FI64936C - Foerfarande foer framstaellning av nya terapeutiskt verksamma foereningar av diarylalkylamintyp - Google Patents

Foerfarande foer framstaellning av nya terapeutiskt verksamma foereningar av diarylalkylamintyp Download PDF

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Publication number
FI64936C
FI64936C FI782093A FI782093A FI64936C FI 64936 C FI64936 C FI 64936C FI 782093 A FI782093 A FI 782093A FI 782093 A FI782093 A FI 782093A FI 64936 C FI64936 C FI 64936C
Authority
FI
Finland
Prior art keywords
formula
bromophenyl
group
compound
methyl
Prior art date
Application number
FI782093A
Other languages
English (en)
Finnish (fi)
Other versions
FI64936B (fi
FI782093A7 (fi
Inventor
Bernt Sigfrid E Carnmalm
Thomas Hoegberg
Tomas De Paulis
Svante Bertil Ross
Original Assignee
Astra Laekemedel Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astra Laekemedel Ab filed Critical Astra Laekemedel Ab
Publication of FI782093A7 publication Critical patent/FI782093A7/fi
Publication of FI64936B publication Critical patent/FI64936B/fi
Application granted granted Critical
Publication of FI64936C publication Critical patent/FI64936C/fi

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/44—Iso-indoles; Hydrogenated iso-indoles
    • C07D209/48—Iso-indoles; Hydrogenated iso-indoles with oxygen atoms in positions 1 and 3, e.g. phthalimide
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/26—Psychostimulants, e.g. nicotine, cocaine
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C217/00—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton
    • C07C217/54—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having etherified hydroxy groups bound to carbon atoms of at least one six-membered aromatic ring and amino groups bound to acyclic carbon atoms or to carbon atoms of rings other than six-membered aromatic rings of the same carbon skeleton
    • C07C217/56—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having etherified hydroxy groups bound to carbon atoms of at least one six-membered aromatic ring and amino groups bound to acyclic carbon atoms or to carbon atoms of rings other than six-membered aromatic rings of the same carbon skeleton with amino groups linked to the six-membered aromatic ring, or to the condensed ring system containing that ring, by carbon chains not further substituted by singly-bound oxygen atoms
    • C07C217/62—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having etherified hydroxy groups bound to carbon atoms of at least one six-membered aromatic ring and amino groups bound to acyclic carbon atoms or to carbon atoms of rings other than six-membered aromatic rings of the same carbon skeleton with amino groups linked to the six-membered aromatic ring, or to the condensed ring system containing that ring, by carbon chains not further substituted by singly-bound oxygen atoms linked by carbon chains having at least three carbon atoms between the amino groups and the six-membered aromatic ring or the condensed ring system containing that ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/61—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups
    • C07C45/67—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton
    • C07C45/68—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton by increase in the number of carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/61—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups
    • C07C45/67—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton
    • C07C45/68—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton by increase in the number of carbon atoms
    • C07C45/72—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton by increase in the number of carbon atoms by reaction of compounds containing >C = O groups with the same or other compounds containing >C = O groups

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Psychiatry (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Biomedical Technology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Pain & Pain Management (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pyridine Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
FI782093A 1977-07-04 1978-06-29 Foerfarande foer framstaellning av nya terapeutiskt verksamma foereningar av diarylalkylamintyp FI64936C (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB27992/77A GB1602290A (en) 1977-07-04 1977-07-04 Substituted aralkyl amines and amino-aryl alkenes having therapeutic activity
GB2799277 1978-05-31

Publications (3)

Publication Number Publication Date
FI782093A7 FI782093A7 (fi) 1979-01-05
FI64936B FI64936B (fi) 1983-10-31
FI64936C true FI64936C (fi) 1984-02-10

Family

ID=10268546

Family Applications (1)

Application Number Title Priority Date Filing Date
FI782093A FI64936C (fi) 1977-07-04 1978-06-29 Foerfarande foer framstaellning av nya terapeutiskt verksamma foereningar av diarylalkylamintyp

Country Status (9)

Country Link
JP (1) JPS5439057A (da)
AT (1) AT363456B (da)
AU (1) AU519960B2 (da)
CA (1) CA1111041A (da)
DK (1) DK295178A (da)
FI (1) FI64936C (da)
GB (1) GB1602290A (da)
IT (1) IT1105075B (da)
NO (1) NO146743C (da)

Also Published As

Publication number Publication date
IT7850142A0 (it) 1978-07-03
GB1602290A (en) 1981-11-11
JPS5439057A (en) 1979-03-24
AT363456B (de) 1981-08-10
AU519960B2 (en) 1982-01-07
DK295178A (da) 1979-01-05
FI64936B (fi) 1983-10-31
CA1111041A (en) 1981-10-20
IT1105075B (it) 1985-10-28
NO146743B (no) 1982-08-23
NO782305L (no) 1979-01-05
FI782093A7 (fi) 1979-01-05
ATA483578A (de) 1981-01-15
NO146743C (no) 1982-12-01
AU3761278A (en) 1980-01-03

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Date Code Title Description
MM Patent lapsed

Owner name: ASTRA LAEKEMEDEL AKTIEBOLAG