FI820992L - Bis-estrar av 1,1,-alkandioler med 6-beta(hydroxi-metyl)penicillansyra-1,1-dioxid och beta-lactamantibioottika - Google Patents

Bis-estrar av 1,1,-alkandioler med 6-beta(hydroxi-metyl)penicillansyra-1,1-dioxid och beta-lactamantibioottika

Info

Publication number
FI820992L
FI820992L FI820992A FI820992A FI820992L FI 820992 L FI820992 L FI 820992L FI 820992 A FI820992 A FI 820992A FI 820992 A FI820992 A FI 820992A FI 820992 L FI820992 L FI 820992L
Authority
FI
Finland
Prior art keywords
beta
dioxide
bis
penicillansyra
lactamantibiotics
Prior art date
Application number
FI820992A
Other languages
English (en)
Other versions
FI74285C (fi
FI74285B (fi
Inventor
Michael Stephen Kellogg
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of FI820992L publication Critical patent/FI820992L/fi
Application granted granted Critical
Publication of FI74285B publication Critical patent/FI74285B/fi
Publication of FI74285C publication Critical patent/FI74285C/fi

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Cephalosporin Compounds (AREA)
  • Pyrrole Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Apparatus Associated With Microorganisms And Enzymes (AREA)
FI820992A 1981-03-23 1982-03-22 Foerfarande foer framstaellning av terapeutiskt anvaendbara 6- -(d-2-aminofenylacetamido)penicillanoylioximetyl -6'- -(hydroximetyl)penicillanat-1',1'-dioxid och 6- -/d-2-amino-2-(p- hydroxifenyl)acetamido/penicillanoyloximetyl-6'- -(hydroximetyl) penicillanat-1,1'-dioxid samt mellanprodukter som anvaen FI74285C (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US06/246,505 US4342768A (en) 1979-10-22 1981-03-23 Bis-esters of 1,1-alkanediols with 6-beta-hydroxymethylpenicillanic acid 1,1-dioxide and beta-lactam antibiotics
US24650581 1981-03-23

Publications (3)

Publication Number Publication Date
FI820992L true FI820992L (fi) 1982-09-24
FI74285B FI74285B (fi) 1987-09-30
FI74285C FI74285C (fi) 1988-01-11

Family

ID=22930958

Family Applications (1)

Application Number Title Priority Date Filing Date
FI820992A FI74285C (fi) 1981-03-23 1982-03-22 Foerfarande foer framstaellning av terapeutiskt anvaendbara 6- -(d-2-aminofenylacetamido)penicillanoylioximetyl -6'- -(hydroximetyl)penicillanat-1',1'-dioxid och 6- -/d-2-amino-2-(p- hydroxifenyl)acetamido/penicillanoyloximetyl-6'- -(hydroximetyl) penicillanat-1,1'-dioxid samt mellanprodukter som anvaen

Country Status (26)

Country Link
US (1) US4342768A (fi)
EP (1) EP0061313B1 (fi)
JP (1) JPS57169492A (fi)
KR (1) KR860000425B1 (fi)
AT (1) ATE11291T1 (fi)
AU (1) AU527895B2 (fi)
CA (1) CA1201709A (fi)
CS (1) CS228921B2 (fi)
DD (1) DD203723A5 (fi)
DE (1) DE3261898D1 (fi)
DK (1) DK126982A (fi)
ES (1) ES8305769A1 (fi)
FI (1) FI74285C (fi)
GR (1) GR76107B (fi)
GT (1) GT198274394A (fi)
HU (1) HU186487B (fi)
IE (1) IE52812B1 (fi)
IL (1) IL65306A (fi)
NO (1) NO820897L (fi)
NZ (1) NZ200068A (fi)
PH (1) PH18040A (fi)
PL (1) PL130110B1 (fi)
PT (1) PT74624B (fi)
SU (1) SU1122230A3 (fi)
YU (1) YU61882A (fi)
ZA (1) ZA821901B (fi)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU559689B2 (en) * 1981-09-22 1987-03-19 Kureha Kagaku Kogyo K.K. Penicillin derivative
US4452796A (en) * 1982-06-14 1984-06-05 Pfizer Inc. 6-Aminoalkylpenicillanic acid 1,1-dioxides as beta-lactamase inhibitors
EP0084730A1 (en) * 1982-01-22 1983-08-03 Beecham Group Plc Esters of penicillin derivatives with beta-lactamase inhibitors, their preparation and their use
JPS58128387A (ja) * 1982-01-26 1983-07-30 レオ・フア−マシユ−テイカル・プロダクツ・リミテツド・エイ／エス（レ−ベンス・ケミスケ・フアブリツク・プロデユクチオンスアクチ−セルスカブ） 新規β−ラクタム化合物およびその製法と用途
US4462934A (en) * 1983-03-31 1984-07-31 Pfizer Inc. Bis-esters of dicarboxylic acids with amoxicillin and certain hydroxymethylpenicillanate 1,1-dioxides
US4536393A (en) * 1983-06-06 1985-08-20 Pfizer Inc. 6-(Aminomethyl)penicillanic acid 1,1-dioxide esters and intermediates therefor
US4503040A (en) * 1984-02-27 1985-03-05 Pfizer Inc. 6-(Aminoacyloxymethyl)penicillanic acid 1,1-dioxides as beta-lactamase inhibitors
US4591459A (en) * 1984-12-03 1986-05-27 Pfizer Inc. Intermediates for 6-(aminoacyloxymethyl) penicillanic acid 1,1-dioxides
US4675186A (en) * 1985-04-18 1987-06-23 Pfizer Inc. 6-(1-acyl-1-hydroxymethyl)penicillanic acid derivatives
US4762921A (en) * 1985-04-18 1988-08-09 Pfizer Inc. 6-(1-acyl-1-hydroxymethyl)penicillanic acid derivatives
JPS63144296U (fi) * 1987-03-12 1988-09-22
CN108107120B (zh) * 2017-12-12 2020-12-01 山东鑫泉医药有限公司 采用高效液相法测定中间产物6,6-二溴青霉烷酸的方法

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4207323A (en) * 1975-11-21 1980-06-10 Merck & Co., Inc. 6-Substituted methyl penicillins, derivatives and analogues thereof
IE49880B1 (en) 1979-02-13 1986-01-08 Leo Pharm Prod Ltd Penicillin derivatives
US4244951A (en) * 1979-05-16 1981-01-13 Pfizer Inc. Bis-esters of methanediol with penicillins and penicillanic acid 1,1-dioxide

Also Published As

Publication number Publication date
KR860000425B1 (ko) 1986-04-19
IE820656L (en) 1982-09-23
PT74624B (en) 1984-11-26
US4342768A (en) 1982-08-03
JPS6325593B2 (fi) 1988-05-26
DD203723A5 (de) 1983-11-02
EP0061313A2 (en) 1982-09-29
PT74624A (en) 1982-04-01
PL130110B1 (en) 1984-07-31
KR830009110A (ko) 1983-12-17
NO820897L (no) 1982-09-24
ATE11291T1 (de) 1985-02-15
FI74285C (fi) 1988-01-11
JPS57169492A (en) 1982-10-19
HU186487B (en) 1985-08-28
SU1122230A3 (ru) 1984-10-30
ES510656A0 (es) 1983-04-16
IL65306A (en) 1986-02-28
DK126982A (da) 1982-09-24
DE3261898D1 (en) 1985-02-28
NZ200068A (en) 1985-08-16
IL65306A0 (en) 1982-05-31
FI74285B (fi) 1987-09-30
AU527895B2 (en) 1983-03-31
IE52812B1 (en) 1988-03-16
EP0061313A3 (en) 1982-12-08
CS228921B2 (en) 1984-05-14
PL235576A1 (en) 1983-03-14
CA1201709A (en) 1986-03-11
YU61882A (en) 1985-03-20
GR76107B (fi) 1984-08-03
AU8176182A (en) 1982-11-04
EP0061313B1 (en) 1985-01-16
ES8305769A1 (es) 1983-04-16
GT198274394A (es) 1983-09-08
ZA821901B (en) 1983-01-26
PH18040A (en) 1985-03-08

Similar Documents

Publication Publication Date Title
SE8003603L (sv) Bis-estrar av metandiol med penicilliner och penicillansyra-1,1-dioxid
DK543787A (da) Naphthyridin-, quinolin- og benzoxazincarboxylsyreforbindelser med antibakteriel aktivitet
OA05606A (fr) Procédé de préparation de nouvelles acoyloximes dérivées de l'acide 7-amino thiazolyl acétamino oéphalosporanique.
OA05964A (fr) Dérivés de l, l-dioxyde d'acide pénicillanique.
FI820992L (fi) Bis-estrar av 1,1,-alkandioler med 6-beta(hydroxi-metyl)penicillansyra-1,1-dioxid och beta-lactamantibioottika
IT7949678A0 (it) Procedimento per produrre acidi tio metil-3-cefem-4-carbossilici sostituiti come intermedi per cefalosporine
DK166353C (da) Penicillansyre-1,1-dioxid-derivater
ES2052511T3 (es) Acidos 4-halogeno-2-oxiimino-3-oxobutiricos.
ES509782A0 (es) Un procedimiento para la preparacion de nuevos bis-esteres de metanodiol y etanodiol.
IT8025223A0 (it) Procedimento per la produzione di derivati dell'acido penicillanico.
NO160517C (no) Fremgangsmaate for fremstilling av klormetylestere av penicillansyre-sulfon.
MC1421A1 (fr) Derives acyles
FI812331L (fi) Nya kefalosporinderivat deras framstaellning och anvaendning
DE3263337D1 (de) Salts of penicillanic acid 1,1-dioxide
NO162463C (no) Mellomprodukter for fremstilling av derivater av (okso-4-4h-(1)-benzopyran-8-yl)-eddiksyre.
DE68922207T2 (de) Verfahren zur Herstellung von Alkalimetall-Salze von 3,7-substituierten 7-Aminocephalosporansauerderivaten.
ES8505687A1 (es) Procedimiento para la obtencion del ester pivaloiloximetilico del acido penicilanico 1 1-dioxido
IT7919896A0 (it) Procedimento per la preparazione di sali, diversi dal cloridrato, dell'estere ftalidilico dell'acido 6-[d(-)-alfa-aminofenilacetamido]penicillanico.
BA97159B1 (bs) Postupak za dobivanje 1,1-dioksida penicilanske kiseline i njegovih estara
JPS5283491A (en) Preparation of novel penicillin derivatives
IT7919895A0 (it) Procedimento per la preparazione del cloridrato dell'estere ftalidilico dell'acido 6-[d(-)alfaaminofenilacetamido]penicillanico
IT8024849A0 (it) Procedimento per la preparazione di derivati dell'acido 7-amminocefalosporanico.
IT1188790B (it) Combinazioni di 1,1-diossido dell'acido penicillanico con l'acido 7-(d-2-(4-etilpiperazin-2,3-dion-1-carbossammido)-2-(4-idrossifenil)acetammido)-3-(1-metil-5-tetrazolil)tiometil)-3-desacetossimetilcefalosporanico
IT8025307A0 (it) Procedimento migliorato per la purificazione dell'acido 7-amino-3-(5-metil-1,3,4-tiadiazoli l)-3-cefem-4-carbossilico.

Legal Events

Date Code Title Description
MM Patent lapsed

Owner name: PFIZER INC.