expired - Fee Related
- 1996-04-18 JP JP8534070A patent/JPH11506430A/ja not_active Withdrawn
- 1996-04-18 CA CA002218088A patent/CA2218088A1/en not_active Abandoned
- 1996-04-18 KR KR1019970707926A patent/KR100463771B1/ko not_active IP Right Cessation
- 1996-04-18 NZ NZ306310A patent/NZ306310A/en unknown
- 1996-04-18 MX MX9708627A patent/MX9708627A/es not_active IP Right Cessation
- 1996-04-18 CN CN96193861A patent/CN1068328C/zh not_active Expired - Fee Related
- 1996-04-18 AU AU54849/96A patent/AU702752B2/en not_active Ceased
- 1996-04-18 EP EP96911768A patent/EP0828741B1/en not_active Expired - Lifetime
-
1997
- 1997-11-10 NO NO19975158A patent/NO311298B1/no unknown
- 1997-11-10 FI FI974180A patent/FI974180A/fi unknown
-
1998
- 1998-09-04 HK HK98110441A patent/HK1009449A1/xx not_active IP Right Cessation
-
2000
- 2000-10-31 CN CN00132826A patent/CN1336375A/zh active Pending
-
2002
- 2002-05-31 HK HK02104105.2A patent/HK1042093A1/zh unknown
Also Published As
Publication number | Publication date |
---|---|
MX9708627A (es) | 1998-02-28 |
DE69614847T2 (de) | 2002-04-04 |
FI974180A (fi) | 1997-11-10 |
NO975158L (no) | 1998-01-09 |
AU702752B2 (en) | 1999-03-04 |
KR19990008399A (ko) | 1999-01-25 |
CA2218088A1 (en) | 1996-11-14 |
AU5484996A (en) | 1996-11-29 |
HK1042093A1 (zh) | 2002-08-02 |
DK0828741T3 (da) | 2001-11-26 |
DE69614847D1 (de) | 2001-10-04 |
NZ306310A (en) | 2001-05-25 |
KR100463771B1 (ko) | 2005-05-16 |
EP0828741A1 (en) | 1998-03-18 |
NO311298B1 (no) | 2001-11-12 |
HK1009449A1 (en) | 1999-09-10 |
CN1336375A (zh) | 2002-02-20 |
PT828741E (pt) | 2002-02-28 |
US6090820A (en) | 2000-07-18 |
WO1996035691A1 (en) | 1996-11-14 |
ATE204874T1 (de) | 2001-09-15 |
JPH11506430A (ja) | 1999-06-08 |
CN1068328C (zh) | 2001-07-11 |
NO975158D0 (no) | 1997-11-10 |
EP0828741B1 (en) | 2001-08-29 |
ES2162047T3 (es) | 2001-12-16 |
CN1184481A (zh) | 1998-06-10 |
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