FI944015A - Makrolidien 2-aminosokerijohdannaiset - Google Patents

Makrolidien 2-aminosokerijohdannaiset Download PDF

Info

Publication number
FI944015A
FI944015A FI944015A FI944015A FI944015A FI 944015 A FI944015 A FI 944015A FI 944015 A FI944015 A FI 944015A FI 944015 A FI944015 A FI 944015A FI 944015 A FI944015 A FI 944015A
Authority
FI
Finland
Prior art keywords
pct
macrolides
amino sugar
sugar derivative
group
Prior art date
Application number
FI944015A
Other languages
English (en)
Swedish (sv)
Other versions
FI944015A0 (fi
FI107537B (fi
Inventor
Kevin Koch
Gary R Schulte
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of FI944015A publication Critical patent/FI944015A/fi
Publication of FI944015A0 publication Critical patent/FI944015A0/fi
Application granted granted Critical
Publication of FI107537B publication Critical patent/FI107537B/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/01Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing oxygen
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • A61P37/06Immunosuppressants, e.g. drugs for graft rejection

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Immunology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Transplantation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
FI944015A 1992-03-02 1994-09-01 Makrolidien 2-aminosokerijohdannaiset FI107537B (fi)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US84433992A 1992-03-02 1992-03-02
US84433992 1992-03-02
US9300427 1993-01-27
PCT/US1993/000427 WO1993018048A1 (en) 1992-03-02 1993-01-27 2-aminosugar derivatives of macrolides

Publications (3)

Publication Number Publication Date
FI944015A true FI944015A (fi) 1994-09-01
FI944015A0 FI944015A0 (fi) 1994-09-01
FI107537B FI107537B (fi) 2001-08-31

Family

ID=25292446

Family Applications (1)

Application Number Title Priority Date Filing Date
FI944015A FI107537B (fi) 1992-03-02 1994-09-01 Makrolidien 2-aminosokerijohdannaiset

Country Status (11)

Country Link
US (1) US5631235A (fi)
EP (1) EP0636136B1 (fi)
JP (1) JP2562001B2 (fi)
AT (1) ATE159725T1 (fi)
CA (1) CA2131373C (fi)
DE (1) DE69314947T2 (fi)
DK (1) DK0636136T3 (fi)
ES (1) ES2108261T3 (fi)
FI (1) FI107537B (fi)
GR (1) GR3025672T3 (fi)
WO (1) WO1993018048A1 (fi)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AUPP584198A0 (en) 1998-09-14 1998-10-08 Fujisawa Pharmaceutical Co., Ltd. New use
US7160867B2 (en) 2003-05-16 2007-01-09 Isotechnika, Inc. Rapamycin carbohydrate derivatives
CA2571710A1 (en) 2004-06-24 2006-11-02 Nicholas Valiante Small molecule immunopotentiators and assays for their detection

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4894366A (en) * 1984-12-03 1990-01-16 Fujisawa Pharmaceutical Company, Ltd. Tricyclo compounds, a process for their production and a pharmaceutical composition containing the same
AU6286690A (en) * 1989-08-18 1991-04-03 Fisons Plc Macrocyclic compounds
DK0427680T3 (da) * 1989-11-09 1995-12-18 Sandoz Ltd Heteroatom-holdige cykliske forbindelser
IE904050A1 (en) * 1989-11-13 1991-05-22 Merck & Co Inc Aminomacrolides and derivatives having immunosuppressive¹activity
EP0466365A3 (en) * 1990-07-03 1992-04-15 Merck & Co. Inc. Novel immunosuppressant fermentation products of a microorganism

Also Published As

Publication number Publication date
CA2131373C (en) 1999-01-26
WO1993018048A1 (en) 1993-09-16
DE69314947T2 (de) 1998-03-05
EP0636136B1 (en) 1997-10-29
JP2562001B2 (ja) 1996-12-11
EP0636136A1 (en) 1995-02-01
US5631235A (en) 1997-05-20
DK0636136T3 (da) 1997-12-22
FI944015A0 (fi) 1994-09-01
DE69314947D1 (de) 1997-12-04
GR3025672T3 (en) 1998-03-31
CA2131373A1 (en) 1993-09-16
FI107537B (fi) 2001-08-31
JPH07500350A (ja) 1995-01-12
ATE159725T1 (de) 1997-11-15
ES2108261T3 (es) 1997-12-16

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