FI970110A0 - Helico-bakteerin vastaisia heterosyklisiä atsolonijohdannaisia - Google Patents

Helico-bakteerin vastaisia heterosyklisiä atsolonijohdannaisia

Info

Publication number
FI970110A0
FI970110A0 FI970110A FI970110A FI970110A0 FI 970110 A0 FI970110 A0 FI 970110A0 FI 970110 A FI970110 A FI 970110A FI 970110 A FI970110 A FI 970110A FI 970110 A0 FI970110 A0 FI 970110A0
Authority
FI
Finland
Prior art keywords
helicobacterial
heterocyclic
azolone
derivatives
azolone derivatives
Prior art date
Application number
FI970110A
Other languages
English (en)
Swedish (sv)
Other versions
FI970110A (fi
Inventor
Jan Heeres
Raymond Antoine Stokbroekx
Marc Willems
Robert Jozef Maria Hendrickx
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Publication of FI970110A publication Critical patent/FI970110A/fi
Publication of FI970110A0 publication Critical patent/FI970110A0/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Compounds Containing Sulfur Atoms (AREA)
  • Polymerization Catalysts (AREA)
FI970110A 1994-07-12 1997-01-10 Helico-bakteerin vastaisia heterosyklisiä atsolonijohdannaisia FI970110A0 (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP94202018 1994-07-12
PCT/EP1995/002616 WO1996001821A1 (en) 1994-07-12 1995-07-05 Anti-helicobacter heterocyclic derivatives of azolones

Publications (2)

Publication Number Publication Date
FI970110A FI970110A (fi) 1997-01-10
FI970110A0 true FI970110A0 (fi) 1997-01-10

Family

ID=8217031

Family Applications (1)

Application Number Title Priority Date Filing Date
FI970110A FI970110A0 (fi) 1994-07-12 1997-01-10 Helico-bakteerin vastaisia heterosyklisiä atsolonijohdannaisia

Country Status (20)

Country Link
US (1) US5607932A (fi)
EP (1) EP0770073A1 (fi)
JP (1) JPH10502383A (fi)
CN (1) CN1067999C (fi)
AU (1) AU684986B2 (fi)
BR (1) BR9508380A (fi)
CA (1) CA2194563A1 (fi)
CZ (1) CZ2697A3 (fi)
FI (1) FI970110A0 (fi)
HU (1) HUT76641A (fi)
IL (1) IL114534A (fi)
MX (1) MX9700338A (fi)
MY (1) MY131785A (fi)
NO (1) NO310289B1 (fi)
NZ (1) NZ290116A (fi)
PL (1) PL318142A1 (fi)
RU (1) RU2152940C1 (fi)
SK (1) SK2197A3 (fi)
WO (1) WO1996001821A1 (fi)
ZA (1) ZA955753B (fi)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR100411190B1 (ko) * 1995-12-26 2004-03-26 에스케이케미칼주식회사 에틸렌글리콜의회수방법
US6169102B1 (en) 1996-06-25 2001-01-02 Takeda Chemical Industries, Ltd. Oxazolone derivatives and their use as anti-Helicobacter pylori agent
WO1997049703A2 (en) * 1996-06-25 1997-12-31 Takeda Chemical Industries, Ltd. Oxazolone derivatives and their use as anti-helicobacter pylori agents
CN101083992A (zh) 2004-09-20 2007-12-05 泽农医药公司 抑制人硬脂酰CoA去饱和酶的哒嗪衍生物
CA2580857A1 (en) 2004-09-20 2006-09-28 Xenon Pharmaceuticals Inc. Heterocyclic derivatives and their use as stearoyl-coa desaturase inhibitors
JP5094398B2 (ja) 2004-09-20 2012-12-12 ゼノン・ファーマシューティカルズ・インコーポレイテッド 複素環式誘導体およびステアロイル−CoAデサチュラーゼのメディエータとしてのそれらの使用
US7919496B2 (en) 2004-09-20 2011-04-05 Xenon Pharmaceuticals Inc. Heterocyclic derivatives for the treatment of diseases mediated by stearoyl-CoA desaturase enzymes
EP1807085B1 (en) 2004-09-20 2013-08-21 Xenon Pharmaceuticals Inc. Heterocyclic derivatives and their use as stearoyl-coa desaturase inhibitors
JP5043668B2 (ja) 2004-09-20 2012-10-10 ゼノン・ファーマシューティカルズ・インコーポレイテッド 複素環誘導体および治療薬としてのそれらの使用
BRPI0515489A (pt) 2004-09-20 2008-07-29 Xenon Pharmaceuticals Inc derivados heterocìclicos e sua utilização como inibidores de estearoil-coa desaturase
WO2007130075A1 (en) 2005-06-03 2007-11-15 Xenon Pharmaceuticals Inc. Aminothiazole derivatives as human stearoyl-coa desaturase inhibitors
EA201100049A1 (ru) 2008-06-27 2011-08-30 Новартис Аг Органические соединения
JP6240667B2 (ja) 2012-05-22 2017-11-29 アウトイフオンイ トヘラペウトイクス リミテッド Kv3阻害剤としてのトリアゾール
WO2017205709A1 (en) * 2016-05-27 2017-11-30 Bristol-Myers Squibb Company Triazolones and tetrazolones as inhibitors of rock

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4791111A (en) * 1985-12-23 1988-12-13 Janssen Pharmaceutica, N.V. [[4-[4-(4-phenyl-1-piperazinyl)phenoxymethyl]-1,3-dioxolan-2-yl]methyl]-1H-imidazoles and 1H-1,2,4-triazoles having anti-microbial properties
CA1331757C (en) * 1988-02-29 1994-08-30 Janssen Pharmaceutica Naamloze Vennootschap 5-lipoxygenase inhibiting 4-(4-phenyl-1-piperazinyl)phenols
CA2076257A1 (en) * 1991-09-13 1993-03-14 Jan Heeres 4-¬4-¬4-(4-hydroxyphenyl)-1- piperazinyl|phenyl|-5-methyl-3h -1,2,4-triazol-3-one derivatives
TW279864B (fi) * 1993-02-19 1996-07-01 Janssen Pharmaceutica Nv

Also Published As

Publication number Publication date
NO970086D0 (no) 1997-01-09
ZA955753B (en) 1997-01-11
EP0770073A1 (en) 1997-05-02
HUT76641A (en) 1997-10-28
HU9700077D0 (en) 1997-02-28
RU2152940C1 (ru) 2000-07-20
CA2194563A1 (en) 1996-01-25
PL318142A1 (en) 1997-05-12
NO310289B1 (no) 2001-06-18
JPH10502383A (ja) 1998-03-03
AU3075595A (en) 1996-02-09
AU684986B2 (en) 1998-01-08
CN1067999C (zh) 2001-07-04
NZ290116A (en) 1997-11-24
CZ2697A3 (en) 1997-09-17
WO1996001821A1 (en) 1996-01-25
FI970110A (fi) 1997-01-10
NO970086L (no) 1997-03-10
IL114534A0 (en) 1995-11-27
CN1152310A (zh) 1997-06-18
MY131785A (en) 2007-08-30
IL114534A (en) 1999-08-17
SK2197A3 (en) 1997-11-05
US5607932A (en) 1997-03-04
MX9700338A (es) 1997-05-31
BR9508380A (pt) 1997-12-23

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