FI68828C - Foerfarande foer framstaellning av nya neuroleptiska 2-(aminoalkyl)-5-fenyl-2,3,4,4a,5,9b-hexahydro-4a,9b-trans-1h-pyrido(4,3-b)indolderivat - Google Patents

Foerfarande foer framstaellning av nya neuroleptiska 2-(aminoalkyl)-5-fenyl-2,3,4,4a,5,9b-hexahydro-4a,9b-trans-1h-pyrido(4,3-b)indolderivat Download PDF

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Publication number
FI68828C
FI68828C FI802371A FI802371A FI68828C FI 68828 C FI68828 C FI 68828C FI 802371 A FI802371 A FI 802371A FI 802371 A FI802371 A FI 802371A FI 68828 C FI68828 C FI 68828C
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FI
Finland
Prior art keywords
formula
trans
pyrido
hexahydro
amino
Prior art date
Application number
FI802371A
Other languages
English (en)
Finnish (fi)
Swedish (sv)
Other versions
FI68828B (fi
FI802371A (fi
Inventor
Willard Mckowan Welch
Charles Armon Harbert
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of FI802371A publication Critical patent/FI802371A/fi
Publication of FI68828B publication Critical patent/FI68828B/fi
Application granted granted Critical
Publication of FI68828C publication Critical patent/FI68828C/fi

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Neurology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Biomedical Technology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Neurosurgery (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Psychiatry (AREA)
  • Anesthesiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Indole Compounds (AREA)
FI802371A 1979-07-30 1980-07-29 Foerfarande foer framstaellning av nya neuroleptiska 2-(aminoalkyl)-5-fenyl-2,3,4,4a,5,9b-hexahydro-4a,9b-trans-1h-pyrido(4,3-b)indolderivat FI68828C (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US06/061,573 US4252811A (en) 1979-07-30 1979-07-30 Hexahydro-trans-pyridoindole neuroleptic agents
US6157379 1979-07-30

Publications (3)

Publication Number Publication Date
FI802371A FI802371A (fi) 1981-01-31
FI68828B FI68828B (fi) 1985-07-31
FI68828C true FI68828C (fi) 1985-11-11

Family

ID=22036658

Family Applications (1)

Application Number Title Priority Date Filing Date
FI802371A FI68828C (fi) 1979-07-30 1980-07-29 Foerfarande foer framstaellning av nya neuroleptiska 2-(aminoalkyl)-5-fenyl-2,3,4,4a,5,9b-hexahydro-4a,9b-trans-1h-pyrido(4,3-b)indolderivat

Country Status (33)

Country Link
US (1) US4252811A (no)
JP (1) JPS5626891A (no)
KR (1) KR840000914B1 (no)
AR (1) AR226314A1 (no)
AT (1) AT375659B (no)
AU (1) AU513948B2 (no)
BE (1) BE884530A (no)
CA (1) CA1133483A (no)
CH (1) CH644379A5 (no)
CS (1) CS221974B2 (no)
DD (1) DD153691A5 (no)
DE (1) DE3028555A1 (no)
DK (1) DK148140C (no)
EG (1) EG14903A (no)
ES (1) ES8105732A1 (no)
FI (1) FI68828C (no)
FR (1) FR2463140A1 (no)
GB (1) GB2055372B (no)
GR (1) GR69664B (no)
IE (1) IE50035B1 (no)
IL (1) IL60695A (no)
IT (1) IT1194815B (no)
LU (1) LU82662A1 (no)
NL (1) NL180216C (no)
NO (1) NO153729C (no)
NZ (1) NZ194467A (no)
PH (1) PH22657A (no)
PL (1) PL133456B1 (no)
PT (1) PT71623B (no)
SE (1) SE438505B (no)
SU (1) SU1172450A3 (no)
YU (1) YU42223B (no)
ZA (1) ZA804604B (no)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4337250A (en) * 1979-07-30 1982-06-29 Pfizer Inc. Hexahydro-trans- and tetrahydropyridoindole neuroleptic agents
US4748247A (en) * 1986-10-21 1988-05-31 American Home Products Corporation 2-[4-[4-(2-Pyrimidinyl)-1-piperazinyl]alkyl]alkyl]pyrido- and pyrazino-indole-1,3-dione derivatives as histamine H1 antagonists
US5229517A (en) * 1990-09-27 1993-07-20 Hoechst-Roussel Pharmaceuticals Incorporated 2-(4-Piperindinyl)-1H-pyrido[4,3-B]indol-1-ones and related compounds
US5102889B1 (en) * 1990-09-27 1993-05-11 2-(4-piperidinyl)-1h-pyrido(4,3-b)indol-1-ones and related compounds
JPH05101365A (ja) * 1991-03-22 1993-04-23 Tdk Corp 垂直磁気記録媒体およびその製造方法

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3687961A (en) * 1971-05-03 1972-08-29 Abbott Lab 8-fluoro-2-{8 3-(4-fluorophenylanilinopropyl{9 -gamma-carboline
AR205452A1 (es) * 1973-12-06 1976-05-07 Endo Lab Metodo para preparar nuevos trans-2, 3, 4, 4a, 5, 9b-hexahidro-5-fenil-1h-pirido(4,3-b) indoles
JPS50126699A (no) * 1974-03-20 1975-10-04
US4001263A (en) * 1974-04-01 1977-01-04 Pfizer Inc. 5-Aryl-1,2,3,4-tetrahydro-γ-carbolines
SE7702301L (sv) * 1976-04-08 1977-10-09 Endo Lab Trans-hexahydro-pyrido-indoler

Also Published As

Publication number Publication date
SE438505B (sv) 1985-04-22
ES493818A0 (es) 1981-05-16
CS221974B2 (en) 1983-04-29
PH22657A (en) 1988-10-28
IE50035B1 (en) 1986-02-05
US4252811A (en) 1981-02-24
JPS6357433B2 (no) 1988-11-11
PL225940A1 (no) 1982-11-08
LU82662A1 (fr) 1981-03-24
SE8005453L (sv) 1981-01-31
YU191780A (en) 1983-12-31
PT71623B (en) 1982-06-09
DK148140C (da) 1985-09-16
DD153691A5 (de) 1982-01-27
IT8023785A0 (it) 1980-07-29
JPS5626891A (en) 1981-03-16
GB2055372B (en) 1983-05-05
AT375659B (de) 1984-08-27
CA1133483A (en) 1982-10-12
NO802274L (no) 1981-02-02
PT71623A (en) 1980-08-01
NO153729C (no) 1986-05-14
FI68828B (fi) 1985-07-31
ZA804604B (en) 1981-07-29
DK260080A (da) 1981-01-31
ATA393280A (de) 1984-01-15
GR69664B (no) 1982-07-07
GB2055372A (en) 1981-03-04
EG14903A (en) 1985-12-31
IL60695A (en) 1983-11-30
NL180216C (nl) 1987-01-16
FI802371A (fi) 1981-01-31
IE801576L (en) 1981-01-30
FR2463140A1 (fr) 1981-02-20
SU1172450A3 (ru) 1985-08-07
DK148140B (da) 1985-03-18
BE884530A (fr) 1981-01-29
KR840000914B1 (ko) 1984-06-28
NO153729B (no) 1986-02-03
CH644379A5 (fr) 1984-07-31
NZ194467A (en) 1984-05-31
ES8105732A1 (es) 1981-05-16
AR226314A1 (es) 1982-06-30
IT1194815B (it) 1988-09-28
AU513948B2 (en) 1981-01-15
IL60695A0 (en) 1980-09-16
FR2463140B1 (no) 1983-07-22
YU42223B (en) 1988-06-30
NL8004332A (nl) 1981-02-03
KR830003480A (ko) 1983-06-20
PL133456B1 (en) 1985-06-29
NL180216B (nl) 1986-08-18
DE3028555A1 (de) 1981-02-12

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Owner name: PFIZER INC.