FI63757C - Foerfarande foer framstaellning av nya terapeutiskt anvaendbara kinoxalin- och kinazolinderivat - Google Patents

Foerfarande foer framstaellning av nya terapeutiskt anvaendbara kinoxalin- och kinazolinderivat Download PDF

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Publication number
FI63757C
FI63757C FI436/73A FI43673A FI63757C FI 63757 C FI63757 C FI 63757C FI 436/73 A FI436/73 A FI 436/73A FI 43673 A FI43673 A FI 43673A FI 63757 C FI63757 C FI 63757C
Authority
FI
Finland
Prior art keywords
quinoxaline
formula
compound
quinazoline
och
Prior art date
Application number
FI436/73A
Other languages
English (en)
Finnish (fi)
Other versions
FI63757B (fi
Inventor
John Christopher Danilewicz
Michael Snarey
Geoffrey Noel Thomas
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Application granted granted Critical
Publication of FI63757B publication Critical patent/FI63757B/fi
Publication of FI63757C publication Critical patent/FI63757C/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D215/00Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/18Halogen atoms or nitro radicals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D215/00Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/38Nitrogen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D215/00Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/38Nitrogen atoms
    • C07D215/40Nitrogen atoms attached in position 8
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D241/00Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
    • C07D241/36Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings condensed with carbocyclic rings or ring systems
    • C07D241/38Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings condensed with carbocyclic rings or ring systems with only hydrogen or carbon atoms directly attached to the ring nitrogen atoms
    • C07D241/40Benzopyrazines
    • C07D241/42Benzopyrazines with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
FI436/73A 1972-02-29 1973-02-14 Foerfarande foer framstaellning av nya terapeutiskt anvaendbara kinoxalin- och kinazolinderivat FI63757C (fi)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
GB919672A GB1381979A (en) 1972-02-29 1972-02-29 Amino derivatives of quinoline quinoxaline and quinazoline
GB919672 1972-02-29
GB5162972 1972-11-08
GB5162972 1972-11-08

Publications (2)

Publication Number Publication Date
FI63757B FI63757B (fi) 1983-04-29
FI63757C true FI63757C (fi) 1983-08-10

Family

ID=26242776

Family Applications (1)

Application Number Title Priority Date Filing Date
FI436/73A FI63757C (fi) 1972-02-29 1973-02-14 Foerfarande foer framstaellning av nya terapeutiskt anvaendbara kinoxalin- och kinazolinderivat

Country Status (16)

Country Link
US (1) US3890319A (show.php)
JP (2) JPS5754516B2 (show.php)
AR (1) AR213705A1 (show.php)
AU (1) AU471598B2 (show.php)
BE (1) BE795970A (show.php)
CA (1) CA981678A (show.php)
CH (2) CH576975A5 (show.php)
DE (1) DE2309160A1 (show.php)
ES (2) ES411804A1 (show.php)
FI (1) FI63757C (show.php)
FR (1) FR2181776B1 (show.php)
GB (1) GB1381979A (show.php)
IE (1) IE37519B1 (show.php)
MX (1) MX3042E (show.php)
NL (1) NL159102B (show.php)
SE (1) SE417204B (show.php)

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* Cited by examiner, † Cited by third party
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JPS6118950U (ja) * 1984-07-10 1986-02-03 財団法人鉄道総合技術研究所 トロリ線の給油装置
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Also Published As

Publication number Publication date
JPS5745439B2 (show.php) 1982-09-28
AU471598B2 (en) 1976-04-29
CH577500A5 (show.php) 1976-07-15
FR2181776B1 (show.php) 1976-08-13
ES411804A1 (es) 1976-05-01
DE2309160A1 (de) 1973-09-27
NL159102B (nl) 1979-01-15
MX3042E (es) 1980-03-04
CA981678A (en) 1976-01-13
FR2181776A1 (show.php) 1973-12-07
FI63757B (fi) 1983-04-29
BE795970A (fr) 1973-08-27
US3890319A (en) 1975-06-17
GB1381979A (en) 1975-01-29
JPS4897878A (show.php) 1973-12-13
IE37519L (en) 1973-08-29
CH576975A5 (show.php) 1976-06-30
AU5198573A (en) 1974-08-08
ES412102A1 (es) 1976-05-16
NL7302799A (show.php) 1973-08-31
IE37519B1 (en) 1977-08-17
JPS5625176A (en) 1981-03-10
SE417204B (sv) 1981-03-02
JPS5754516B2 (show.php) 1982-11-18
AR213705A1 (es) 1979-03-15

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