FI74010C - Foerfarande foer framstaellning av saosom anxiolyter anvaendbara imidazo/1,2-a/pyrimidiner. - Google Patents
Foerfarande foer framstaellning av saosom anxiolyter anvaendbara imidazo/1,2-a/pyrimidiner. Download PDFInfo
- Publication number
- FI74010C FI74010C FI833055A FI833055A FI74010C FI 74010 C FI74010 C FI 74010C FI 833055 A FI833055 A FI 833055A FI 833055 A FI833055 A FI 833055A FI 74010 C FI74010 C FI 74010C
- Authority
- FI
- Finland
- Prior art keywords
- formula
- compound
- group
- pyrimidin
- imidazo
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
- C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
- C07D239/72—Quinazolines; Hydrogenated quinazolines
- C07D239/95—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in positions 2 and 4
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Psychiatry (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Veterinary Medicine (AREA)
- Neurology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Pain & Pain Management (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB8224606 | 1982-08-27 | ||
| GB8224606 | 1982-08-27 | ||
| GB838303612A GB8303612D0 (en) | 1983-02-09 | 1983-02-09 | Imidazo 1,2-a pyrimidines |
| GB8303612 | 1983-02-09 |
Publications (4)
| Publication Number | Publication Date |
|---|---|
| FI833055A0 FI833055A0 (fi) | 1983-08-26 |
| FI833055L FI833055L (fi) | 1984-02-28 |
| FI74010B FI74010B (fi) | 1987-08-31 |
| FI74010C true FI74010C (fi) | 1987-12-10 |
Family
ID=26283682
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| FI833055A FI74010C (fi) | 1982-08-27 | 1983-08-26 | Foerfarande foer framstaellning av saosom anxiolyter anvaendbara imidazo/1,2-a/pyrimidiner. |
Country Status (19)
Families Citing this family (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IL69417A (en) * | 1982-08-27 | 1987-12-20 | Roussel Uclaf | 2-acyl imidazo(1,2-a)pyrimidines,their preparation and pharmaceutical compositions containing them |
| GB8334210D0 (en) * | 1983-12-22 | 1984-02-01 | Roussel Lab Ltd | Imidazo(1 2-c)pyrimidines |
| GB8432073D0 (en) * | 1984-12-19 | 1985-01-30 | Roussel Lab Ltd | Chemical compounds |
| GB8613591D0 (en) * | 1986-06-04 | 1986-07-09 | Roussel Lab Ltd | Chemical compounds |
| GB8620060D0 (en) * | 1986-08-18 | 1986-10-01 | Roussel Lab Ltd | Chemical compounds |
| US4731446A (en) * | 1987-05-01 | 1988-03-15 | The Dow Chemical Company | Imidazo[1,2-a]pyrimidine sulfonic acids and acid halides |
| GB8712466D0 (en) * | 1987-05-27 | 1987-07-01 | Roussel Lab Ltd | Chemical compounds |
| GB8719368D0 (en) * | 1987-08-15 | 1987-09-23 | Wellcome Found | Heterocyclic compounds |
| US5302586A (en) * | 1991-12-19 | 1994-04-12 | G. D. Searle & Co. | Phosphonomethyl-imidazo[1,2-a]pyrimidine-2-carboxylic acid compounds for treatment of neurotoxic injury |
| CA2434558A1 (en) * | 2001-01-26 | 2002-08-01 | Dmitry Zuev | Imidazolyl derivatives as corticotropin releasing factor inhibitors |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3594379A (en) * | 1968-09-16 | 1971-07-20 | Sandoz Ag | 2,3-dihydroimidazo(1,2-c)quinazolines |
| US4223031A (en) * | 1978-05-05 | 1980-09-16 | Mead Johnson & Company | Azolopyrimidinones |
| US4236005A (en) * | 1979-07-02 | 1980-11-25 | American Cyanamid Company | Imidazo[1,5-a]pyrimidines |
| FR2502622A1 (fr) * | 1981-03-25 | 1982-10-01 | Synthelabo | Derives d'imidazo (1,2-a) pyrimidines, leur preparation et leur application en therapeutique |
| US4374988A (en) * | 1981-11-05 | 1983-02-22 | American Cyanamid Company | 4-Heteroarylimidazo-[1,5-A]pyrimidines |
| IL69417A (en) * | 1982-08-27 | 1987-12-20 | Roussel Uclaf | 2-acyl imidazo(1,2-a)pyrimidines,their preparation and pharmaceutical compositions containing them |
-
1983
- 1983-08-03 IL IL69417A patent/IL69417A/xx unknown
- 1983-08-23 DE DE8383401696T patent/DE3366467D1/de not_active Expired
- 1983-08-23 EP EP83401696A patent/EP0104104B1/fr not_active Expired
- 1983-08-24 PH PH29567A patent/PH20037A/en unknown
- 1983-08-24 US US06/526,046 patent/US4532243A/en not_active Expired - Fee Related
- 1983-08-25 GR GR72300A patent/GR79375B/el unknown
- 1983-08-25 AR AR294010A patent/AR241020A1/es active
- 1983-08-25 KR KR1019830003982A patent/KR890003000B1/ko not_active Expired
- 1983-08-26 ES ES525186A patent/ES8506314A1/es not_active Expired
- 1983-08-26 AU AU18461/83A patent/AU559419B2/en not_active Ceased
- 1983-08-26 IE IE2001/83A patent/IE55900B1/en not_active IP Right Cessation
- 1983-08-26 SU SU833643057A patent/SU1287752A3/ru active
- 1983-08-26 FI FI833055A patent/FI74010C/fi not_active IP Right Cessation
- 1983-08-26 NZ NZ205387A patent/NZ205387A/en unknown
- 1983-08-26 CA CA000435419A patent/CA1228589A/en not_active Expired
- 1983-08-26 GB GB08322993A patent/GB2128989B/en not_active Expired
- 1983-08-26 DD DD83254274A patent/DD215550A5/de not_active IP Right Cessation
- 1983-08-26 DK DK390583A patent/DK390583A/da not_active Application Discontinuation
- 1983-08-26 PT PT77258A patent/PT77258B/pt not_active IP Right Cessation
-
1985
- 1985-05-15 US US06/734,590 patent/US4588720A/en not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| GB2128989B (en) | 1986-03-19 |
| GB2128989A (en) | 1984-05-10 |
| DK390583D0 (da) | 1983-08-26 |
| EP0104104A1 (fr) | 1984-03-28 |
| GB8322993D0 (en) | 1983-09-28 |
| IL69417A0 (en) | 1983-11-30 |
| ES525186A0 (es) | 1985-07-01 |
| DD215550A5 (de) | 1984-11-14 |
| KR890003000B1 (ko) | 1989-08-18 |
| FI833055A0 (fi) | 1983-08-26 |
| DE3366467D1 (en) | 1986-10-30 |
| IE832001L (en) | 1984-02-27 |
| PH20037A (en) | 1986-09-04 |
| DK390583A (da) | 1984-02-28 |
| FI833055L (fi) | 1984-02-28 |
| EP0104104B1 (fr) | 1986-09-24 |
| PT77258B (en) | 1986-03-21 |
| CA1228589A (en) | 1987-10-27 |
| US4588720A (en) | 1986-05-13 |
| NZ205387A (en) | 1986-06-11 |
| US4532243A (en) | 1985-07-30 |
| SU1287752A3 (ru) | 1987-01-30 |
| FI74010B (fi) | 1987-08-31 |
| PT77258A (en) | 1983-09-01 |
| AR241020A2 (es) | 1991-04-30 |
| IL69417A (en) | 1987-12-20 |
| ES8506314A1 (es) | 1985-07-01 |
| IE55900B1 (en) | 1991-02-14 |
| AR241020A1 (es) | 1991-04-30 |
| KR840005812A (ko) | 1984-11-19 |
| AU559419B2 (en) | 1987-03-12 |
| GR79375B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | 1984-10-22 |
| AU1846183A (en) | 1984-03-01 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| MM | Patent lapsed |
Owner name: ROUSSEL-UCLAF |