FI970110A - Helico-bakteerin vastaisia heterosyklisiä atsolonijohdannaisia - Google Patents

Helico-bakteerin vastaisia heterosyklisiä atsolonijohdannaisia Download PDF

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Publication number
FI970110A
FI970110A FI970110A FI970110A FI970110A FI 970110 A FI970110 A FI 970110A FI 970110 A FI970110 A FI 970110A FI 970110 A FI970110 A FI 970110A FI 970110 A FI970110 A FI 970110A
Authority
FI
Finland
Prior art keywords
helicobacterial
heterocyclic
azolone
derivatives
azolone derivatives
Prior art date
Application number
FI970110A
Other languages
English (en)
Finnish (fi)
Swedish (sv)
Other versions
FI970110A0 (fi
Inventor
Jan Heeres
Raymond Antoine Stokbroekx
Marc Willems
Robert Jozef Maria Hendrickx
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Publication of FI970110A0 publication Critical patent/FI970110A0/fi
Publication of FI970110A publication Critical patent/FI970110A/fi

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Polymerization Catalysts (AREA)
  • Heterocyclic Compounds Containing Sulfur Atoms (AREA)
FI970110A 1994-07-12 1997-01-10 Helico-bakteerin vastaisia heterosyklisiä atsolonijohdannaisia FI970110A (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP94202018 1994-07-12
PCT/EP1995/002616 WO1996001821A1 (fr) 1994-07-12 1995-07-05 Derives heterocycliques anti-helicobacter d'azolones

Publications (2)

Publication Number Publication Date
FI970110A0 FI970110A0 (fi) 1997-01-10
FI970110A true FI970110A (fi) 1997-01-10

Family

ID=8217031

Family Applications (1)

Application Number Title Priority Date Filing Date
FI970110A FI970110A (fi) 1994-07-12 1997-01-10 Helico-bakteerin vastaisia heterosyklisiä atsolonijohdannaisia

Country Status (20)

Country Link
US (1) US5607932A (fr)
EP (1) EP0770073A1 (fr)
JP (1) JPH10502383A (fr)
CN (1) CN1067999C (fr)
AU (1) AU684986B2 (fr)
BR (1) BR9508380A (fr)
CA (1) CA2194563A1 (fr)
CZ (1) CZ2697A3 (fr)
FI (1) FI970110A (fr)
HU (1) HUT76641A (fr)
IL (1) IL114534A (fr)
MX (1) MX9700338A (fr)
MY (1) MY131785A (fr)
NO (1) NO310289B1 (fr)
NZ (1) NZ290116A (fr)
PL (1) PL318142A1 (fr)
RU (1) RU2152940C1 (fr)
SK (1) SK2197A3 (fr)
WO (1) WO1996001821A1 (fr)
ZA (1) ZA955753B (fr)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR100411190B1 (ko) * 1995-12-26 2004-03-26 에스케이케미칼주식회사 에틸렌글리콜의회수방법
KR20000005291A (ko) 1996-06-25 2000-01-25 다케다 야쿠힌 고교 가부시키가이샤 옥사졸론 유도체 및 항-헬리코박터 파일로리 제제로서의 이의용도
EP0923577A2 (fr) * 1996-06-25 1999-06-23 Takeda Chemical Industries, Ltd. Derives de l'oxazolone et leur utilisation en tant qu'agent anti-helicobacter pylori
WO2006034279A1 (fr) 2004-09-20 2006-03-30 Xenon Pharmaceuticals Inc. Derives heterocycliques et leur utilisation comme agents therapeutiques
AU2005329423A1 (en) 2004-09-20 2006-09-28 Xenon Pharmaceuticals Inc. Heterocyclic derivatives and their use as stearoyl-CoA desaturase inhibitors
TW200626155A (en) 2004-09-20 2006-08-01 Xenon Pharmaceuticals Inc Heterocyclic derivatives and their use as therapeutic agents
BRPI0515478A (pt) 2004-09-20 2008-07-22 Xenon Pharmaceuticals Inc derivados heterocìclicos e seu uso como mediadores de estearoil-coa-desaturase
TW200626154A (en) 2004-09-20 2006-08-01 Xenon Pharmaceuticals Inc Heterocyclic derivatives and their use as therapeutic agents
CN101083982A (zh) 2004-09-20 2007-12-05 泽农医药公司 用于治疗硬脂酰CoA去饱和酶介导的疾病的杂环衍生物
CN101084207A (zh) 2004-09-20 2007-12-05 泽农医药公司 杂环衍生物及其作为硬脂酰CoA去饱和酶抑制剂的用途
BRPI0611187A2 (pt) 2005-06-03 2010-08-24 Xenon Pharmaceuticals Inc derivados aminotiazàis como inibidores da estearoil-coa desaturase humana
CN102119152B (zh) * 2008-06-27 2014-07-02 诺华股份有限公司 有机化合物
EP2852589B1 (fr) 2012-05-22 2021-04-28 Autifony Therapeutics Limited Triazoles en tant qu'inhibiteurs de kv3
US10562887B2 (en) * 2016-05-27 2020-02-18 Bristol-Myers Squibb Company Triazolones and tetrazolones as inhibitors of ROCK

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4791111A (en) * 1985-12-23 1988-12-13 Janssen Pharmaceutica, N.V. [[4-[4-(4-phenyl-1-piperazinyl)phenoxymethyl]-1,3-dioxolan-2-yl]methyl]-1H-imidazoles and 1H-1,2,4-triazoles having anti-microbial properties
CA1331757C (fr) * 1988-02-29 1994-08-30 Janssen Pharmaceutica Naamloze Vennootschap 5-lipoxygenase inhibant les 4-(4-phenyl-1-piperazinyl)phenols
CA2076257A1 (fr) * 1991-09-13 1993-03-14 Jan Heeres Derives de 4-{4-¬4-(4-hydroxyphenyl)-1-piperazinyl|phenyl}-5-methyl-3h-1,2,4-triazol-3-one
TW279864B (fr) * 1993-02-19 1996-07-01 Janssen Pharmaceutica Nv

Also Published As

Publication number Publication date
JPH10502383A (ja) 1998-03-03
CZ2697A3 (en) 1997-09-17
ZA955753B (en) 1997-01-11
RU2152940C1 (ru) 2000-07-20
SK2197A3 (en) 1997-11-05
MY131785A (en) 2007-08-30
NO310289B1 (no) 2001-06-18
NO970086D0 (no) 1997-01-09
HU9700077D0 (en) 1997-02-28
WO1996001821A1 (fr) 1996-01-25
CN1152310A (zh) 1997-06-18
PL318142A1 (en) 1997-05-12
EP0770073A1 (fr) 1997-05-02
MX9700338A (es) 1997-05-31
AU3075595A (en) 1996-02-09
AU684986B2 (en) 1998-01-08
FI970110A0 (fi) 1997-01-10
NZ290116A (en) 1997-11-24
NO970086L (no) 1997-03-10
IL114534A (en) 1999-08-17
IL114534A0 (en) 1995-11-27
CA2194563A1 (fr) 1996-01-25
CN1067999C (zh) 2001-07-04
BR9508380A (pt) 1997-12-23
HUT76641A (en) 1997-10-28
US5607932A (en) 1997-03-04

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