FI965022A0 - Pyratsolo- ja pyrrolopyridiinejä - Google Patents

Pyratsolo- ja pyrrolopyridiinejä

Info

Publication number
FI965022A0
FI965022A0 FI965022A FI965022A FI965022A0 FI 965022 A0 FI965022 A0 FI 965022A0 FI 965022 A FI965022 A FI 965022A FI 965022 A FI965022 A FI 965022A FI 965022 A0 FI965022 A0 FI 965022A0
Authority
FI
Finland
Prior art keywords
pyrrolopyridines
pyrazolo
formulawherein
stress
compounds
Prior art date
Application number
FI965022A
Other languages
English (en)
Swedish (sv)
Other versions
FI965022A (fi
FI112659B (fi
Inventor
Yuhpyng L Chen
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of FI965022A publication Critical patent/FI965022A/fi
Publication of FI965022A0 publication Critical patent/FI965022A0/fi
Application granted granted Critical
Publication of FI112659B publication Critical patent/FI112659B/fi

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/08—Antiepileptics; Anticonvulsants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/26—Psychostimulants, e.g. nicotine, cocaine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/04—Immunostimulants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/10—Drugs for disorders of the endocrine system of the posterior pituitary hormones, e.g. oxytocin, ADH
    • A61P5/12—Drugs for disorders of the endocrine system of the posterior pituitary hormones, e.g. oxytocin, ADH for decreasing, blocking or antagonising the activity of the posterior pituitary hormones
FI965022A 1994-06-16 1996-12-13 Pyratsolopyridiinejä FI112659B (fi)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US26005594A 1994-06-16 1994-06-16
US26005594 1994-06-16
PCT/IB1995/000373 WO1995034563A1 (en) 1994-06-16 1995-05-18 Pyrazolo and pyrrolopyridines
IB9500373 1995-05-18

Publications (3)

Publication Number Publication Date
FI965022A FI965022A (fi) 1996-12-13
FI965022A0 true FI965022A0 (fi) 1996-12-13
FI112659B FI112659B (fi) 2003-12-31

Family

ID=22987613

Family Applications (1)

Application Number Title Priority Date Filing Date
FI965022A FI112659B (fi) 1994-06-16 1996-12-13 Pyratsolopyridiinejä

Country Status (27)

Country Link
US (1) US6248753B1 (fi)
EP (1) EP0765327B1 (fi)
JP (1) JP2891544B2 (fi)
KR (1) KR100235277B1 (fi)
CN (1) CN1056611C (fi)
AT (1) ATE182332T1 (fi)
AU (1) AU687196B2 (fi)
BR (1) BR9502707A (fi)
CA (1) CA2192820C (fi)
CO (1) CO4290424A1 (fi)
CZ (1) CZ287613B6 (fi)
DE (1) DE69510940T2 (fi)
DK (1) DK0765327T3 (fi)
ES (1) ES2135062T3 (fi)
FI (1) FI112659B (fi)
GR (1) GR3031166T3 (fi)
HU (1) HU219911B (fi)
IL (1) IL114003A (fi)
MX (1) MX9606504A (fi)
NO (1) NO307968B1 (fi)
NZ (1) NZ284846A (fi)
PE (1) PE13396A1 (fi)
PL (1) PL181895B1 (fi)
RU (1) RU2135498C1 (fi)
TW (1) TW432064B (fi)
WO (1) WO1995034563A1 (fi)
ZA (1) ZA954679B (fi)

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RU2153494C2 (ru) 1993-10-12 2000-07-27 Дзе Дюпон Мерк Фармасьютикал Компани 1-n-алкил-n-арилпиримидинамины, способ лечения заболеваний, фармацевтическая композиция

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NO307968B1 (no) 2000-06-26
CA2192820A1 (en) 1995-12-21
MX9606504A (es) 1997-03-29
CO4290424A1 (es) 1996-04-17
NZ284846A (en) 1998-12-23
AU2350595A (en) 1996-01-05
DE69510940D1 (de) 1999-08-26
FI965022A (fi) 1996-12-13
PL181895B1 (pl) 2001-10-31
GR3031166T3 (en) 1999-12-31
KR100235277B1 (ko) 1999-12-15
RU2135498C1 (ru) 1999-08-27
DK0765327T3 (da) 1999-11-29
CZ287613B6 (en) 2001-01-17
US6248753B1 (en) 2001-06-19
AU687196B2 (en) 1998-02-19
EP0765327B1 (en) 1999-07-21
NO965378L (no) 1996-12-13
JPH09507855A (ja) 1997-08-12
CA2192820C (en) 2000-11-28
CZ367096A3 (en) 1997-10-15
DE69510940T2 (de) 1999-11-11
HU219911B (hu) 2001-09-28
JP2891544B2 (ja) 1999-05-17
NO965378D0 (no) 1996-12-13
FI112659B (fi) 2003-12-31
ZA954679B (en) 1996-12-09
BR9502707A (pt) 1996-06-04
HUT75776A (en) 1997-05-28
EP0765327A1 (en) 1997-04-02
TW432064B (en) 2001-05-01
IL114003A0 (en) 1995-10-31
IL114003A (en) 1999-12-31
HU9603469D0 (en) 1997-02-28
CN1150803A (zh) 1997-05-28
PL317705A1 (en) 1997-04-28
ES2135062T3 (es) 1999-10-16
ATE182332T1 (de) 1999-08-15
WO1995034563A1 (en) 1995-12-21
CN1056611C (zh) 2000-09-20
PE13396A1 (es) 1996-04-27

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