FI56840C - Foerfarande foer framstaellning av saosom antibakteriska aemnen anvaendbara 6-(2-fenyl-2-(amidino- och imidoylamino-alkanoylamino)acetamido)penicillansyror - Google Patents

Foerfarande foer framstaellning av saosom antibakteriska aemnen anvaendbara 6-(2-fenyl-2-(amidino- och imidoylamino-alkanoylamino)acetamido)penicillansyror Download PDF

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Publication number
FI56840C
FI56840C FI2405/73A FI240573A FI56840C FI 56840 C FI56840 C FI 56840C FI 2405/73 A FI2405/73 A FI 2405/73A FI 240573 A FI240573 A FI 240573A FI 56840 C FI56840 C FI 56840C
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FI
Finland
Prior art keywords
phenyl
acetamido
amidino
imidoylamino
triethylamine
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Application number
FI2405/73A
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English (en)
Finnish (fi)
Other versions
FI56840B (fi
Inventor
Ernest Seiichi Hamanaka
John Gerritt Stam
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Pfizer
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Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
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Publication of FI56840B publication Critical patent/FI56840B/fi
Publication of FI56840C publication Critical patent/FI56840C/fi

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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D207/00Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/30Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
    • C07D207/32Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • C07D207/33Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms with substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • C07D207/335Radicals substituted by nitrogen atoms not forming part of a nitro radical
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D207/00Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/30Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
    • C07D207/34Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D213/00Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/72Nitrogen atoms
    • C07D213/74Amino or imino radicals substituted by hydrocarbon or substituted hydrocarbon radicals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D307/00Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/02Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
    • C07D307/34Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D307/38Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D307/52Radicals substituted by nitrogen atoms not forming part of a nitro radical
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D307/00Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/02Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
    • C07D307/34Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D307/56Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D307/66Nitrogen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D333/00Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/26Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D333/30Hetero atoms other than halogen
    • C07D333/36Nitrogen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D333/00Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/26Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D333/38Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D499/00Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
FI2405/73A 1972-08-02 1973-07-31 Foerfarande foer framstaellning av saosom antibakteriska aemnen anvaendbara 6-(2-fenyl-2-(amidino- och imidoylamino-alkanoylamino)acetamido)penicillansyror FI56840C (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US27706472A 1972-08-02 1972-08-02
US27706472 1972-08-02

Publications (2)

Publication Number Publication Date
FI56840B FI56840B (fi) 1979-12-31
FI56840C true FI56840C (fi) 1980-04-10

Family

ID=23059254

Family Applications (1)

Application Number Title Priority Date Filing Date
FI2405/73A FI56840C (fi) 1972-08-02 1973-07-31 Foerfarande foer framstaellning av saosom antibakteriska aemnen anvaendbara 6-(2-fenyl-2-(amidino- och imidoylamino-alkanoylamino)acetamido)penicillansyror

Country Status (30)

Country Link
JP (1) JPS5318039B2 (ru)
AR (1) AR206879A1 (ru)
AT (1) AT327382B (ru)
AU (1) AU472676B2 (ru)
BE (1) BE803094A (ru)
BG (1) BG25798A3 (ru)
CA (1) CA1015355A (ru)
CH (1) CH574447A5 (ru)
CS (1) CS168459B2 (ru)
DD (1) DD106849A5 (ru)
DE (1) DE2338389A1 (ru)
DK (1) DK137047B (ru)
EG (1) EG10896A (ru)
ES (1) ES417461A1 (ru)
FI (1) FI56840C (ru)
FR (1) FR2194415B1 (ru)
GB (1) GB1418656A (ru)
HU (1) HU167653B (ru)
IE (1) IE37961B1 (ru)
IL (1) IL42820A (ru)
LU (1) LU68143A1 (ru)
NL (1) NL7310696A (ru)
NO (1) NO144831C (ru)
PH (1) PH12770A (ru)
PL (1) PL96500B1 (ru)
RO (2) RO63748A (ru)
SE (1) SE415977B (ru)
SU (2) SU576944A3 (ru)
YU (1) YU36966B (ru)
ZA (1) ZA735236B (ru)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4024130A (en) * 1975-03-31 1977-05-17 Pfizer Inc. Process for the manufacture of alkali metal salts of 6-[2-phenyl-2-(imidoylaminoalkanoylamino)acetamido]penicillanic acids
US4073780A (en) * 1976-06-03 1978-02-14 Pfizer Inc. 4-Pyridylformimidoylglycyl-D-phenylglycine

Also Published As

Publication number Publication date
CH574447A5 (ru) 1976-04-15
IE37961L (en) 1974-02-02
GB1418656A (en) 1975-12-24
FR2194415B1 (ru) 1976-12-31
SU576944A3 (ru) 1977-10-15
FR2194415A1 (ru) 1974-03-01
EG10896A (en) 1976-07-31
HU167653B (ru) 1975-11-28
PH12770A (en) 1979-08-17
BG25798A3 (en) 1978-12-12
SE415977B (sv) 1980-11-17
CA1015355A (en) 1977-08-09
AT327382B (de) 1976-01-26
AU472676B2 (en) 1976-06-03
LU68143A1 (ru) 1974-02-11
SU576945A3 (ru) 1977-10-15
DK137047C (ru) 1978-08-07
ATA680773A (de) 1975-04-15
NL7310696A (ru) 1974-02-05
CS168459B2 (ru) 1976-06-29
YU36966B (en) 1984-08-31
FI56840B (fi) 1979-12-31
JPS4945089A (ru) 1974-04-27
NO144831B (no) 1981-08-10
AR206879A1 (es) 1976-08-31
YU208673A (en) 1982-02-25
RO63748A (fr) 1979-01-15
DD106849A5 (ru) 1974-07-05
ZA735236B (en) 1974-07-31
JPS5318039B2 (ru) 1978-06-13
IL42820A (en) 1977-06-30
ES417461A1 (es) 1976-03-01
NO144831C (no) 1981-11-18
IL42820A0 (en) 1973-10-25
PL96500B1 (pl) 1977-12-31
BE803094A (fr) 1974-02-01
IE37961B1 (en) 1977-11-23
AU5843373A (en) 1975-01-30
RO68719A2 (ro) 1980-08-15
DK137047B (da) 1978-01-09
DE2338389A1 (de) 1974-02-28

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