FI940011A0 - Mono- ja bis-alkyyliaminoantrasykliinit - Google Patents

Mono- ja bis-alkyyliaminoantrasykliinit

Info

Publication number
FI940011A0
FI940011A0 FI940011A FI940011A FI940011A0 FI 940011 A0 FI940011 A0 FI 940011A0 FI 940011 A FI940011 A FI 940011A FI 940011 A FI940011 A FI 940011A FI 940011 A0 FI940011 A0 FI 940011A0
Authority
FI
Finland
Prior art keywords
group
formula
hydrogen
hydroxy
anthracyclines
Prior art date
Application number
FI940011A
Other languages
English (en)
Swedish (sv)
Other versions
FI940011A (fi
FI106204B (fi
Inventor
Alberto Bargiotti
Michele Caruso
Daniela Faiardi
Antonino Suarato
Nicola Mongelli
Original Assignee
Erba Carlo Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Erba Carlo Spa filed Critical Erba Carlo Spa
Publication of FI940011A0 publication Critical patent/FI940011A0/fi
Publication of FI940011A publication Critical patent/FI940011A/fi
Application granted granted Critical
Publication of FI106204B publication Critical patent/FI106204B/fi

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20Carbocyclic rings
    • C07H15/24Condensed ring systems having three or more rings
    • C07H15/252Naphthacene radicals, e.g. daunomycins, adriamycins

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Molecular Biology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
FI940011A 1991-07-05 1994-01-03 Menetelmä mono- ja bis-alkyyliaminoantrasykliiniglykosidien valmistamiseksi FI106204B (fi)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
GB919114549A GB9114549D0 (en) 1991-07-05 1991-07-05 Mono and bis alkylamino-anthracyclines
GB9114549 1991-07-05
EP9201504 1992-07-03
PCT/EP1992/001504 WO1993001201A1 (en) 1991-07-05 1992-07-03 Mono and bis alkylamino-anthracyclines

Publications (3)

Publication Number Publication Date
FI940011A0 true FI940011A0 (fi) 1994-01-03
FI940011A FI940011A (fi) 1994-01-03
FI106204B FI106204B (fi) 2000-12-15

Family

ID=10697877

Family Applications (1)

Application Number Title Priority Date Filing Date
FI940011A FI106204B (fi) 1991-07-05 1994-01-03 Menetelmä mono- ja bis-alkyyliaminoantrasykliiniglykosidien valmistamiseksi

Country Status (24)

Country Link
US (1) US5496808A (fi)
EP (1) EP0521458B1 (fi)
JP (1) JP3153552B2 (fi)
KR (1) KR100235365B1 (fi)
CN (1) CN1031878C (fi)
AT (1) ATE134376T1 (fi)
AU (1) AU661012B2 (fi)
CA (1) CA2112818C (fi)
CZ (1) CZ2494A3 (fi)
DE (1) DE69208400T2 (fi)
FI (1) FI106204B (fi)
GB (1) GB9114549D0 (fi)
GR (1) GR3019429T3 (fi)
HK (1) HK1006460A1 (fi)
HU (1) HU218913B (fi)
IE (1) IE76921B1 (fi)
IL (1) IL102409A (fi)
MX (1) MX9203928A (fi)
NO (1) NO300099B1 (fi)
NZ (1) NZ243450A (fi)
RU (1) RU2118328C1 (fi)
TW (1) TW201753B (fi)
WO (1) WO1993001201A1 (fi)
ZA (1) ZA924971B (fi)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9325420D0 (en) * 1993-12-13 1994-02-16 Erba Carlo Spa 4'-o-sulfonyl-anthracycline derivatives
CA2199734A1 (en) * 1994-09-12 1996-03-21 Fraser Aird Corticotropin release inhibiting factor and methods of using same
ATE176242T1 (de) * 1995-10-16 1999-02-15 Kyowa Hakko Kogyo Kk Uck14-verbindungen
DE19548474A1 (de) * 1995-12-22 1997-06-26 Wacker Chemie Gmbh Aliphatisch ungesättigte Reste aufweisende Organopolysiloxane, deren Herstellung und deren Verwendung in vernetzbaren Massen
GB9613433D0 (en) * 1996-06-26 1996-08-28 Pharmacia Spa Fluoro labelled anthracyclinone and anthracycline derivatives
AU6150498A (en) * 1997-02-07 1998-08-26 Wistar Institute, The Methods and compositions for the inhibition of interleukin-12 production
GB9806324D0 (en) * 1998-03-24 1998-05-20 Pharmacia & Upjohn Spa Antitumour synergetic composition
GB9904386D0 (en) 1999-02-25 1999-04-21 Pharmacia & Upjohn Spa Antitumour synergistic composition
GB9904387D0 (en) * 1999-02-25 1999-04-21 Pharmacia & Upjohn Spa Antitumour synergistic composition

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU570439B2 (en) * 1983-03-28 1988-03-17 Compression Labs, Inc. A combined intraframe and interframe transform coding system
US4591637A (en) * 1985-01-17 1986-05-27 Sri International Open chain-morpholino adriamycins
FR2591599B1 (fr) * 1985-12-17 1988-08-05 Hoechst Lab Nouvelles anthracyclines et medicaments les contenant
DE3842836A1 (de) * 1988-12-20 1990-06-21 Behringwerke Ag Rhodomycine mit einer modifizierten kohlenhydrat-einheit

Also Published As

Publication number Publication date
CA2112818A1 (en) 1993-01-21
JP3153552B2 (ja) 2001-04-09
HUT70480A (en) 1995-10-30
DE69208400D1 (de) 1996-03-28
HK1006460A1 (en) 1999-02-26
NO940026L (no) 1994-02-16
AU2229492A (en) 1993-02-11
IL102409A (en) 1995-12-08
KR100235365B1 (ko) 1999-12-15
GR3019429T3 (en) 1996-06-30
JPH06508841A (ja) 1994-10-06
CN1031878C (zh) 1996-05-29
CZ2494A3 (en) 1994-07-13
EP0521458B1 (en) 1996-02-21
NO300099B1 (no) 1997-04-07
ATE134376T1 (de) 1996-03-15
DE69208400T2 (de) 1996-06-27
RU2118328C1 (ru) 1998-08-27
FI940011A (fi) 1994-01-03
TW201753B (fi) 1993-03-11
FI106204B (fi) 2000-12-15
IL102409A0 (en) 1993-01-14
AU661012B2 (en) 1995-07-13
CN1069981A (zh) 1993-03-17
US5496808A (en) 1996-03-05
IE922177A1 (en) 1993-01-13
HU9400022D0 (en) 1994-05-30
EP0521458A1 (en) 1993-01-07
MX9203928A (es) 1993-04-01
NO940026D0 (no) 1994-01-04
GB9114549D0 (en) 1991-08-21
WO1993001201A1 (en) 1993-01-21
HU218913B (hu) 2000-12-28
ZA924971B (en) 1993-03-31
CA2112818C (en) 2003-02-04
NZ243450A (en) 1993-11-25
IE76921B1 (en) 1997-11-05

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Legal Events

Date Code Title Description
GB Transfer or assigment of application

Owner name: PHARMACIA & UPJOHN S.P.A.