FI59102C - Foerfarande foer framstaellning av nya terapeutiskt effektiva piperazinyliminorifamycinfoereningar - Google Patents
Foerfarande foer framstaellning av nya terapeutiskt effektiva piperazinyliminorifamycinfoereningar Download PDFInfo
- Publication number
- FI59102C FI59102C FI760561A FI760561A FI59102C FI 59102 C FI59102 C FI 59102C FI 760561 A FI760561 A FI 760561A FI 760561 A FI760561 A FI 760561A FI 59102 C FI59102 C FI 59102C
- Authority
- FI
- Finland
- Prior art keywords
- cyclopentyl
- rifampicin
- derivative
- effective
- compound
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D498/08—Bridged systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Communicable Diseases (AREA)
- Pharmacology & Pharmacy (AREA)
- Oncology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB1002075 | 1975-03-05 | ||
GB10020/75A GB1478563A (en) | 1975-03-05 | 1975-03-05 | Rifamycin derivatives |
Publications (3)
Publication Number | Publication Date |
---|---|
FI760561A FI760561A (nl) | 1976-09-06 |
FI59102B FI59102B (fi) | 1981-02-27 |
FI59102C true FI59102C (fi) | 1981-06-10 |
Family
ID=9959968
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
FI760561A FI59102C (fi) | 1975-03-05 | 1976-03-05 | Foerfarande foer framstaellning av nya terapeutiskt effektiva piperazinyliminorifamycinfoereningar |
Country Status (27)
Country | Link |
---|---|
US (1) | US4002752A (nl) |
JP (1) | JPS51113900A (nl) |
AR (1) | AR210113A1 (nl) |
AT (1) | AT344896B (nl) |
BE (1) | BE839255A (nl) |
CA (1) | CA1057748A (nl) |
CH (1) | CH610325A5 (nl) |
DD (1) | DD123888A5 (nl) |
DE (1) | DE2608218C3 (nl) |
DK (1) | DK136655B (nl) |
ES (1) | ES445790A1 (nl) |
FI (1) | FI59102C (nl) |
FR (1) | FR2302742A1 (nl) |
GB (1) | GB1478563A (nl) |
HK (1) | HK35282A (nl) |
HU (1) | HU170451B (nl) |
IE (1) | IE42881B1 (nl) |
KE (1) | KE3099A (nl) |
LU (1) | LU74478A1 (nl) |
MX (1) | MX3737E (nl) |
NL (1) | NL165745C (nl) |
NO (1) | NO143796C (nl) |
PT (1) | PT64866B (nl) |
SE (1) | SE420728B (nl) |
SU (1) | SU575030A3 (nl) |
YU (1) | YU39477B (nl) |
ZA (1) | ZA761043B (nl) |
Families Citing this family (18)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE2728869A1 (de) * | 1976-06-25 | 1977-12-29 | Antibiotice Iasi Intreprindere | Rifamycinen und verfahren zu deren herstellung |
GR64108B (en) * | 1977-04-15 | 1980-01-24 | Dso Pharmachim | Method for the preparation of azomethine-derivatives of rifamycin s.v |
GB1576886A (en) * | 1977-04-20 | 1980-10-15 | Lepetit Spa | Rifamycin derivatives |
GB1594134A (en) * | 1977-11-25 | 1981-07-30 | Holco Investment Inc | Rifamycins |
AU536524B2 (en) * | 1979-06-28 | 1984-05-10 | Gruppo Lepetit S.P.A. | Water soluble hydrozones of 3-formylifamyan |
US4447432A (en) * | 1981-11-17 | 1984-05-08 | Farmitalia Carlo Erba S.P.A. | Azino rifamycins |
US4681938A (en) * | 1984-08-27 | 1987-07-21 | Ciba-Geigy Corporation | Novel polycyclic hydrazones of rifamycins, their manufacture, and their pharmaceutical compositions for treating tuberculosis |
ATE47857T1 (de) * | 1985-10-18 | 1989-11-15 | Ciba Geigy Ag | Substituierte 4-benzyl-piperazinyl-verbindungen. |
US4916126A (en) * | 1987-09-25 | 1990-04-10 | Ciba-Geigy Corporation | Diacyl derivatives of 4-(trialkylbenzyl)-piperazinyl compounds |
GB8816620D0 (en) * | 1988-07-13 | 1988-08-17 | Lepetit Spa | Rifapentine hydrohalides |
JP3350861B2 (ja) * | 1990-06-29 | 2002-11-25 | アベンテイス・バルク・ソチエタ・ペル・アチオニ | リファペンチンの純粋の結晶型 |
AU2006339058B2 (en) | 2005-08-11 | 2012-09-06 | Targanta Therapeutics Inc. | Phosphonated rifamycins and uses thereof for the prevention and treatment of bone and joint infections |
WO2010019511A2 (en) | 2008-08-13 | 2010-02-18 | Targanta Therapeutics Corp. | Phosphonated rifamycins and uses thereof for the prevention and treatment of bone and joint infections |
RU2496475C2 (ru) | 2011-10-26 | 2013-10-27 | Александр Васильевич Иващенко | Фармацевтическая композиция и набор для лечения бактериальных инфекций |
PT2882435T (pt) | 2012-08-13 | 2021-06-18 | Kiril Asenov Ninov | Formulações farmacêuticas contendo 3-(4-cinamil-lpiperazinil)amino derivados da 3-formilrifamicina s |
CN103951677B (zh) * | 2014-03-17 | 2016-04-06 | 四川省长征药业股份有限公司 | 利福喷丁的制备方法 |
WO2022225384A1 (es) * | 2021-04-21 | 2022-10-27 | Interquim, S.A. De C.V. | Proceso de obtención de rifapentina. con una nueva forma cristalina |
CN115047122B (zh) * | 2022-06-29 | 2023-05-02 | 重庆华邦胜凯制药有限公司 | 利福喷丁及其合成过程中所产生的杂质的分析方法 |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR208F (nl) * | 1964-07-31 | |||
AR205434A1 (es) * | 1972-03-27 | 1976-05-07 | Lepetit Spa | Proceso para la preparacion de 3-acilhidrazonometil rifamicinas sv |
GB1392272A (en) * | 1972-05-31 | 1975-04-30 | Lepetit Spa | 3-formylrifamycin azines |
-
1975
- 1975-03-05 GB GB10020/75A patent/GB1478563A/en not_active Expired
-
1976
- 1976-02-19 NO NO760549A patent/NO143796C/no unknown
- 1976-02-23 ZA ZA1043A patent/ZA761043B/xx unknown
- 1976-02-23 SE SE7602122A patent/SE420728B/xx not_active IP Right Cessation
- 1976-02-25 DK DK78476AA patent/DK136655B/da not_active IP Right Cessation
- 1976-02-26 US US05/661,587 patent/US4002752A/en not_active Expired - Lifetime
- 1976-02-28 DE DE2608218A patent/DE2608218C3/de not_active Expired
- 1976-03-03 NL NL7602191.A patent/NL165745C/nl not_active IP Right Cessation
- 1976-03-03 AR AR262431A patent/AR210113A1/es active
- 1976-03-03 SU SU7602329559A patent/SU575030A3/ru active
- 1976-03-04 CA CA247,156A patent/CA1057748A/en not_active Expired
- 1976-03-04 LU LU74478A patent/LU74478A1/xx unknown
- 1976-03-04 IE IE448/76A patent/IE42881B1/en not_active IP Right Cessation
- 1976-03-04 HU HULE790A patent/HU170451B/hu unknown
- 1976-03-04 CH CH271376A patent/CH610325A5/xx not_active IP Right Cessation
- 1976-03-04 MX MX7636U patent/MX3737E/es unknown
- 1976-03-04 JP JP51023701A patent/JPS51113900A/ja active Granted
- 1976-03-04 PT PT64866A patent/PT64866B/pt unknown
- 1976-03-05 DD DD191727A patent/DD123888A5/xx unknown
- 1976-03-05 AT AT162876A patent/AT344896B/de not_active IP Right Cessation
- 1976-03-05 BE BE164907A patent/BE839255A/xx not_active IP Right Cessation
- 1976-03-05 FI FI760561A patent/FI59102C/fi not_active IP Right Cessation
- 1976-03-05 ES ES445790A patent/ES445790A1/es not_active Expired
- 1976-03-05 YU YU572/76A patent/YU39477B/xx unknown
- 1976-03-05 FR FR7606379A patent/FR2302742A1/fr active Granted
-
1980
- 1980-11-01 KE KE3099A patent/KE3099A/xx unknown
-
1982
- 1982-08-03 HK HK352/82A patent/HK35282A/xx unknown
Also Published As
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
MA | Patent expired | ||
MA | Patent expired |
Owner name: GRUPPO LEPETIT S.P.A |