DK0636136T3 - 2-aminosukkerderivater af makrolider - Google Patents

2-aminosukkerderivater af makrolider

Info

Publication number
DK0636136T3
DK0636136T3 DK93903554.9T DK93903554T DK0636136T3 DK 0636136 T3 DK0636136 T3 DK 0636136T3 DK 93903554 T DK93903554 T DK 93903554T DK 0636136 T3 DK0636136 T3 DK 0636136T3
Authority
DK
Denmark
Prior art keywords
pct
macrolides
sugar derivatives
amino sugar
group
Prior art date
Application number
DK93903554.9T
Other languages
Danish (da)
English (en)
Inventor
Gary R Schulte
Kevin Koch
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Application granted granted Critical
Publication of DK0636136T3 publication Critical patent/DK0636136T3/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/01Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing oxygen
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • A61P37/06Immunosuppressants, e.g. drugs for graft rejection

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Immunology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Transplantation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
DK93903554.9T 1992-03-02 1993-01-27 2-aminosukkerderivater af makrolider DK0636136T3 (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US84433992A 1992-03-02 1992-03-02

Publications (1)

Publication Number Publication Date
DK0636136T3 true DK0636136T3 (da) 1997-12-22

Family

ID=25292446

Family Applications (1)

Application Number Title Priority Date Filing Date
DK93903554.9T DK0636136T3 (da) 1992-03-02 1993-01-27 2-aminosukkerderivater af makrolider

Country Status (11)

Country Link
US (1) US5631235A (es)
EP (1) EP0636136B1 (es)
JP (1) JP2562001B2 (es)
AT (1) ATE159725T1 (es)
CA (1) CA2131373C (es)
DE (1) DE69314947T2 (es)
DK (1) DK0636136T3 (es)
ES (1) ES2108261T3 (es)
FI (1) FI107537B (es)
GR (1) GR3025672T3 (es)
WO (1) WO1993018048A1 (es)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AUPP584198A0 (en) 1998-09-14 1998-10-08 Fujisawa Pharmaceutical Co., Ltd. New use
US7160867B2 (en) 2003-05-16 2007-01-09 Isotechnika, Inc. Rapamycin carbohydrate derivatives
CA2571710A1 (en) 2004-06-24 2006-11-02 Nicholas Valiante Small molecule immunopotentiators and assays for their detection

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4894366A (en) * 1984-12-03 1990-01-16 Fujisawa Pharmaceutical Company, Ltd. Tricyclo compounds, a process for their production and a pharmaceutical composition containing the same
AU6286690A (en) * 1989-08-18 1991-04-03 Fisons Plc Macrocyclic compounds
DK0427680T3 (da) * 1989-11-09 1995-12-18 Sandoz Ltd Heteroatom-holdige cykliske forbindelser
IE904050A1 (en) * 1989-11-13 1991-05-22 Merck & Co Inc Aminomacrolides and derivatives having immunosuppressive¹activity
EP0466365A3 (en) * 1990-07-03 1992-04-15 Merck & Co. Inc. Novel immunosuppressant fermentation products of a microorganism

Also Published As

Publication number Publication date
CA2131373C (en) 1999-01-26
WO1993018048A1 (en) 1993-09-16
DE69314947T2 (de) 1998-03-05
FI944015A (fi) 1994-09-01
EP0636136B1 (en) 1997-10-29
JP2562001B2 (ja) 1996-12-11
EP0636136A1 (en) 1995-02-01
US5631235A (en) 1997-05-20
FI944015A0 (fi) 1994-09-01
DE69314947D1 (de) 1997-12-04
GR3025672T3 (en) 1998-03-31
CA2131373A1 (en) 1993-09-16
FI107537B (fi) 2001-08-31
JPH07500350A (ja) 1995-01-12
ATE159725T1 (de) 1997-11-15
ES2108261T3 (es) 1997-12-16

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