FI60200C - Foerfarande foer framstaellning av farmakologiskt vaerdefulla n-arylalkylpiperidylsubstituerade bensamider - Google Patents
Foerfarande foer framstaellning av farmakologiskt vaerdefulla n-arylalkylpiperidylsubstituerade bensamider Download PDFInfo
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- FI60200C FI60200C FI750825A FI750825A FI60200C FI 60200 C FI60200 C FI 60200C FI 750825 A FI750825 A FI 750825A FI 750825 A FI750825 A FI 750825A FI 60200 C FI60200 C FI 60200C
- Authority
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- Finland
- Prior art keywords
- amino
- methoxy
- compounds
- acid
- piperidyl
- Prior art date
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- C—CHEMISTRY; METALLURGY
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- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D211/56—Nitrogen atoms
- C07D211/58—Nitrogen atoms attached in position 4
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
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- A—HUMAN NECESSITIES
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-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/08—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
- C07D211/18—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D211/26—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by nitrogen atoms
- C07D211/28—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by nitrogen atoms to which a second hetero atom is attached
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/68—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
- C07D211/72—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, directly attached to ring carbon atoms
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Medicinal Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Public Health (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Neurosurgery (AREA)
- Pain & Pain Management (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Otolaryngology (AREA)
- Anesthesiology (AREA)
- Hospice & Palliative Care (AREA)
- Rheumatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Hydrogenated Pyridines (AREA)
- Plural Heterocyclic Compounds (AREA)
- Other In-Based Heterocyclic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Pyridine Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB12572/74A GB1507462A (en) | 1974-03-21 | 1974-03-21 | N-heterocyclic substituted benzamides methods for their preparation and compositions containing them |
| GB1257274 | 1974-03-21 | ||
| GB3540274 | 1974-08-12 | ||
| GB3540274 | 1974-08-12 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| FI750825A7 FI750825A7 (pm) | 1975-09-22 |
| FI60200B FI60200B (fi) | 1981-08-31 |
| FI60200C true FI60200C (fi) | 1981-12-10 |
Family
ID=26249107
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| FI750825A FI60200C (fi) | 1974-03-21 | 1975-03-20 | Foerfarande foer framstaellning av farmakologiskt vaerdefulla n-arylalkylpiperidylsubstituerade bensamider |
Country Status (11)
| Country | Link |
|---|---|
| JP (1) | JPS584019B2 (pm) |
| AR (1) | AR216043A1 (pm) |
| CH (1) | CH602641A5 (pm) |
| DK (1) | DK147854C (pm) |
| ES (5) | ES435756A1 (pm) |
| FI (1) | FI60200C (pm) |
| FR (1) | FR2264530A1 (pm) |
| KE (1) | KE2900A (pm) |
| NL (1) | NL159660B (pm) |
| NO (1) | NO144108C (pm) |
| SE (1) | SE427750B (pm) |
Families Citing this family (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB1513631A (en) * | 1976-02-17 | 1978-06-07 | Gallardo Antonio Sa | Piperidine derivatives |
| GB1561023A (en) * | 1977-04-22 | 1980-02-13 | Beecham Group Ltd | 2-methoxy - 5 - chloro aniline derivatives |
| FR2446274A1 (fr) * | 1979-01-15 | 1980-08-08 | Delalande Sa | Nouveaux derives de salicylamide, leur procede de preparation et leur application en therapeutique |
| EP0343307A1 (en) * | 1988-05-26 | 1989-11-29 | Fabrica Espanola De Productos Quimicos Y Farmaceuticos, S.A. | 4-Piperidinealkanamine derivatives |
| FR2674849B1 (fr) * | 1991-04-02 | 1994-12-23 | Logeais Labor Jacques | Nouveaux derives de n-cyclohexyl benzamides ou thiobenzamides, leurs preparations et leurs applications en therapeutique. |
| FR2766484B1 (fr) * | 1997-07-25 | 1999-09-17 | Logeais Labor Jacques | Nouveaux derives benzamides stimulants de la motricite gastrointestinale haute et basse |
| FR2766486B1 (fr) * | 1997-07-25 | 1999-09-17 | Logeais Labor Jacques | Cycloalkyles benzamides stimulants de la motricite gastrointestinale haute et basse |
| WO2006128803A1 (en) * | 2005-06-02 | 2006-12-07 | F. Hoffmann-La Roche Ag | Piperidin-4-yl-amide derivatives and their use as sst receptor subtype 5 antagonists |
| KR100976063B1 (ko) * | 2007-03-16 | 2010-08-17 | 동아제약주식회사 | 신규한 벤즈아미드 유도체 화합물 및 그의 제조방법 |
| CN103958477B (zh) * | 2011-11-29 | 2017-03-29 | (株)威沃尊 | 苯甲酰胺衍生物及其用途 |
-
1975
- 1975-03-17 AR AR257994A patent/AR216043A1/es active
- 1975-03-18 ES ES435756A patent/ES435756A1/es not_active Expired
- 1975-03-18 ES ES435757A patent/ES435757A1/es not_active Expired
- 1975-03-18 ES ES435755A patent/ES435755A1/es not_active Expired
- 1975-03-18 ES ES435754A patent/ES435754A1/es not_active Expired
- 1975-03-18 ES ES435753A patent/ES435753A1/es not_active Expired
- 1975-03-20 CH CH355075A patent/CH602641A5/xx not_active IP Right Cessation
- 1975-03-20 NO NO750957A patent/NO144108C/no unknown
- 1975-03-20 SE SE7503196A patent/SE427750B/xx not_active IP Right Cessation
- 1975-03-20 FR FR7509371A patent/FR2264530A1/fr active Granted
- 1975-03-20 FI FI750825A patent/FI60200C/fi not_active IP Right Cessation
- 1975-03-20 DK DK117675A patent/DK147854C/da not_active IP Right Cessation
- 1975-03-21 NL NL7503417.A patent/NL159660B/xx not_active IP Right Cessation
- 1975-03-22 JP JP7534871A patent/JPS584019B2/ja not_active Expired
-
1978
- 1978-11-14 KE KE2900A patent/KE2900A/xx unknown
Also Published As
| Publication number | Publication date |
|---|---|
| FI60200B (fi) | 1981-08-31 |
| ES435755A1 (es) | 1977-04-01 |
| DK117675A (pm) | 1975-09-22 |
| ES435753A1 (es) | 1977-04-01 |
| JPS584019B2 (ja) | 1983-01-24 |
| KE2900A (en) | 1978-12-01 |
| CH602641A5 (pm) | 1978-07-31 |
| SE427750B (sv) | 1983-05-02 |
| NL159660B (nl) | 1979-03-15 |
| ES435757A1 (es) | 1977-04-01 |
| SE7503196L (pm) | 1975-09-22 |
| NO144108B (no) | 1981-03-16 |
| FI750825A7 (pm) | 1975-09-22 |
| NO750957L (pm) | 1975-09-23 |
| ES435754A1 (es) | 1977-04-01 |
| AR216043A1 (es) | 1979-11-30 |
| DK147854C (da) | 1985-07-22 |
| NL7503417A (nl) | 1975-09-23 |
| NO144108C (no) | 1981-06-24 |
| ES435756A1 (es) | 1977-04-01 |
| DK147854B (da) | 1984-12-24 |
| FR2264530A1 (en) | 1975-10-17 |
| JPS50129573A (pm) | 1975-10-13 |
| FR2264530B1 (pm) | 1978-11-10 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| MA | Patent expired | ||
| MA | Patent expired |
Owner name: FORDONAL S.A. |