FI111715B - Menetelmä terapeuttisesti käyttökelpoisten sykloalkyyli-substituoitujen glutaramidiyhdisteiden valmistamiseksi - Google Patents

Menetelmä terapeuttisesti käyttökelpoisten sykloalkyyli-substituoitujen glutaramidiyhdisteiden valmistamiseksi Download PDF

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FI111715B
FI111715B FI894158A FI894158A FI111715B FI 111715 B FI111715 B FI 111715B FI 894158 A FI894158 A FI 894158A FI 894158 A FI894158 A FI 894158A FI 111715 B FI111715 B FI 111715B
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alkyl
formula
aryl
group
heterocyclyl
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FI894158A
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Finnish (fi)
Swedish (sv)
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FI894158A (fi
FI894158A0 (fi
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Keith James
John Christopher Danilewicz
Ryszard Jurek Kobylecki
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Pfizer
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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/02—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
    • C07D307/34—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D307/56—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D307/68—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
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    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
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    • A61P27/00—Drugs for disorders of the senses
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    • C07C235/82—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups and doubly-bound oxygen atoms bound to the same carbon skeleton with the carbon atom of at least one of the carboxamide groups bound to a carbon atom of a ring other than a six-membered aromatic ring
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    • C07C271/22—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms to carbon atoms of hydrocarbon radicals substituted by carboxyl groups
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    • C07C311/06—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton having the nitrogen atoms of the sulfonamide groups bound to hydrogen atoms or to acyclic carbon atoms to acyclic carbon atoms of hydrocarbon radicals substituted by carboxyl groups
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    • C07C311/02—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton
    • C07C311/08—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton having the nitrogen atom of at least one of the sulfonamide groups bound to a carbon atom of a six-membered aromatic ring
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    • C07C311/15—Sulfonamides having sulfur atoms of sulfonamide groups bound to carbon atoms of six-membered aromatic rings
    • C07C311/16—Sulfonamides having sulfur atoms of sulfonamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the sulfonamide groups bound to hydrogen atoms or to an acyclic carbon atom
    • C07C311/19—Sulfonamides having sulfur atoms of sulfonamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the sulfonamide groups bound to hydrogen atoms or to an acyclic carbon atom to an acyclic carbon atom of a hydrocarbon radical substituted by carboxyl groups
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    • C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/08—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon radicals, substituted by hetero atoms, attached to ring carbon atoms
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    • C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/10—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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    • C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
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    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
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    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
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    • C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
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    • C07D233/64—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms, e.g. histidine
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    • C07D317/10—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 not condensed with other rings
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  • Bioinformatics & Cheminformatics (AREA)
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  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Ophthalmology & Optometry (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Obesity (AREA)
  • Endocrinology (AREA)
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  • Urology & Nephrology (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Hydrogenated Pyridines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Furan Compounds (AREA)
  • Pyridine Compounds (AREA)
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FI894158A 1988-09-05 1989-09-04 Menetelmä terapeuttisesti käyttökelpoisten sykloalkyyli-substituoitujen glutaramidiyhdisteiden valmistamiseksi FI111715B (fi)

Priority Applications (1)

Application Number Priority Date Filing Date Title
FI982485A FI982485A0 (fi) 1988-09-05 1998-11-17 Terapeuttisesti käyttökelpoiset sykloalkyyli-substituoidut glutaramidiyhdisteet

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Application Number Priority Date Filing Date Title
GB8820844 1988-09-05
GB888820844A GB8820844D0 (en) 1988-09-05 1988-09-05 Therapeutic agents

Publications (3)

Publication Number Publication Date
FI894158A0 FI894158A0 (fi) 1989-09-04
FI894158A FI894158A (fi) 1990-03-06
FI111715B true FI111715B (fi) 2003-09-15

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FI894158A FI111715B (fi) 1988-09-05 1989-09-04 Menetelmä terapeuttisesti käyttökelpoisten sykloalkyyli-substituoitujen glutaramidiyhdisteiden valmistamiseksi

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US (1) US4975444A (hu)
EP (1) EP0358398B1 (hu)
JP (1) JPH0660144B2 (hu)
CN (1) CN1031051C (hu)
AT (1) ATE86606T1 (hu)
AU (1) AU604195B2 (hu)
CA (1) CA1341046C (hu)
CY (1) CY1811A (hu)
CZ (1) CZ282142B6 (hu)
DD (1) DD284222A5 (hu)
DE (1) DE68905272T2 (hu)
DK (1) DK175082B1 (hu)
EG (1) EG18936A (hu)
ES (1) ES2054009T3 (hu)
FI (1) FI111715B (hu)
GB (1) GB8820844D0 (hu)
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NO893546L (no) 1990-03-06
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MX17418A (es) 1993-11-01
EG18936A (en) 1994-11-30
FI894158A (fi) 1990-03-06
RU2012556C1 (ru) 1994-05-15
HUT51293A (en) 1990-04-28
IL91460A (en) 1995-08-31
IL91460A0 (en) 1990-04-29
NO177747C (no) 1995-11-15
HU211536A9 (en) 1995-12-28
PH26272A (en) 1992-04-01
ES2054009T3 (es) 1994-08-01
PT91623A (pt) 1990-03-30
YU168489A (en) 1991-06-30
DK436289D0 (da) 1989-09-04
HK130394A (en) 1994-12-02
AU604195B2 (en) 1990-12-06
DK175082B1 (da) 2004-05-24
CN1040986A (zh) 1990-04-04
EP0358398A1 (en) 1990-03-14
EP0358398B1 (en) 1993-03-10
FI894158A0 (fi) 1989-09-04
IE62020B1 (en) 1994-12-14
DD284222A5 (de) 1990-11-07
DE68905272T2 (de) 1993-06-17
NO893546D0 (no) 1989-09-04
IE892833L (en) 1990-03-05
GB8820844D0 (en) 1988-10-05
PL161527B1 (en) 1993-07-30
CA1341046C (en) 2000-07-04
HU215440B (hu) 2000-04-28
DK436289A (da) 1990-03-06
CN1031051C (zh) 1996-02-21
CZ510889A3 (en) 1997-02-12
PT91623B (pt) 1995-05-31
AU4105289A (en) 1990-03-08
ZA896760B (en) 1991-04-24
NZ230550A (en) 1991-02-26
MY106606A (en) 1995-06-30
JPH02124862A (ja) 1990-05-14
ATE86606T1 (de) 1993-03-15
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NO177747B (no) 1995-08-07
RU2108322C1 (ru) 1998-04-10

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