FI107537B - Makrolidien 2-aminosokerijohdannaiset - Google Patents

Makrolidien 2-aminosokerijohdannaiset Download PDF

Info

Publication number
FI107537B
FI107537B FI944015A FI944015A FI107537B FI 107537 B FI107537 B FI 107537B FI 944015 A FI944015 A FI 944015A FI 944015 A FI944015 A FI 944015A FI 107537 B FI107537 B FI 107537B
Authority
FI
Finland
Prior art keywords
formula
independently
compound
occurrence
alkyl
Prior art date
Application number
FI944015A
Other languages
English (en)
Finnish (fi)
Swedish (sv)
Other versions
FI944015A (fi
FI944015A0 (fi
Inventor
Gary R Schulte
Kevin Koch
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of FI944015A publication Critical patent/FI944015A/fi
Publication of FI944015A0 publication Critical patent/FI944015A0/fi
Application granted granted Critical
Publication of FI107537B publication Critical patent/FI107537B/fi

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/01—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing oxygen
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/06—Immunosuppressants, e.g. drugs for graft rejection

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Immunology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Transplantation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
FI944015A 1992-03-02 1994-09-01 Makrolidien 2-aminosokerijohdannaiset FI107537B (fi)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US84433992A 1992-03-02 1992-03-02
US84433992 1992-03-02
US9300427 1993-01-27
PCT/US1993/000427 WO1993018048A1 (en) 1992-03-02 1993-01-27 2-aminosugar derivatives of macrolides

Publications (3)

Publication Number Publication Date
FI944015A FI944015A (fi) 1994-09-01
FI944015A0 FI944015A0 (fi) 1994-09-01
FI107537B true FI107537B (fi) 2001-08-31

Family

ID=25292446

Family Applications (1)

Application Number Title Priority Date Filing Date
FI944015A FI107537B (fi) 1992-03-02 1994-09-01 Makrolidien 2-aminosokerijohdannaiset

Country Status (11)

Country Link
US (1) US5631235A (es)
EP (1) EP0636136B1 (es)
JP (1) JP2562001B2 (es)
AT (1) ATE159725T1 (es)
CA (1) CA2131373C (es)
DE (1) DE69314947T2 (es)
DK (1) DK0636136T3 (es)
ES (1) ES2108261T3 (es)
FI (1) FI107537B (es)
GR (1) GR3025672T3 (es)
WO (1) WO1993018048A1 (es)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AUPP584198A0 (en) 1998-09-14 1998-10-08 Fujisawa Pharmaceutical Co., Ltd. New use
US7160867B2 (en) 2003-05-16 2007-01-09 Isotechnika, Inc. Rapamycin carbohydrate derivatives
CA2571710A1 (en) 2004-06-24 2006-11-02 Nicholas Valiante Small molecule immunopotentiators and assays for their detection

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4894366A (en) * 1984-12-03 1990-01-16 Fujisawa Pharmaceutical Company, Ltd. Tricyclo compounds, a process for their production and a pharmaceutical composition containing the same
AU6286690A (en) * 1989-08-18 1991-04-03 Fisons Plc Macrocyclic compounds
DK0427680T3 (da) * 1989-11-09 1995-12-18 Sandoz Ltd Heteroatom-holdige cykliske forbindelser
IE904050A1 (en) * 1989-11-13 1991-05-22 Merck & Co Inc Aminomacrolides and derivatives having immunosuppressive¹activity
EP0466365A3 (en) * 1990-07-03 1992-04-15 Merck & Co. Inc. Novel immunosuppressant fermentation products of a microorganism

Also Published As

Publication number Publication date
CA2131373C (en) 1999-01-26
WO1993018048A1 (en) 1993-09-16
DE69314947T2 (de) 1998-03-05
FI944015A (fi) 1994-09-01
EP0636136B1 (en) 1997-10-29
JP2562001B2 (ja) 1996-12-11
EP0636136A1 (en) 1995-02-01
US5631235A (en) 1997-05-20
DK0636136T3 (da) 1997-12-22
FI944015A0 (fi) 1994-09-01
DE69314947D1 (de) 1997-12-04
GR3025672T3 (en) 1998-03-31
CA2131373A1 (en) 1993-09-16
JPH07500350A (ja) 1995-01-12
ATE159725T1 (de) 1997-11-15
ES2108261T3 (es) 1997-12-16

Similar Documents

Publication Publication Date Title
IE69974B1 (en) Heteroatoms-containing tricyclic compounds
EP0629203B1 (en) Desosamino derivatives of macrolides as immunosuppressants and antifungal agents
PL172789B1 (pl) Sposób wytwarzania nowych makrolidów imidazolilowych PL PL PL
CA2077638A1 (en) N-heteroaryl, n-alkylheteroaryl, n-alkenylheteroaryl and n- alkynylheteroarylmacrolides having immunosuppressive activity
CA2029860A1 (en) Aminomacrolides and derivatives having immuno-suppressive activity
CA2124260C (en) Tetrahydropyran derivatives
FI107536B (fi) Makrolidien fluorisokerijohdannaiset
HU211135A9 (en) Heteroatoms-containing tricyclic compounds
FI107537B (fi) Makrolidien 2-aminosokerijohdannaiset
EP2706061A1 (en) A chemo-enzymatic approach to the synthesis of pimecrolimus
FI107535B (fi) Makrolidien sokerijohdannaiset
US5210227A (en) Immunosuppressive compounds
US5359060A (en) Phosponated derivatives of macrolides
IE54283B1 (en) Omt ester derivatives
JPS6152839B2 (es)
CA2040551A1 (en) Deoxymacrolide derivatives having immunosuppressive activity
US6664243B1 (en) Benzyllactobionamides as inhibitors of smooth muscle cell proliferation
US20040092457A1 (en) Benzyllactobionamides as inhibitors of smooth muscle cell proliferation
US7132402B2 (en) Acylated benzylmaltosides as inhibitors of smooth muscle cell proliferation
JPH0559085A (ja) イミダゾール塩基を有するオキセタノシン誘導体
WO2000031092A2 (en) Benzyllactobionamides as inhibitors of smooth muscle cell proliferation