FI900925A0 - Foerfarande foer framstaellning av nya 19-nor-steroider med en kolvaetekedja i 11b-staellningen och innehaollande en amid- eller karbamatgrupp. - Google Patents

Foerfarande foer framstaellning av nya 19-nor-steroider med en kolvaetekedja i 11b-staellningen och innehaollande en amid- eller karbamatgrupp.

Info

Publication number
FI900925A0
FI900925A0 FI900925A FI900925A FI900925A0 FI 900925 A0 FI900925 A0 FI 900925A0 FI 900925 A FI900925 A FI 900925A FI 900925 A FI900925 A FI 900925A FI 900925 A0 FI900925 A0 FI 900925A0
Authority
FI
Finland
Prior art keywords
alkyl
optionally
steroider
staellningen
kolvaetekedja
Prior art date
Application number
FI900925A
Other languages
English (en)
Finnish (fi)
Inventor
Andr Claussner
Lucien Nedelec
Daniel Philibert
De Velde Patrick Van
Original Assignee
Roussel Uclaf
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Roussel Uclaf filed Critical Roussel Uclaf
Publication of FI900925A0 publication Critical patent/FI900925A0/fi

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C07J41/0033—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
    • C07J41/0077—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 substituted in position 11-beta by a carbon atom, further substituted by a group comprising at least one further carbon atom
    • C07J41/0083—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 substituted in position 11-beta by a carbon atom, further substituted by a group comprising at least one further carbon atom substituted in position 11-beta by an optionally substituted phenyl group not further condensed with other rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C07J41/0033—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
    • C07J41/0077—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 substituted in position 11-beta by a carbon atom, further substituted by a group comprising at least one further carbon atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J43/00—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • C07J43/003—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton not condensed

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Diabetes (AREA)
  • Endocrinology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Other Investigation Or Analysis Of Materials By Electrical Means (AREA)
  • Saccharide Compounds (AREA)
FI900925A 1989-02-24 1990-02-23 Foerfarande foer framstaellning av nya 19-nor-steroider med en kolvaetekedja i 11b-staellningen och innehaollande en amid- eller karbamatgrupp. FI900925A0 (fi)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR8902384A FR2643638B1 (fr) 1989-02-24 1989-02-24 Nouveaux 19-nor steroides ayant en position 11beta une chaine carbonee comportant une fonction amide ou carbamate, leur procede de preparation et les intermediaires de ce procede, leur application comme medicaments et les compositions pharmaceutiques les contenant

Publications (1)

Publication Number Publication Date
FI900925A0 true FI900925A0 (fi) 1990-02-23

Family

ID=9379072

Family Applications (1)

Application Number Title Priority Date Filing Date
FI900925A FI900925A0 (fi) 1989-02-24 1990-02-23 Foerfarande foer framstaellning av nya 19-nor-steroider med en kolvaetekedja i 11b-staellningen och innehaollande en amid- eller karbamatgrupp.

Country Status (23)

Country Link
US (2) US5149696A (pt)
EP (1) EP0384842B1 (pt)
JP (1) JP3009169B2 (pt)
KR (1) KR910015590A (pt)
CN (1) CN1046166A (pt)
AT (1) ATE99320T1 (pt)
AU (1) AU631853B2 (pt)
CA (1) CA2010826A1 (pt)
DE (1) DE69005480T2 (pt)
DK (1) DK0384842T3 (pt)
ES (1) ES2062431T3 (pt)
FI (1) FI900925A0 (pt)
FR (1) FR2643638B1 (pt)
HU (1) HU207341B (pt)
IE (1) IE63483B1 (pt)
IL (1) IL93500A0 (pt)
MA (1) MA21754A1 (pt)
MX (1) MX19599A (pt)
OA (1) OA09195A (pt)
PL (1) PL162151B1 (pt)
PT (1) PT93263B (pt)
TN (1) TNSN90018A1 (pt)
ZA (1) ZA901356B (pt)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2650748B1 (fr) * 1989-08-08 1991-11-08 Roussel Uclaf Nouveaux esters d'acides organiques avec des alcools derives de 19-nor steroides et leurs sels, leur procede de preparation et les intermediaires de ce procede, leur application a titre de medicaments et les compositions les renfermant
DE69128820T2 (de) * 1990-08-14 1998-06-10 Hoechst Marion Roussel Inc Neue 19-Nor Steroide, die eine Amid tragende Gruppe in der 11-Beta-Stelle haben, ihre Herstellung, ihre Verwendung als Medikamente und pharmazeutische Präparate davon
GB9126766D0 (en) * 1991-12-17 1992-02-12 Coombes Raoul C D Pharmaceutical compositions
FR2685332A1 (fr) * 1991-12-20 1993-06-25 Roussel Uclaf Nouveaux 19-nor sterouides ayant en position 11beta une chaine thiocarbonee, leur procede de preparation et les intermediaires et leur application a titre de medicaments.
FR2700548B1 (fr) * 1993-01-20 1995-03-03 Roussel Uclaf Nouveau procédé de préparation de stéroïdes 16 alpha-méthylés.
FR2706454B1 (fr) * 1993-06-17 1995-09-15 Roussel Uclaf Nouveaux 19-Nor stéroïdes, procédé et intermédiaires de préparation, application comme médicaments et compositions pharmaceutiques les contenant.
CA2149496C (en) * 1994-05-19 2006-12-19 Ronald Gebhard 11,21-bisphenyl-19-norpregnane derivatives
JP3744559B2 (ja) * 1995-03-17 2006-02-15 独立行政法人情報通信研究機構 立体カメラ、立体ディスプレイ、及び、立体映像システム
US5929262A (en) * 1995-03-30 1999-07-27 The United States Of America As Represented By The Department Of Health And Human Services Method for preparing 17α-acetoxy-11β-(4-N, N-dimethylaminophyl)-19-Norpregna-4,9-diene-3, 20-dione, intermediates useful in the method, and methods for the preparation of such intermediates
FR2757519B1 (fr) * 1996-12-23 1999-06-11 Hoechst Marion Roussel Inc Steroides substitues en position 11, leur procede de preparation, leur application comme medicament et les compositions pharmaceutiques les renfermant
DE19724187A1 (de) 1997-06-02 1998-12-03 Schering Ag 11beta-Arylsubstituierte 14,17-Ethanoestratriene, Verfahren zur Herstellung dieser Verbindungen, sowie ihre Verwendung zur Herstellung von Arzneimitteln
FR2771096B1 (fr) * 1997-11-17 2000-08-11 Hoechst Marion Roussel Inc Nouveaux 19-nor steroides, substitues en position 11beta, procede et intermediaires de preparation, application comme medicaments et compositions pharmaceutiques les renfermant
US6262042B1 (en) 1998-05-29 2001-07-17 Research Triangle Institute 17β-amino and hydroxylamino-11β-arylsteroids and their derivatives having agonist or antagonist hormonal properties
FR2789993B1 (fr) * 1999-02-22 2003-03-07 Hoechst Marion Roussel Inc Nouveaux derives de steroides, leurs procedes de preparation et intermediaires de ce procede, leur application a titre de medicaments et compositions pharmaceutiques les renfermant
DE19929715A1 (de) * 1999-06-24 2000-12-28 Schering Ag 11ß-langkettig-substituierte Estratriene, Verfahren zur Herstellung , pharmazeutische Präparate, die diese 11ß-langkettig-substituierten Estratriene enthalten, sowie deren Verwendung zur Herstellung von Arzneimitteln
FR2826004B1 (fr) * 2001-06-13 2008-03-28 Aventis Pharma Sa Procede de preparation de derives estrogenes
EP1452293A1 (en) * 2003-02-25 2004-09-01 Mold-Masters Limited Injection molding system with flow control and method of injection molding
DE102009034367A1 (de) * 2009-07-20 2011-01-27 Bayer Schering Pharma Aktiengesellschaft 17-Hydroxy-17-pentafluorethyl-estra-4,9(10)-dien-11-benzyliden-Derivate, Verfahren zu deren Herstellung und deren Verwendung zur Behandlung von Krankheiten
CA2813433C (en) 2010-10-27 2019-08-20 Dignity Health Trimegestone (tmg) for treatment of preterm birth

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2235949B1 (pt) * 1973-06-18 1978-03-17 Roussel Uclaf
ZA8231B (en) * 1981-01-09 1982-11-24 Roussel Uclaf New 11 -substituted steroid derivatives, their preparation, their use as medicaments, the compositions containing them and the new intermediates thus obtained
FR2522328B1 (fr) * 1982-03-01 1986-02-14 Roussel Uclaf Nouveaux produits derives de la structure 3-ceto 4,9 19-nor steroides, leur procede de preparation et leur application comme medicaments
GB8327256D0 (en) * 1983-10-12 1983-11-16 Ici Plc Steroid derivatives
AU580843B2 (en) * 1985-02-07 1989-02-02 Schering Aktiengesellschaft 11``-phenyl-gonanes, their manufacture and pharmaceutical preparations containing them
GB8513723D0 (en) * 1985-05-31 1985-07-03 Erba Farmitalia 11-beta substituted steroids
DE3621024C2 (de) * 1986-06-20 1999-10-28 Schering Ag 11beta-Phenylestradiene, deren Herstellung und diese enthaltende pharmazeutische Präparate

Also Published As

Publication number Publication date
EP0384842A1 (fr) 1990-08-29
PT93263B (pt) 1996-01-31
US5149696A (en) 1992-09-22
AU631853B2 (en) 1992-12-10
MX19599A (es) 1994-04-29
ATE99320T1 (de) 1994-01-15
HU207341B (en) 1993-03-29
OA09195A (fr) 1992-06-30
IL93500A0 (en) 1990-11-29
CN1046166A (zh) 1990-10-17
EP0384842B1 (fr) 1993-12-29
TNSN90018A1 (fr) 1991-03-05
PT93263A (pt) 1990-08-31
PL283941A1 (en) 1991-01-14
US5290771A (en) 1994-03-01
FR2643638A1 (fr) 1990-08-31
JP3009169B2 (ja) 2000-02-14
DE69005480T2 (de) 1994-05-19
IE900662L (en) 1990-08-24
KR910015590A (ko) 1991-09-30
DE69005480D1 (de) 1994-02-10
PL162151B1 (en) 1993-09-30
JPH02268194A (ja) 1990-11-01
CA2010826A1 (fr) 1990-08-24
HUT55032A (en) 1991-04-29
ZA901356B (en) 1991-04-24
AU5007290A (en) 1990-08-30
HU900273D0 (en) 1990-03-28
IE63483B1 (en) 1995-05-03
DK0384842T3 (da) 1994-03-28
ES2062431T3 (es) 1994-12-16
MA21754A1 (fr) 1990-10-01
FR2643638B1 (fr) 1991-06-14

Similar Documents

Publication Publication Date Title
FI900925A0 (fi) Foerfarande foer framstaellning av nya 19-nor-steroider med en kolvaetekedja i 11b-staellningen och innehaollande en amid- eller karbamatgrupp.
DK490288D0 (da) Hidtil ukendte forbindelser
NO893166L (no) Makrocykliske forbindelser.
ATE102193T1 (de) Thiazolidinedionederivate.
DE69112989D1 (de) Aminocoumaranderivate, ihre Herstellung und Verwendung.
KR930016402A (ko) 항-hiv 활성을 갖는 이미다졸 유도체
NO164351C (no) Analogifremgangsmaate for fremstilling av terapeutisk aktive 5-alkyl-l-fenyl-2-piperazinoalkylpyrazolin-3-on-forbindelser.
ATE59844T1 (de) Indolcarboxamidderivate, ihre salze, verfahren und zwischenprodukte, anwendung als heilmittel und zusammensetzungen die sie enthalten.
SE8403268L (sv) 1,4-dihydropyridinderivat, deras framstellning och farmaceutiska beredningar innehallande dessa
ES2058569T3 (es) Derivados de la fenotiazina analgesicas.
IT1159151B (it) Steroidi esterificati nella posizione 17 e tioesterificati nella posizione 21 loro procedimento di preparazione e loro uso medicinale
SE7902788L (sv) Substituerade steroid-spiro-oxazolidinonderivat jemte sett for deras framstellning
FI824043A0 (fi) Foerfarande foer framstaellning av nya cefalosporinderivat, vilka aer substituerade i 3-staellningengruppen heterosyklisk rest-tiometyl
ES524524A0 (es) Procedimiento para la preparacion de un aducto de un diisocianato
SE8008189L (sv) Foreningar med antiallergisk och antiulceros verkan, nemligen 1-oxo-1h-tiazolo(3,2-a)pyrimidin-2-karboxamider och mellanprodukter for dessa
KR880004015A (ko) 감광제 및 중합성 조성물
SE7908439L (sv) Nya beta-laktonderivat av 2-hydroxicyklopentankarboxylsyra, sett for framstellning och anvendning derav som lekemedel samt farmaceutiska kompositioner innehallande dessa foreningar
ATE55123T1 (de) Alkylcarbonsaeureamide von pyridinalkylaminen, ihre herstellung und ihre verwendung als arzneimittel.
FR2448544A1 (fr) Derives de thiazole et leur application en therapeutique
FR2392969A1 (fr) Nouveaux derives d'a-methyl-b-aminopropiophenone et leur utilisation en tant que bronchodilatateurs
SE8106633L (sv) Nya 4-(2,1,3-bensoxadiazol-4-yl)-1,4-dihydro-pyridinderivat, deras framstellning och kompositioner innehallande dessa
JPS5340719A (en) Organophosphorus compound and chlorine-containing resin composition
SE8802162D0 (sv) Nya aminoacylater av glycerolacetal
JPS5325554A (en) 2-omega,omega-bis(alkyulthio)-or omega,omega(alkylenedithio)-alkyl-5-methylfuran and their preparation
ATE24887T1 (de) Cycloaliphatische alkohole.

Legal Events

Date Code Title Description
FD Application lapsed
MM Patent lapsed

Owner name: ROUSSEL-UCLAF